Synthesis and mechanism of action of novel pyrimidinyl pyrazole derivatives possessing antiproliferative activity
Ohki, Hitoshi, Hirotani, Kenji, Naito, Hiroyuki, Ohsuki, Satoru, Minami, Megumi, Ejima, Akio, Koiso, Yukiko, Hashimoto, Yuichi
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Get full text
Journal Article
Synthesis and antitumor activity of novel pyrimidinyl pyrazole derivatives. II. Optimization of the phenylpiperazine moiety of 1-[5-methyl-1-(2-pyrimidinyl)-4-pyrazolyl]-3-phenyl piperazinyl-1-trans-propanes
Naito, H, Ohsuki, S, Sugimori, M, Atsumi, R, Minami, M, Nakamura, Y, Ishii, M, Hirotani, K, Kumazawa, E, Ejima, A
Published in Chemical & pharmaceutical bulletin (01.04.2002)
Published in Chemical & pharmaceutical bulletin (01.04.2002)
Get full text
Journal Article
Synthesis and Antitumor Activity of Novel Pyrimidinyl Pyrazole Derivatives. III. Synthesis and Antitumor Activity of 3-Phenylpiperazinyl-1-trans-propenes
Naito, Hiroyuki, Ohsuki, Satoru, Atsumi, Ryo, Minami, Megumi, Mochizuki, Mineko, Hirotani, Kenji, Kumazawa, Eiji, Ejima, Akio
Published in Chemical & pharmaceutical bulletin (01.02.2005)
Published in Chemical & pharmaceutical bulletin (01.02.2005)
Get full text
Journal Article
A New Water‐soluble Camptothecin Derivative, DX‐8951f, Exhibits Potent Antitumor Activity against Human Tumors in vitro and in vivo
Mitsui, Ikuo, Kumazawa, Eiji, Hirota, Yasuhide, Aonuma, Masashi, Sugimori, Masamichi, Ohsuki, Satoru, Uoto, Kouichi, Ejima, Akio, Terasawa, Hirofumi, Sato, Keiki
Published in Cancer science (01.08.1995)
Published in Cancer science (01.08.1995)
Get full text
Journal Article
New highly active taxoids from 9β-dihydrobaccatin-9,10-acetals
ISHIYAMA, Takashi, LIMURA, Shin, OHSUKI, Satoru, UOTO, Kouichi, TERASAWA, Hirofumi, SOGA, Tsunehiko
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
Get full text
Journal Article
Synthesis and Structure-Activity Relationships of Novel 2', 2'-Difluoro Analogues of Docetaxel
UOTO, Kouichi, OHSUKI, Satoru, TAKENOSHITA, Haruhiro, ISHIYAMA, Takashi, IIMURA, Shin, HIROTA, Yasuhide, MITSUI, Ikuo, TERASAWA, Hirofumi, SOGA, Tsunehiko
Published in Chemical & pharmaceutical bulletin (01.11.1997)
Published in Chemical & pharmaceutical bulletin (01.11.1997)
Get full text
Journal Article
Synthesis and Antitumor Activity of Ring A- and F-Modified Hexacyclic Camptothecin Analogues
Sugimori, Masamichi, Ejima, Akio, Ohsuki, Satoru, Uoto, Kouichi, Mitsui, Ikuo, Kawato, Yasuyoshi, Hirota, Yasuhide, Sato, Keiki, Terasawa, Hirofumi
Published in Journal of medicinal chemistry (18.06.1998)
Published in Journal of medicinal chemistry (18.06.1998)
Get full text
Journal Article
Orally active docetaxel analogue: Synthesis of 10-deoxy-10-C-morpholinoethyl docetaxel analogues
LIMURA, Shin, UOTO, Kouichi, OHSUKI, Satoru, CHIBA, Jun, YOSHINO, Toshiharu, IWAHANA, Michio, JIMBO, Takeshi, TERASAWA, Hirofumi, SOGA, Tsunehiko
