Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure−Activity Relationships of 2-Piperazin-1-yl-1H-benzimidazoles
Ognyanov, Vassil I, Balan, Chenera, Bannon, Anthony W, Bo, Yunxin, Dominguez, Celia, Fotsch, Christopher, Gore, Vijay K, Klionsky, Lana, Ma, Vu V, Qian, Yi-Xin, Tamir, Rami, Wang, Xianghong, Xi, Ning, Xu, Shimin, Zhu, Dawn, Gavva, Narender R, Treanor, James J. S, Norman, Mark H
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
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Novel Vanilloid Receptor-1 Antagonists: 2. Structure−Activity Relationships of 4-Oxopyrimidines Leading to the Selection of a Clinical Candidate
Doherty, Elizabeth M, Fotsch, Christopher, Bannon, Anthony W, Bo, Yunxin, Chen, Ning, Dominguez, Celia, Falsey, James, Gavva, Narender R, Katon, Jodie, Nixey, Thomas, Ognyanov, Vassil I, Pettus, Liping, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Zhu, Jiawang, Treanor, James J. S, Norman, Mark H
Published in Journal of medicinal chemistry (26.07.2007)
Published in Journal of medicinal chemistry (26.07.2007)
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Preparation of chiral cyanohydrins by an oxynitrilase-mediated transcyanation
Ognyanov, Vassil I, Datcheva, Violeta K, Kyler, Keith S
Published in Journal of the American Chemical Society (01.08.1991)
Published in Journal of the American Chemical Society (01.08.1991)
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Discovery of Potent, Orally Available Vanilloid Receptor-1 Antagonists. Structure−Activity Relationship of N-Aryl Cinnamides
Doherty, Elizabeth M, Fotsch, Christopher, Bo, Yunxin, Chakrabarti, Partha P, Chen, Ning, Gavva, Narender, Han, Nianhe, Kelly, Michael G, Kincaid, John, Klionsky, Lana, Liu, Qingyian, Ognyanov, Vassil I, Tamir, Rami, Wang, Xianghong, Zhu, Jiawang, Norman, Mark H, Treanor, James J. S
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
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Novel Vanilloid Receptor-1 Antagonists: 1. Conformationally Restricted Analogues of trans-Cinnamides
Norman, Mark H, Zhu, Jiawang, Fotsch, Christopher, Bo, Yunxin, Chen, Ning, Chakrabarti, Partha, Doherty, Elizabeth M, Gavva, Narender R, Nishimura, Nobuko, Nixey, Thomas, Ognyanov, Vassil I, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Viswanadhan, Vellarkad N, Treanor, James J. S
Published in Journal of medicinal chemistry (26.07.2007)
Published in Journal of medicinal chemistry (26.07.2007)
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Trisubstituted pyrimidines as transient receptor potential vanilloid 1 (TRPV1) antagonists with improved solubility
Wang, Xianghong, Chakrabarti, Partha P., Ognyanov, Vassil I., Pettus, Liping H., Tamir, Rami, Tan, Helming, Tang, Phi, Treanor, James J.S., Gavva, Narender R., Norman, Mark H.
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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Deoxygenated inositol 1,4,5-trisphosphate analogs and their interaction with metabolic enzymes. (1R,2R,4R)-Cyclohexane-1,2,4-tris(methylenesulfonate): a potent selective 5-phosphatase inhibitor
Kozikowski, Alan P, Ognyanov, Vassil I, Chen, Chinpiao, Fauq, Abdul H, Safrany, Stephen T, Wilcox, Robert A, Nahorski, Stefan R
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
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1D-myo-inositol 1,4,5-trisphosphate and 1D-myo-inositol 1,3,4,5-tetrakisphosphate analogues modified at C-3; synthesis of 1D-3-C-(trifluoromethyl)-myo-inositol 1,4,5-trisphosphate and 1L-chiro-insitol 1,2,3,5-tetrakisphosphate from L-quebrachitol
Kozikowski, Alan P., Ognyanov, Vassil I., Fauq, Abdul H., Wilcox, Robert A., Nahorski, Stefan R.
Published in Journal of the Chemical Society. Chemical communications (1994)
Published in Journal of the Chemical Society. Chemical communications (1994)
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Journal Article
Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure−Activity Relationships of 2-Piperazin-1-yl-1 H -benzimidazoles
Ognyanov, Vassil I., Balan, Chenera, Bannon, Anthony W., Bo, Yunxin, Dominguez, Celia, Fotsch, Christopher, Gore, Vijay K., Klionsky, Lana, Ma, Vu V., Qian, Yi-Xin, Tamir, Rami, Wang, Xianghong, Xi, Ning, Xu, Shimin, Zhu, Dawn, Gavva, Narender R., Treanor, James J. S., Norman, Mark H.
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Probing the D-1,4,5-IP3/D-1,3,4,5-IP4 functional interface. Synthesis and pharmacology of novel D-3-modified myo-inositol trisphosphate analogues
FAUQ, A. H, KOZIKOWSKI, A. P, OGNYANOV, V. I, WILCOX, R. A, NAHORSKI, S. R
Published in Journal of the Chemical Society. Chemical communications (1994)
Published in Journal of the Chemical Society. Chemical communications (1994)
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Glycine transport inhibitors: A new class of antipsychotics?
Borden, Laurence A., Bell, Stanley C., Ognyanov, Vassil I., Albert, Vivian R., Zhang, Jing, De Vivo, Michael, Yokoyama, Midori, Xie, Xiaping, Berger, Theodore, Gerhardt, Greg, McKelvy, Jeffrey F.
Published in Schizophrenia research (1997)
Published in Schizophrenia research (1997)
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