Selective targeting of the stress chaperome as a therapeutic strategy
Taldone, Tony, Ochiana, Stefan O, Patel, Pallav D, Chiosis, Gabriela
Published in Trends in pharmacological sciences (Regular ed.) (01.11.2014)
Published in Trends in pharmacological sciences (Regular ed.) (01.11.2014)
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Heat shock protein 90 inhibitors in the treatment of cancer: current status and future directions
Jhaveri, Komal, Ochiana, Stefan O, Dunphy, Mark Ps, Gerecitano, John F, Corben, Adriana D, Peter, Radu I, Janjigian, Yelena Y, Gomes-DaGama, Erica M, Koren, 3rd, John, Modi, Shanu, Chiosis, Gabriela
Published in Expert opinion on investigational drugs (01.05.2014)
Published in Expert opinion on investigational drugs (01.05.2014)
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Journal Article
Ligand deconstruction: Why some fragment binding positions are conserved and others are not
Kozakov, Dima, Hall, David R., Jehle, Stefan, Luo, Lingqi, Ochiana, Stefan O., Jones, Elizabeth V., Pollastri, Michael, Allen, Karen N., Whitty, Adrian, Vajda, Sandor
Published in Proceedings of the National Academy of Sciences - PNAS (19.05.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (19.05.2015)
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A Hyperactive Signalosome in Acute Myeloid Leukemia Drives Addiction to a Tumor-Specific Hsp90 Species
Zong, Hongliang, Gozman, Alexander, Caldas-Lopes, Eloisi, Taldone, Tony, Sturgill, Eric, Brennan, Sarah, Ochiana, Stefan O., Gomes-DaGama, Erica M., Sen, Siddhartha, Rodina, Anna, Koren, John, Becker, Michael W., Rudin, Charles M., Melnick, Ari, Levine, Ross L., Roboz, Gail J., Nimer, Stephen D., Chiosis, Gabriela, Guzman, Monica L.
Published in Cell reports (Cambridge) (15.12.2015)
Published in Cell reports (Cambridge) (15.12.2015)
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Chemical tools for epichaperome-mediated interactome dysfunctions of the central nervous system
Bolaender, Alexander, Zatorska, Danuta, He, Huazhong, Joshi, Suhasini, Sharma, Sahil, Digwal, Chander S., Patel, Hardik J., Sun, Weilin, Imber, Brandon S., Ochiana, Stefan O., Patel, Maulik R., Shrestha, Liza, Shah, Smit. K., Wang, Shuo, Karimov, Rashad, Tao, Hui, Patel, Pallav D., Martin, Ananda Rodilla, Yan, Pengrong, Panchal, Palak, Almodovar, Justina, Corben, Adriana, Rimner, Andreas, Ginsberg, Stephen D., Lyashchenko, Serge, Burnazi, Eva, Ku, Anson, Kalidindi, Teja, Lee, Sang Gyu, Grkovski, Milan, Beattie, Bradley J., Zanzonico, Pat, Lewis, Jason S., Larson, Steve, Rodina, Anna, Pillarsetty, Nagavarakishore, Tabar, Viviane, Dunphy, Mark P., Taldone, Tony, Shimizu, Fumiko, Chiosis, Gabriela
Published in Nature communications (03.08.2021)
Published in Nature communications (03.08.2021)
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Journal Article
Affinity Purification Probes of Potential Use To Investigate the Endogenous Hsp70 Interactome in Cancer
Rodina, Anna, Taldone, Tony, Kang, Yanlong, Patel, Pallav D, Koren, John, Yan, Pengrong, DaGama Gomes, Erica M, Yang, Chenghua, Patel, Maulik R, Shrestha, Liza, Ochiana, Stefan O, Santarossa, Cristina, Maharaj, Ronnie, Gozman, Alexander, Cox, Marc B, Erdjument-Bromage, Hediye, Hendrickson, Ronald C, Cerchietti, Leandro, Melnick, Ari, Guzman, Monica L, Chiosis, Gabriela
Published in ACS chemical biology (15.08.2014)
Published in ACS chemical biology (15.08.2014)
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Journal Article
Structure–Activity Relationship in a Purine-Scaffold Compound Series with Selectivity for the Endoplasmic Reticulum Hsp90 Paralog Grp94
Patel, Hardik J, Patel, Pallav D, Ochiana, Stefan O, Yan, Pengrong, Sun, Weilin, Patel, Maulik R, Shah, Smit K, Tramentozzi, Elisa, Brooks, James, Bolaender, Alexander, Shrestha, Liza, Stephani, Ralph, Finotti, Paola, Leifer, Cynthia, Li, Zihai, Gewirth, Daniel T, Taldone, Tony, Chiosis, Gabriela
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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Journal Article
First-in-Human Trial of Epichaperome-Targeted PET in Patients with Cancer
Dunphy, Mark P S, Pressl, Christina, Pillarsetty, Nagavarakishore, Grkovski, Milan, Modi, Shanu, Jhaveri, Komal, Norton, Larry, Beattie, Bradley J, Zanzonico, Pat B, Zatorska, Danuta, Taldone, Tony, Ochiana, Stefan O, Uddin, Mohammad M, Burnazi, Eva M, Lyashchenko, Serge K, Hudis, Clifford A, Bromberg, Jacqueline, Schöder, Heiko M, Fox, Josef J, Zhang, Hanwen, Chiosis, Gabriela, Lewis, Jason S, Larson, Steven M
Published in Clinical cancer research (01.10.2020)
Published in Clinical cancer research (01.10.2020)
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Journal Article
The human Aurora kinase inhibitor danusertib is a lead compound for anti-trypanosomal drug discovery via target repurposing
Ochiana, Stefan O., Pandarinath, Vidya, Wang, Zhouxi, Kapoor, Rishika, Ondrechen, Mary Jo, Ruben, Larry, Pollastri, Michael P.
