Prolyl isomerase Pin1 plays an essential role in SARS-CoV-2 proliferation, indicating its possibility as a novel therapeutic target
Yamamotoya, Takeshi, Nakatsu, Yusuke, Kanna, Machi, Hasei, Shun, Ohata, Yukino, Encinas, Jeffrey, Ito, Hisanaka, Okabe, Takayoshi, Asano, Tomoichiro, Sakaguchi, Takemasa
Published in Scientific reports (17.09.2021)
Published in Scientific reports (17.09.2021)
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Oxysterol-Binding Protein Family I Is the Target of Minor Enviroxime-Like Compounds
Arita, Minetaro, Kojima, Hirotatsu, Nagano, Tetsuo, Okabe, Takayoshi, Wakita, Takaji, Shimizu, Hiroyuki
Published in Journal of Virology (01.04.2013)
Published in Journal of Virology (01.04.2013)
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Oxytocin/vasopressin-like peptide inotocin regulates cuticular hydrocarbon synthesis and water balancing in ants
Koto, Akiko, Motoyama, Naoto, Tahara, Hiroki, McGregor, Sean, Moriyama, Minoru, Okabe, Takayoshi, Miura, Masayuki, Keller, Laurent
Published in Proceedings of the National Academy of Sciences - PNAS (19.03.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (19.03.2019)
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Drug cytotoxicity screening using human intestinal organoids propagated with extensive cost-reduction strategies
Takahashi, Yu, Inoue, Yu, Sato, Shintaro, Okabe, Takayoshi, Kojima, Hirotatsu, Kiyono, Hiroshi, Shimizu, Makoto, Yamauchi, Yoshio, Sato, Ryuichiro
Published in Scientific reports (03.04.2023)
Published in Scientific reports (03.04.2023)
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Application of Acoustic Ejection MS System to High-Throughput Screening for SARS-CoV-2 3CL Protease Inhibitors
Hasegawa, Tsukasa, Imamura, Riyo M., Suzuki, Tateki, Hashiguchi, Takao, Nomura, Takao, Otsuguro, Satoko, Maenaka, Katsumi, Sasaki, Michihito, Orba, Yasuko, Sawa, Hirofumi, Sato, Akihiko, Okabe, Takayoshi, Nagano, Tetsuo, Kojima, Hirotatsu
Published in Chemical & pharmaceutical bulletin (01.03.2022)
Published in Chemical & pharmaceutical bulletin (01.03.2022)
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Inhibitors of the protein-protein interaction between phosphorylated p62 and Keap1 attenuate chemoresistance in a human hepatocellular carcinoma cell line
Yasuda, Daisuke, Ohe, Tomoyuki, Takahashi, Kyoko, Imamura, Riyo, Kojima, Hirotatsu, Okabe, Takayoshi, Ichimura, Yoshinobu, Komatsu, Masaaki, Yamamoto, Masayuki, Nagano, Tetsuo, Mashino, Tadahiko
Published in Free radical research (01.12.2020)
Published in Free radical research (01.12.2020)
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Dephospho-Coenzyme A Kinase Is an Exploitable Drug Target against Plasmodium falciparum: Identification of Selective Inhibitors by High-Throughput Screening of a Large Chemical Compound Library
Nurkanto, Arif, Imamura, Riyo, Rahmawati, Yulia, Prabandari, Erwahyuni Endang, Waluyo, Danang, Annoura, Takeshi, Yamamoto, Kazuki, Sekijima, Masakazu, Nishimura, Yuki, Okabe, Takayoshi, Shiba, Tomoo, Shibata, Norio, Kojima, Hirotatsu, Duffy, James, Nozaki, Tomoyoshi
Published in Antimicrobial agents and chemotherapy (15.11.2022)
Published in Antimicrobial agents and chemotherapy (15.11.2022)
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A novel diacylglycerol kinase α-selective inhibitor, CU-3, induces cancer cell apoptosis and enhances immune response[S]
Liu, Ke, Kunii, Naoko, Sakuma, Megumi, Yamaki, Atsumi, Mizuno, Satoru, Sato, Mayu, Sakai, Hiromichi, Kado, Sayaka, Kumagai, Kazuo, Kojima, Hirotatsu, Okabe, Takayoshi, Nagano, Tetsuo, Shirai, Yasuhito, Sakane, Fumio
Published in Journal of lipid research (01.03.2016)
Published in Journal of lipid research (01.03.2016)
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Discovery and Mechanistic Characterization of Selective Inhibitors of H2S-producing Enzyme: 3-Mercaptopyruvate Sulfurtransferase (3MST) Targeting Active-site Cysteine Persulfide
