TAS3681, an androgen receptor antagonist, prevents drug resistance driven by aberrant androgen receptor signaling in prostate cancer
Yoshida, Shohei, Kajiwara, Daisuke, Seki, Masanao, Tayama, Manabu, Tanaka, Yuki, Mizutani, Hiroya, Fujita, Ryoto, Yamamura, Keisuke, Okajima, Shigeo, Asai, Masanori, Minamiguchi, Kazuhisa
Published in Molecular oncology (01.08.2024)
Published in Molecular oncology (01.08.2024)
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Journal Article
1,2-Silyl-Migrative Cyclization of Vinylsilanes Bearing a Hydroxy Group: Stereoselective Synthesis of Multisubstituted Tetrahydropyrans and Tetrahydrofurans1
Miura, Katsukiyo, Hondo, Takeshi, Okajima, Shigeo, Nakagawa, Takahiro, Takahashi, Tatsuyuki, Hosomi, Akira
Published in Journal of organic chemistry (23.08.2002)
Published in Journal of organic chemistry (23.08.2002)
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Journal Article
TAS 3681, an androgen receptor antagonist, prevents drug resistance driven by aberrant androgen receptor signaling in prostate cancer
Yoshida, Shohei, Kajiwara, Daisuke, Seki, Masanao, Tayama, Manabu, Tanaka, Yuki, Mizutani, Hiroya, Fujita, Ryoto, Yamamura, Keisuke, Okajima, Shigeo, Asai, Masanori, Minamiguchi, Kazuhisa
Published in Molecular oncology (01.08.2024)
Published in Molecular oncology (01.08.2024)
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Journal Article
Acid-Catalyzed Cyclization of Vinylsilanes Bearing a Hydroxy Group: A New Method for Stereoselective Synthesis of Disubstituted Tetrahydrofurans1
Miura, Katsukiyo, Okajima, Shigeo, Hondo, Takeshi, Nakagawa, Takahiro, Takahashi, Tatsuyuki, Hosomi, Akira
Published in Journal of the American Chemical Society (22.11.2000)
Published in Journal of the American Chemical Society (22.11.2000)
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The impact of TAS3681, a new type of androgen receptor antagonist, on aberrant AR signaling that drives tumor resistance to AR-targeted therapies by down-regulating full length and splice variant AR
Kajiwara, Daisuke, Minamiguchi, Kazuhisa, Seki, Masanao, Mizutani, Hiroya, Yamamura, Keisuke, Okajima, Shigeo, Sasaki, Eiji, Utsugi, Teruhiro, Iwasawa, Yoshikazu
Published in Journal of clinical oncology (20.02.2017)
Published in Journal of clinical oncology (20.02.2017)
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Silicon-directed cyclization of vinylsilanes bearing hydroxy group catalyzed by an acid
Miura, Katsukiyo, Okajima, Shigeo, Hondo, Takeshi, Hosomi, Akira
Published in Tetrahedron letters (27.02.1995)
Published in Tetrahedron letters (27.02.1995)
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Effect of a new type androgen receptor antagonist, TAS3681, on ligand-independent AR activation through its AR downregulation activity
Kajiwara, Daisuke, Minamiguchi, Kazuhisa, Seki, Masanao, Mizutani, Hiroya, Aoyagi, Hiroki, Okajima, Shigeo, Sasaki, Eiji, Utsugi, Teruhiro, Iwasawa, Yoshikazu
Published in Journal of clinical oncology (10.01.2016)
Published in Journal of clinical oncology (10.01.2016)
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Abstract PR09: TAS3681, a new type androgen receptor antagonist, suppresses ligand-independent AR activation through its AR downregulation activity
Kajiwara, Daisuke, Minamiguchi, Kazuhisa, Seki, Masanao, Mizutani, Hiroya, Aoyagi, Hiroki, Okajima, Shigeo, Sasaki, Eiji, Utsugi, Teruhiro, Iwasawa, Yoshikazu
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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TAS3681: New class of androgen receptor antagonist with androgen receptor downregulating activity
Minamiguchi, Kazuhisa, Seki, Masanao, Aoyagi, Hiroki, Kajiwara, Daisuke, Mori, Tomoko, Masuko, Norio, Fujita, Ryouto, Okajima, Shigeo, Hayashi, Yukio, Sasaki, Eiji, Utsugi, Teruhiro
Published in Journal of clinical oncology (01.03.2015)
Published in Journal of clinical oncology (01.03.2015)
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CONDENSED PYRIMIDINE COMPOUND OR SALT THEREOF
OGINO, Yoshio, ASAI, Takahiro, ASAI, Masanori, OKAJIMA, Shigeo, MINAMIGUCHI, Kazuhisa
Year of Publication 01.06.2017
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Year of Publication 01.06.2017
Patent
NOVEL TETRAHYDROPYRIDOPYRIMIDINE COMPOUND OR SALT THEREOF
ASAI TAKAHIRO, MINAMIGUCHI KAZUHISA, YAMANAKA HIROYOSHI, DOHI SUGURU, OKAJIMA SHIGEO, AOKI SHINICHI, ASAI MASANORI
Year of Publication 11.08.2016
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Year of Publication 11.08.2016
Patent
NOVEL TETRAHYDROPYRIDOPYRIMIDINE COMPOUND OR SALT THEREOF
OKAJIMA, SHIGEO, YAMANAKA, HIROYOSHI, ASAI, MASANORI, DOHI, SUGURU, ASAI, TAKAHIRO, MINAMIGUCHI, KAZUHISA, AOKI, SHINICHI
Year of Publication 03.12.2015
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Year of Publication 03.12.2015
Patent
1,2-silyl-migrative cyclization of vinylsilanes bearing a hydroxy group: Stereoselective synthesis of multisubstituted tetrahydropyrans and tetrahydrofurans
Miura, K, Hondo, T, Okajima, S, Nakagawa, T, Takahashi, T, Hosomi, A
Published in Journal of organic chemistry (23.08.2002)
Published in Journal of organic chemistry (23.08.2002)
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