Discovery and preclinical characterization of [18F]PI-2620, a next-generation tau PET tracer for the assessment of tau pathology in Alzheimer’s disease and other tauopathies
Kroth, Heiko, Oden, Felix, Molette, Jerome, Schieferstein, Hanno, Capotosti, Francesca, Mueller, Andre, Berndt, Mathias, Schmitt-Willich, Heribert, Darmency, Vincent, Gabellieri, Emanuele, Boudou, Cédric, Juergens, Tanja, Varisco, Yvan, Vokali, Efthymia, Hickman, David T., Tamagnan, Gilles, Pfeifer, Andrea, Dinkelborg, Ludger, Muhs, Andreas, Stephens, Andrew
Published in European journal of nuclear medicine and molecular imaging (01.09.2019)
Published in European journal of nuclear medicine and molecular imaging (01.09.2019)
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Potent anti-tumor response by targeting B cell maturation antigen (BCMA) in a mouse model of multiple myeloma
Oden, Felix, Marino, Stephen F., Brand, Janko, Scheu, Susanne, Kriegel, Cathleen, Olal, Daniel, Takvorian, Anna, Westermann, Jörg, Yilmaz, Buket, Hinz, Michael, Daumke, Oliver, Höpken, Uta E., Müller, Gerd, Lipp, Martin
Published in Molecular oncology (01.08.2015)
Published in Molecular oncology (01.08.2015)
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PRECLINICAL CHARACTERIZATION OF PI-2620, A NOVEL TAU PET TRACER FOR DETECTION OF TAU IN AD AND OTHER TAUOPATHIES
Mueller, Andre, Kroth, Heiko, Schieferstein, Hanno, Berndt, Mathias, Oden, Felix, Capotosti, Francesca, Molette, Jerome, Juergens, Tanja, Darmency, Vincent, Schmitt-Willich, Heribert, Hickman, David, Tamagnan, Gilles, Pfeifer, Andrea, Dinkelborg, Ludger, Muhs, Andreas, Stephens, Andrew
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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Structure-activity relationship around PI-2620 highlights the importance of the nitrogen atom position in the tricyclic core
Kroth, Heiko, Oden, Felix, Serra, Andreia Monica, Molette, Jerome, Mueller, Andre, Berndt, Mathias, Capotosti, Francesca, Gabellieri, Emanuele, Schmitt-Willich, Heribert, Hickman, David, Pfeifer, Andrea, Dinkelborg, Ludger, Stephens, Andrew
Published in Bioorganic & medicinal chemistry (15.12.2021)
Published in Bioorganic & medicinal chemistry (15.12.2021)
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Journal Article
PI-2620 Lead Optimization Highlights the Importance of Off-Target Assays to Develop a PET Tracer for the Detection of Pathological Aggregated Tau in Alzheimer’s Disease and Other Tauopathies
Kroth, Heiko, Oden, Felix, Molette, Jerome, Schieferstein, Hanno, Gabellieri, Emanuele, Mueller, Andre, Berndt, Mathias, Sreenivasachary, Nampally, Serra, Andreia Monica, Capotosti, Francesca, Schmitt-Willich, Heribert, Hickman, David, Pfeifer, Andrea, Dinkelborg, Ludger, Stephens, Andrew
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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CAR T Cells with Enhanced Sensitivity to B Cell Maturation Antigen for the Targeting of B Cell Non-Hodgkin’s Lymphoma and Multiple Myeloma
Bluhm, Julia, Kieback, Elisa, Marino, Stephen F., Oden, Felix, Westermann, Jörg, Chmielewski, Markus, Abken, Hinrich, Uckert, Wolfgang, Höpken, Uta E., Rehm, Armin
Published in Molecular therapy (01.08.2018)
Published in Molecular therapy (01.08.2018)
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Discovery of 2-(4-(2-fluoroethoxy)piperidin-1-yl)-9-methyl-9H-pyrrolo[2,3-b:4,5-c’]dipyridine ([18F]PI-2014) as PET tracer for the detection of pathological aggregated tau in Alzheimer’s disease and other tauopathies
Gabellieri, Emanuele, Capotosti, Francesca, Molette, Jerome, Sreenivasachary, Nampally, Mueller, Andre, Berndt, Mathias, Schieferstein, Hanno, Juergens, Tanja, Varisco, Yvan, Oden, Felix, Schmitt-Willich, Heribert, Hickman, David, Dinkelborg, Ludger, Stephens, Andrew, Pfeifer, Andrea, Kroth, Heiko
Published in European journal of medicinal chemistry (15.10.2020)