Published in Bioorganic & medicinal chemistry letters (12.02.2001)
Published in Bioorganic & medicinal chemistry letters (12.02.2001)
Get full text
Journal Article
ANTITUMOR AGENTS .7. SYNTHESIS AND ANTITUMOR-ACTIVITY OF NOVEL HEXACYCLIC CAMPTOTHECIN ANALOGS
SUGIMORI, M, EJIMA, A, OHSUKI, S, UOTO, K, MITSUI, MATSUMOTO, K, KAWATO, Y, YASUOKA, M, SATO, K, TAGAWA, H, TERASAWA, H
Published in Journal of medicinal chemistry (16.09.1994)
Published in Journal of medicinal chemistry (16.09.1994)
Get full text
Journal Article
Synthesis and antitumor activity of non-prodrug water-soluble taxoid: 10-C-aminoalkylated docetaxel analogs
Iimura, S, Ohsuki, S, Chiba, J, Uoto, K, Iwahana, M, Terasawa, H, Soga, T
Published in Heterocycles (01.12.2000)
Published in Heterocycles (01.12.2000)
Get more information
Journal Article
A convenient method for the synthesis of C-10 alkylated docetaxel analogs using tris-(trimethylsilyl)silane as a radical mediator
Iimura, S, Ohsuki, S, Uoto, K, Nakayama, K, Terasawa, H, Soga, T
Published in Heterocycles (01.07.2000)
Published in Heterocycles (01.07.2000)
Get more information
Journal Article
ANTITUMOR AGENTS .6. SYNTHESIS AND ANTITUMOR-ACTIVITY OF RING A-MODIFIED, RING B-MODIFIED, AND RING C-MODIFIED DERIVATIVES OF CAMPTOTHECIN
SUGIMORI, M, EJIMA, A, OHSUKI, S, MATSUMOTO, K, KAWATO, Y, YASUOKA, M, TAGAWA, H, TERASAWA, H
Published in Heterocycles (01.01.1994)
Get more information
Published in Heterocycles (01.01.1994)
Journal Article
Novel bicycloannulation via tandem vinylation and intramolecular Diels-Alder reaction of five-membered heterocycles: a new approach to contruction of psoralen and azapsoralen
HAYAKAWA, K, YODO, M, OHSUKI, S, KANEMATSU, K
Published in Journal of the American Chemical Society (1984)
Get full text
Published in Journal of the American Chemical Society (1984)
Journal Article
Antitumor Agents. V. Synthesis and Antileukemic Activity of E-Ring-Modified (RS)-Camptothecin Analogues
EJIMA, Akio, TERASAWA, Hirofumi, SUGIMORI, Masamichi, OHSUKI, Satoru, MATSUMOTO, Kensuke, KAWATO, Yasuyoshi, YASUOKA, Megumi, TAGAWA, Hiroaki
Published in Chemical & pharmaceutical bulletin (01.03.1992)
Published in Chemical & pharmaceutical bulletin (01.03.1992)
Get full text
Journal Article
A new water-soluble camptothecin derivative, DX-9851f, exhibits potent antitumor activity against human tumors in vitro and in vivo
MITSUI, I, KUMAZAWA, E, HIROTA, Y, AONUMA, M, SUGIMORI, M, OHSUKI, S, UOTO, K, EJIMA, A, TERASAWA, H, SATO, K
Published in Japanese journal of cancer research (Gann) (1995)
Get full text
Published in Japanese journal of cancer research (Gann) (1995)
Journal Article
Pyrazolopyrimidine derivative
OHSUKI SATORU, NAGATA CHIKAHIRO, TENGEIJI ATSUSHI, SHIBATA YOSHIHIRO, IKEDA MASAHIRO, SHIMADA TAKASHI
Year of Publication 09.07.2014
Get full text
Year of Publication 09.07.2014
Patent