Partition coefficient and diffusion coefficient determinations of 50 compounds in human intact skin, isolated skin layers and isolated stratum corneum lipids
Ellison, Corie A., Tankersley, Kevin O., Obringer, Cindy M., Carr, Greg J., Manwaring, John, Rothe, Helga, Duplan, Hélène, Géniès, Camille, Grégoire, Sébastien, Hewitt, Nicola J., Jamin, Carine Jacques, Klaric, Martina, Lange, Daniela, Rolaki, Alexandra, Schepky, Andreas
Published in Toxicology in vitro (01.12.2020)
Published in Toxicology in vitro (01.12.2020)
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Corrigendum to partition coefficient and diffusion coefficient determinations of 50 compounds in human intact skin, isolated skin layers and isolated stratum corneum lipids
Ellison, Corie A., Tankersley, Kevin O., Obringer, Cindy M., Carr, Greg J., Manwaring, John, Rothe, Helga, Duplan, Hélène, Géniès, Camille, Grégoire, Sébastien, Hewitt, Nicola J., Jamin, Carine Jacques, Klaric, Martina, Lange, Daniela, Rolaki, Alexandra, Schepky, Andreas
Published in Toxicology in vitro (01.03.2021)
Published in Toxicology in vitro (01.03.2021)
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Design, Synthesis, and Evaluation of Proline and Pyrrolidine Based Melanocortin Receptor Agonists. A Conformationally Restricted Dipeptide Mimic Approach
Tian, Xinrong, Field, Timothy B, Switzer, Adrian G, Mazur, Adam W, Ebetino, Frank H, Wos, John A, Berberich, Steve M, Jayasinghe, Lalith R, Obringer, Cindy M, Dowty, Martin E, Pinney, Beth B, Farmer, Julie A, Crossdoersen, Doreen, Sheldon, Russell J
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Discovery of Orally Bioavailable 1,3,4-Trisubstituted 2-Oxopiperazine-Based Melanocortin-4 Receptor Agonists as Potential Antiobesity Agents
Tian, Xinrong, Switzer, Adrian G, Derose, Steve A, Mishra, Rajesh K, Solinsky, Mark G, Mumin, Rashid N, Ebetino, Frank H, Jayasinghe, Lalith R, Webster, Mark E, Colson, Anny-Odile, Crossdoersen, Doreen, Pinney, Beth B, Farmer, Julie A, Dowty, Martin E, Obringer, Cindy M, Cruze, Charles A, Burklow, Melissa L, Suchanek, Paula M, Dong, Lily, Dirr, Mary Kay, Sheldon, Russell J, Wos, John A
Published in Journal of medicinal chemistry (09.10.2008)
Published in Journal of medicinal chemistry (09.10.2008)
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Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonists
Meyers, Kenneth M., Méndez-Andino, José, Colson, Anny-Odile, Hu, X. Eric, Wos, John A., Mitchell, Maria C., Hodge, Karen, Howard, Jeremy, Paris, Jennifer L., Dowty, Martin E., Obringer, Cindy M., Reizes, Ofer
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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The efficacy and cardiac evaluation of aminomethyl tetrahydronaphthalene ketopiperazines: A novel class of potent MCH-R1 antagonists
Méndez-Andino, José L., Colson, Anny-Odile, Meyers, Kenneth M., Mitchell, Maria C., Hodge, Karen, Howard, Jeremy M., Kim, Nicholas, Ackley, David C., Holbert, Jerry K., Mittelstadt, Scott W., Dowty, Martin E., Obringer, Cindy M., Suchanek, Paula, Reizes, Ofer, Eric Hu, X., Wos, John A.
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Aminomethyl tetrahydronaphthalene ketopiperazine MCH-R1 antagonists—Increasing selectivity over hERG
Meyers, Kenneth M., Méndez-Andino, José L., Colson, Anny-Odile, Warshakoon, Namal C., Wos, John A., Mitchell, Maria C., Hodge, Karen M., Howard, Jeremy M., Ackley, David C., Holbert, Jerry K., Mittelstadt, Scott W., Dowty, Martin E., Obringer, Cindy M., Reizes, Ofer, Hu, X. Eric
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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