Hanaoka, Kenjiro, Sasakura, Kiyoshi, Suwanai, Yusuke, Toma-Fukai, Sachiko, Shimamoto, Kazuhito, Takano, Yoko, Shibuya, Norihiro, Terai, Takuya, Komatsu, Toru, Ueno, Tasuku, Ogasawara, Yuki, Tsuchiya, Yukihiro, Watanabe, Yasuo, Kimura, Hideo, Wang, Chao, Uchiyama, Masanobu, Kojima, Hirotatsu, Okabe, Takayoshi, Urano, Yasuteru, Shimizu, Toshiyuki, Nagano, Tetsuo
Published in Scientific reports (12.01.2017)
Published in Scientific reports (12.01.2017)
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Development of a Novel Intraocular-Pressure-Lowering Therapy Targeting ATX
Nagano, Norimichi, Honjo, Megumi, Kawaguchi, Mitsuyasu, Nishimasu, Hiroshi, Nureki, Osamu, Kano, Kuniyuki, Aoki, Junken, Komatsu, Toru, Okabe, Takayoshi, Kojima, Hirotatsu, Nagano, Tetsuo, Aihara, Makoto
Published in Biological & pharmaceutical bulletin (01.11.2019)
Published in Biological & pharmaceutical bulletin (01.11.2019)
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Development of Pin1 inhibitors and their potential as therapeutic agents
Nakatsu, Yusuke, Matsunaga, Yasuka, Ueda, Koji, Yamamotoya, Takeshi, Inoue, Yuki, Inoue, Masa-Ki, Mizuno, Yu, Kushiyama, Akifumi, Ono, Hiraku, Fujishiro, Midori, Ito, Hisanaka, Okabe, Takayoshi, Asano, Tomoichiro
Published in Current medicinal chemistry (01.01.2020)
Published in Current medicinal chemistry (01.01.2020)
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Discovery of a cystathionine γ-lyase (CSE) selective inhibitor targeting active-site pyridoxal 5′-phosphate (PLP) via Schiff base formation
Echizen, Honami, Hanaoka, Kenjiro, Shimamoto, Kazuhito, Hibi, Ryota, Toma-Fukai, Sachiko, Ohno, Hisashi, Sasaki, Eita, Komatsu, Toru, Ueno, Tasuku, Tsuchiya, Yukihiro, Watanabe, Yasuo, Otsuka, Takao, Saito, Hiroaki, Nagatoishi, Satoru, Tsumoto, Kouhei, Kojima, Hirotatsu, Okabe, Takayoshi, Shimizu, Toshiyuki, Urano, Yasuteru
Published in Scientific reports (30.09.2023)
Published in Scientific reports (30.09.2023)
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Molecular action of larvicidal flavonoids on ecdysteroidogenic glutathione S-transferase Noppera-bo in Aedes aegypti
Inaba, Kazue, Ebihara, Kana, Senda, Miki, Yoshino, Ryunosuke, Sakuma, Chisako, Koiwai, Kotaro, Takaya, Daisuke, Watanabe, Chiduru, Watanabe, Akira, Kawashima, Yusuke, Fukuzawa, Kaori, Imamura, Riyo, Kojima, Hirotatsu, Okabe, Takayoshi, Uemura, Nozomi, Kasai, Shinji, Kanuka, Hirotaka, Nishimura, Takashi, Watanabe, Kodai, Inoue, Hideshi, Fujikawa, Yuuta, Honma, Teruki, Hirokawa, Takatsugu, Senda, Toshiya, Niwa, Ryusuke
Published in BMC biology (17.02.2022)
Published in BMC biology (17.02.2022)
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Establishment of live-cell-based coupled assay system for identification of compounds to modulate metabolic activities of cells
Yanagi, Kouichi, Komatsu, Toru, Ogihara, Shusuke, Okabe, Takayoshi, Kojima, Hirotatsu, Nagano, Tetsuo, Ueno, Tasuku, Hanaoka, Kenjiro, Urano, Yasuteru
Published in Cell reports (Cambridge) (06.07.2021)
Published in Cell reports (Cambridge) (06.07.2021)
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Small-Molecule-Induced Activation of Cellular Respiration Inhibits Biofilm Formation and Triggers Metabolic Remodeling in Staphylococcus aureus
Okuda, Ken-ichi, Yamada-Ueno, Satomi, Yoshii, Yutaka, Nagano, Tetsuo, Okabe, Takayoshi, Kojima, Hirotatsu, Mizunoe, Yoshimitsu, Kinjo, Yuki
Published in mBio (30.08.2022)
Published in mBio (30.08.2022)
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Organoid-derived intestinal epithelial cells are a suitable model for preclinical toxicology and pharmacokinetic studies
Takahashi, Yu, Noguchi, Makoto, Inoue, Yu, Sato, Shintaro, Shimizu, Makoto, Kojima, Hirotatsu, Okabe, Takayoshi, Kiyono, Hiroshi, Yamauchi, Yoshio, Sato, Ryuichiro
Published in iScience (15.07.2022)
Published in iScience (15.07.2022)
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