Generation of an LFA-1 Antagonist by the Transfer of the ICAM-1 Immunoregulatory Epitope to a Small Molecule
Gadek, T. R., Burdick, D. J., McDowell, R. S., Stanley, M. S., Marsters, J. C., Paris, K. J., Oare, D. A., Reynolds, M. E., Ladner, C., Zioncheck, K. A., Lee, W. P., Gribling, P., Dennis, M. S., Skelton, N. J., Tumas, D. B., Clark, K. R., Keating, S. M., Beresini, M. H., Tilley, J. W., Presta, L. G., Bodary, S. C.
Published in Science (American Association for the Advancement of Science) (08.02.2002)
Published in Science (American Association for the Advancement of Science) (08.02.2002)
Get full text
Journal Article
Benzodiazepine peptidomimetic inhibitors of farnesyltransferase
Marsters, James C., McDowell, Robert S., Reynolds, Mark E., Oare, David A., Somers, Todd C., Stanley, Mark S., Rawson, Thomas E., Struble, Martin E., Burdick, Daniel J., Chan, Kathryn S., Duarte, Charles M., Paris, Kenneth J., Tom, Jeff Y.K., Wan, Dairian T., Xue, Yingchun, Bumier, John P.
Published in Bioorganic & medicinal chemistry (01.09.1994)
Published in Bioorganic & medicinal chemistry (01.09.1994)
Get full text
Journal Article
Acyclic stereoselection. 46. Stereochemistry of the Michael addition of N,N-disubstituted amide and thioamide enolates to .alpha.,.beta.-unsaturated ketones
Oare, David A, Henderson, Mark A, Sanner, Mark A, Heathcock, Clayton H
Published in Journal of organic chemistry (01.01.1990)
Published in Journal of organic chemistry (01.01.1990)
Get full text
Journal Article
Acyclic stereoselection. 30. Stereoselection in the Michael addition reaction. 2. Stereochemistry of the kinetic Michael reaction of amide enolates with enones
Heathcock, Clayton H, Henderson, Mark A, Oare, David A, Sanner, Mark A
Published in Journal of organic chemistry (01.08.1985)
Published in Journal of organic chemistry (01.08.1985)
Get full text
Journal Article