Published in European journal of medicinal chemistry (15.10.2020)
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Development of self-reactive germinal center B cells and plasma cells in autoimmune FcγRIIB-deficient mice
Tiller, Thomas, Kofer, Juliane, Kreschel, Cornelia, Busse, Christian E., Riebel, Stefan, Wickert, Susanne, Oden, Felix, Mertes, Maria M.M., Ehlers, Marc, Wardemann, Hedda
Published in The Journal of experimental medicine (22.11.2010)
Published in The Journal of experimental medicine (22.11.2010)
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Abstract 1141: Preclinical analysis of biodistribution and PET imaging of a zirconium-89 labeled PSMA-targeted antibody-chelator conjugate
Hammer, Stefanie, Zitzmann-Kolbe, Sabine, Oden, Felix, Jannsen, Joerg, Bickel, Eva, Mueller, Andre, Everz, Lothar, Hagemann, Urs B., Karlsson, Jenny, Ryan, Olav B., Hennekes, Hartwig, Cole, Patricia E., Mumberg, Dominik
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Discovery and preclinical characterization of 18FPI-2620, a next-generation tau PET tracer for the assessment of tau pathology in Alzheimer's disease and other tauopathies
Kroth, Heiko, Oden, Felix, Molette, Jerome, Schieferstein, Hanno, Capotosti, Francesca, Mueller, Andre, Berndt, Mathias, Schmitt-Willich, Heribert, Darmency, Vincent, Gabellieri, Emanuele, Boudou, Cédric, Juergens, Tanja, Varisco, Yvan, Vokali, Efthymia, Hickman, David T, Tamagnan, Gilles, Pfeifer, Andrea, Dinkelborg, Ludger, Muhs, Andreas, Stephens, Andrew
Published in European journal of nuclear medicine and molecular imaging (01.09.2019)
Published in European journal of nuclear medicine and molecular imaging (01.09.2019)
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Journal Article
sup 18^F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in The Journal of nuclear medicine (1978) (01.07.2017)
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Published in The Journal of nuclear medicine (1978) (01.07.2017)
Journal Article
18 F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in Journal of Nuclear Medicine (01.07.2017)
Published in Journal of Nuclear Medicine (01.07.2017)
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Journal Article
Characterization of the novel PET Tracer PI-2620 for the assessment of Tau pathology in Alzheimer’s disease and other tauopathies
Mueller, Andre, Kroth, Heiko, Berndt, Mathias, Capotosti, Francesca, Molette, Jerome, Schieferstein, Hanno, Oden, Felix, Juergens, Tanja, Darmency, Vincent, Schmitt-Willich, Heribert, Hickman, David, Tamagnan, Gilles, Pfeifer, Andrea, Dinkelborg, Ludger, Stephens, Andrew, Muhs, Andreas
Published in The Journal of nuclear medicine (1978) (01.05.2017)
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Published in The Journal of nuclear medicine (1978) (01.05.2017)
Journal Article
PRECLINICAL CHARACTERIZATION OF PI-2620, A NOVEL TAU PET TRACER FOR DETECTION OF TAU IN AD AND OTHER TAUOPATHIES
Mueller, Andre, Kroth, Heiko, Schieferstein, Hanno, Berndt, Mathias, Oden, Felix, Capotosti, Francesca, Molette, Jerome, Juergens, Tanja, Darmency, Vincent, Schmitt-Willich, Heribert, Hickman, David, Tamagnan, Gilles, Pfeifer, Andrea, Dinkelborg, Ludger, Muhs, Andreas, Stephens, Andrew
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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타우 단백질 응집체를 이미징하기 위한 화합물
SCHIEFERSTEIN HANNO, ODEN FELIX, GABELLIERI EMANUELE, SCHMITT WILLICH HERIBERT, BERNDT MATHIAS, MOLETTE JEROME, MULLER ANDRE, KROTH HEIKO, DARMENCY VINCENT
Year of Publication 25.03.2019
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Year of Publication 25.03.2019
Patent
18F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in The Journal of nuclear medicine (1978) (01.07.2017)
Published in The Journal of nuclear medicine (1978) (01.07.2017)
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Journal Article