Accelerating the discovery of alkyl halide-derived natural products using halide depletion
Glasser, Nathaniel R., Cui, Dongtao, Risser, Douglas D., Okafor, C. Denise, Balskus, Emily P.
Published in Nature chemistry (01.02.2024)
Published in Nature chemistry (01.02.2024)
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Journal Article
Inhibitors of ApiAP2 protein DNA binding exhibit multistage activity against Plasmodium parasites
Russell, Timothy James, De Silva, Erandi K, Crowley, Valerie M, Shaw-Saliba, Kathryn, Dube, Namita, Josling, Gabrielle, Pasaje, Charisse Flerida A, Kouskoumvekaki, Irene, Panagiotou, Gianni, Niles, Jacquin C, Jacobs-Lorena, Marcelo, Denise Okafor, C, Gamo, Francisco-Javier, Llinás, Manuel
Published in PLoS pathogens (01.10.2022)
Published in PLoS pathogens (01.10.2022)
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Journal Article
Two enhancer binding proteins activate σ54-dependent transcription of a quorum regulatory RNA in a bacterial symbiont
Surrett, Ericka D, Guckes, Kirsten R, Cousins, Shyan, Ruskoski, Terry B, Cecere, Andrew G, Ludvik, Denise A, Okafor, C Denise, Mandel, Mark J, Miyashiro, Tim I
Published in eLife (05.05.2023)
Published in eLife (05.05.2023)
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Journal Article
Structural basis for an unprecedented enzymatic alkylation in cylindrocyclophane biosynthesis
Braffman, Nathaniel R, Ruskoski, Terry B, Davis, Katherine M, Glasser, Nathaniel R, Johnson, Cassidy, Okafor, C Denise, Boal, Amie K, Balskus, Emily P
Published in eLife (25.02.2022)
Published in eLife (25.02.2022)
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Journal Article
How nuclear receptors transition between active and inactive forms: An energetic perspective
Hazarika, Saurov, Fehrle, Matthew, Okafor, C Denise
Published in The Journal of chemical physics (21.03.2024)
Published in The Journal of chemical physics (21.03.2024)
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Journal Article
Identification of an Evolutionarily Conserved Allosteric Network in Steroid Receptors
Dube, Namita, Khan, Sabab Hasan, Sasse, Riley, Okafor, C. Denise
Published in Journal of chemical information and modeling (23.01.2023)
Published in Journal of chemical information and modeling (23.01.2023)
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Journal Article
The nuclear receptor LRH-1 discriminates between ligands using distinct allosteric signaling circuits
Mays, Suzanne G, Hercules, David, Ortlund, Eric A, Okafor, C Denise
Published in Protein science (01.10.2023)
Published in Protein science (01.10.2023)
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Journal Article
Ancestral sequence reconstruction for evolutionary characterization of proteins
Dube, Namita, Khan, Sabab H., Okafor, C. Denise
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (01.01.2022)
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (01.01.2022)
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Journal Article
Structure and assembly of the diiron cofactor in the heme-oxygenase–like domain of the N-nitrosourea–producing enzyme SznF
McBride, Molly J., Pope, Sarah R., Hu, Kai, Okafor, C. Denise, Balskus, Emily P., Bollinger, J. Martin, Boal, Amie K.
Published in Proceedings of the National Academy of Sciences - PNAS (26.01.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (26.01.2021)
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Journal Article
Rewiring Ancient Residue Interaction Networks Drove the Evolution of Specificity in Steroid Receptors
Okafor, C. Denise, Hercules, David, Kell, Steven A., Ortlund, Eric A.
Published in Structure (London) (04.02.2020)
Published in Structure (London) (04.02.2020)
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Journal Article
Cutting in-line with iron: ribosomal function and non-oxidative RNA cleavage
Guth-Metzler, Rebecca, Bray, Marcus S, Frenkel-Pinter, Moran, Suttapitugsakul, Suttipong, Montllor-Albalate, Claudia, Bowman, Jessica C, Wu, Ronghu, Reddi, Amit R, Okafor, C Denise, Glass, Jennifer B, Williams, Loren Dean
Published in Nucleic acids research (04.09.2020)
Published in Nucleic acids research (04.09.2020)
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Journal Article
Allosteric regulation of thioesterase superfamily member 1 by lipid sensor domain binding fatty acids and lysophosphatidylcholine
Tillman, Matthew C., Imai, Norihiro, Li, Yue, Khadka, Manoj, Okafor, C. Denise, Juneja, Puneet, Adhiyaman, Akshitha, Hagen, Susan J., Cohen, David E., Ortlund, Eric A.
Published in Proceedings of the National Academy of Sciences - PNAS (08.09.2020)
Published in Proceedings of the National Academy of Sciences - PNAS (08.09.2020)
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Journal Article
Differential Modulation of Nuclear Receptor LRH‑1 through Targeting Buried and Surface Regions of the Binding Pocket
Cato, Michael L., Cornelison, Jeffery L., Spurlin, Racheal M., Courouble, Valentine V., Patel, Anamika B., Flynn, Autumn R., Johnson, Alyssa M., Okafor, C. Denise, Frank, Filipp, D’Agostino, Emma H., Griffin, Patrick R., Jui, Nathan T., Ortlund, Eric A.
Published in Journal of medicinal chemistry (12.05.2022)
Published in Journal of medicinal chemistry (12.05.2022)
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Journal Article
Development of the First Low Nanomolar Liver Receptor Homolog‑1 Agonist through Structure-guided Design
Mays, Suzanne G, Flynn, Autumn R, Cornelison, Jeffery L, Okafor, C. Denise, Wang, Hongtao, Wang, Guohui, Huang, Xiangsheng, Donaldson, Heather N, Millings, Elizabeth J, Polavarapu, Rohini, Moore, David D, Calvert, John W, Jui, Nathan T, Ortlund, Eric A
Published in Journal of medicinal chemistry (26.12.2019)
Published in Journal of medicinal chemistry (26.12.2019)
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