Published in European journal of medicinal chemistry (01.04.2013)
Published in European journal of medicinal chemistry (01.04.2013)
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Journal Article
Tumor-specific HSP90 inhibition as a therapeutic approach in JAK-mutant acute lymphoblastic leukemias
Kucine, Nicole, Marubayashi, Sachie, Bhagwat, Neha, Papalexi, Efthymia, Koppikar, Priya, Sanchez Martin, Marta, Dong, Lauren, Tallman, Marty S., Paietta, Elisabeth, Wang, Kai, He, Jie, Lipson, Doron, Stephens, Phil, Miller, Vince, Rowe, Jacob M., Teruya-Feldstein, Julie, Mullighan, Charles G., Ferrando, Adolfo A., Krivtsov, Andrei, Armstrong, Scott, Leung, Laura, Ochiana, Stefan O., Chiosis, Gabriela, Levine, Ross L., Kleppe, Maria
Published in Blood (26.11.2015)
Published in Blood (26.11.2015)
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Journal Article
Pharmacological Validation of Trypanosoma brucei Phosphodiesterases B1 and B2 as Druggable Targets for African Sleeping Sickness
Bland, Nicholas D, Wang, Cuihua, Tallman, Craig, Gustafson, Alden E, Wang, Zhouxi, Ashton, Trent D, Ochiana, Stefan O, McAllister, Gregory, Cotter, Kristina, Fang, Anna P, Gechijian, Lara, Garceau, Norman, Gangurde, Rajiv, Ortenberg, Ron, Ondrechen, Mary Jo, Campbell, Robert K, Pollastri, Michael P
Published in Journal of medicinal chemistry (08.12.2011)
Published in Journal of medicinal chemistry (08.12.2011)
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Journal Article
Repurposing Human PDE4 Inhibitors for Neglected Tropical Diseases. Evaluation of Analogs of the Human PDE4 Inhibitor GSK-256066 as Inhibitors of PDEB1 of Trypanosoma brucei
Ochiana, Stefan O., Bland, Nicholas D., Settimo, Luca, Campbell, Robert K., Pollastri, Michael P.
Published in Chemical biology & drug design (01.05.2015)
Published in Chemical biology & drug design (01.05.2015)
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Journal Article
Synthesis and evaluation of human phosphodiesterases (PDE) 5 inhibitor analogs as trypanosomal PDE inhibitors. Part 1. Sildenafil analogs
Wang, Cuihua, Ashton, Trent D., Gustafson, Alden, Bland, Nicholas D., Ochiana, Stefan O., Campbell, Robert K., Pollastri, Michael P.
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Synthesis and evaluation of human phosphodiesterases (PDE) 5 inhibitor analogs as trypanosomal PDE inhibitors. Part 2. Tadalafil analogs
Ochiana, Stefan O., Gustafson, Alden, Bland, Nicholas D., Wang, Cuihua, Russo, Michael J., Campbell, Robert K., Pollastri, Michael P.
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Synthesis and assessment of catechol diether compounds as inhibitors of trypanosomal phosphodiesterase B1 (TbrPDEB1)
Woodring, Jennifer L., Bland, Nicholas D., Ochiana, Stefan O., Campbell, Robert K., Pollastri, Michael P.
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
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Journal Article
Radiosynthesis of the iodine-124 labeled Hsp90 inhibitor PU-H71
Taldone, Tony, Zatorska, Danuta, Ochiana, Stefan O., Smith-Jones, Peter, Koziorowski, Jacek, Dunphy, Mark P., Zanzonico, Pat, Bolaender, Alexander, Lewis, Jason S., Larson, Steven M., Chiosis, Gabriela, Pillarsetty, Naga Vara Kishore
Published in Journal of labelled compounds & radiopharmaceuticals (01.03.2016)
Published in Journal of labelled compounds & radiopharmaceuticals (01.03.2016)
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METHODS AND REAGENTS FOR RADIOLABELING
PILLARSETTY NAGAVARAKISHORE, CHIOSIS GABRIELA, TALDONE TONY, OCHIANA STEFAN O
Year of Publication 24.08.2016
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Year of Publication 24.08.2016
Patent
SELECTIVE GRP94 INHIBITORS AND USES THEREOF
PATEL PALLAV, CHIOSIS GABRIELA, YANG CHENGHUA, TALDONE TONY, OCHIANA STEFAN O, SUN WEILIN, YAN PENGRONG, PATEL HARDIK J
Year of Publication 21.04.2016
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Year of Publication 21.04.2016
Patent
First-in-Human Trial of Epichaperome-Targeted Positron Emission Tomography in Cancer Patients
Dunphy, Mark P., Pressl, Christina, Pillarsetty, Nagavarakishore, Grkovski, Milan, Modi, Shanu, Jhaveri, Komal, Norton, Larry, Beattie, Bradley J., Zanzonico, Pat B., Zatorska, Danuta, Taldone, Tony, Ochiana, Stefan O., Uddin, Mohammad M., Burnazi, Eva M., Lyashchenko, Serge K., Hudis, Clifford A., Bromberg, Jacqueline F., Schöder, Heiko M., Fox, Josef J., Zhang, Hanwen, Chiosis, Gabriela, Lewis, Jason S., Larson, Steven M.
Published in Clinical cancer research (04.05.2020)
Published in Clinical cancer research (04.05.2020)
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Journal Article
Correction: Ligand deconstruction: Why some fragment binding positions are conserved and others are not
Published in Proceedings of the National Academy of Sciences - PNAS
(14.07.2015)
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