Discovery of (1R,2S)‑2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)‑N‑(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Receptor Antagonist
Yoshida, Yu, Naoe, Yoshimitsu, Terauchi, Taro, Ozaki, Fumihiro, Doko, Takashi, Takemura, Ayumi, Tanaka, Toshiaki, Sorimachi, Keiichi, Beuckmann, Carsten T, Suzuki, Michiyuki, Ueno, Takashi, Ozaki, Shunsuke, Yonaga, Masahiro
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Piperidine Carboxylic Acid Derivatives of 10H-Pyrazino[2,3-b][1,4]benzothiazine as Orally-Active Adhesion Molecule Inhibitors
Kaneko, Toshihiko, Clark, Richard S. J., Ohi, Norihito, Ozaki, Fumihiro, Kawahara, Tetsuya, Kamada, Atsushi, Okano, Kazuo, Yokohama, Hiromitsu, Ohkuro, Masayoshi, Muramoto, Kenzo, Takenaka, Osamu, Kobayashi, Seiichi
Published in Chemical & Pharmaceutical Bulletin (01.06.2004)
Published in Chemical & Pharmaceutical Bulletin (01.06.2004)
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Inhibitors of Adhesion Molecules Expression; The Synthesis and Pharmacological Properties of 10H-Pyrazino[2,3-b][1,4]benzothiazine Derivatives
Kaneko, Toshihiko, Clark, Richard S. J., Ohi, Norihito, Kawahara, Tetsuya, Akamatsu, Hiroshi, Ozaki, Fumihiro, Kamada, Atsushi, Okano, Kazuo, Yokohama, Hiromitsu, Muramoto, Kenzo, Ohkuro, Masayoshi, Takenaka, Osamu, Kobayashi, Seiichi
Published in Chemical & pharmaceutical bulletin (01.07.2002)
Published in Chemical & pharmaceutical bulletin (01.07.2002)
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Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists
Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists” [Bioorg. Med. Chem. 22 (2014) 6071–6088]
Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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COMPOSITION FOR CLEANING INSIDE ORAL CAVITY
KODAMA YUSHI, MAEDA YUUICHI, MORITA DAIKI, DOI TOSHIHIRO, OYAIZU MASANORI, OZAKI FUMIHIRO
Year of Publication 09.12.2015
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Year of Publication 09.12.2015
Patent
COMPOSITION FOR CLEANING INSIDE ORAL CAVITY
MAEDA YUICHI, MORITA TAIKI, KODAMA YUJI, DOI TOSHIHIRO, OYAIZU MASANORI, OZAKI FUMIHIRO
Year of Publication 16.10.2014
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Year of Publication 16.10.2014
Patent
COMPOSITION FOR CLEANING INSIDE ORAL CAVITY
OYAIZU, MASANORI, DOI, TOSHIHIRO, MORITA, DAIKI, MAEDA, YUUICHI, KODAMA, YUSHI, OZAKI, FUMIHIRO
Year of Publication 02.10.2014
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Year of Publication 02.10.2014
Patent