Emerging Approaches for the Identification of Protein Targets of Small Molecules - A Practitioners’ Perspective
Comess, Kenneth M, McLoughlin, Shaun M, Oyer, Jon A, Richardson, Paul L, Stöckmann, Henning, Vasudevan, Anil, Warder, Scott E
Published in Journal of medicinal chemistry (11.10.2018)
Published in Journal of medicinal chemistry (11.10.2018)
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A Mutation in Histone H2B Represents a New Class of Oncogenic Driver
Bennett, Richard L, Bele, Aditya, Small, Eliza C, Will, Christine M, Nabet, Behnam, Oyer, Jon A, Huang, Xiaoxiao, Ghosh, Rajarshi P, Grzybowski, Adrian T, Yu, Tao, Zhang, Qiao, Riva, Alberto, Lele, Tanmay P, Schatz, George C, Kelleher, Neil L, Ruthenburg, Alexander J, Liphardt, Jan, Licht, Jonathan D
Published in Cancer discovery (01.10.2019)
Published in Cancer discovery (01.10.2019)
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An activating mutation of the NSD2 histone methyltransferase drives oncogenic reprogramming in acute lymphocytic leukemia
Swaroop, Alok, Oyer, Jon A., Will, Christine M., Huang, Xiaoxiao, Yu, Wenbo, Troche, Catalina, Bulic, Marinka, Durham, Benjamin H., Wen, Qiang Jeremy, Crispino, John D., MacKerell, Alexander D., Bennett, Richard L., Kelleher, Neil L., Licht, Jonathan D.
Published in Oncogene (01.01.2019)
Published in Oncogene (01.01.2019)
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C-terminal domain small phosphatase 1 and MAP kinase reciprocally control REST stability and neuronal differentiation
Nesti, Edmund, Corson, Glen M, McCleskey, Maxwell, Oyer, Jon A, Mandel, Gail
Published in Proceedings of the National Academy of Sciences - PNAS (16.09.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (16.09.2014)
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Journal Article
PRC2 Inhibitors Overcome Glucocorticoid Resistance Driven by NSD2 Mutation in Pediatric Acute Lymphoblastic Leukemia
Li, Jianping, Hlavka-Zhang, Julia, Shrimp, Jonathan H, Piper, Crissandra, Dupéré-Richér, Daphne, Roth, Jacob S, Jing, Duohui, Casellas Román, Heidi L, Troche, Catalina, Swaroop, Alok, Kulis, Marta, Oyer, Jon A, Will, Christine M, Shen, Min, Riva, Alberto, Bennett, Richard L, Ferrando, Adolfo A, Hall, Matthew D, Lock, Richard B, Licht, Jonathan D
Published in Cancer discovery (01.01.2022)
Published in Cancer discovery (01.01.2022)
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Polycomb- and REST-associated histone deacetylases are independent pathways toward a mature neuronal phenotype
McGann, James C, Oyer, Jon A, Garg, Saurabh, Yao, Huilan, Liu, Jun, Feng, Xin, Liao, Lujian, Yates, 3rd, John R, Mandel, Gail
Published in eLife (24.09.2014)
Published in eLife (24.09.2014)
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Cardiovascular and Systemic MicrovascularEffects of Anti-Vascular Endothelial Growth Factor Therapy for Cancer
Belcik, J. Todd, BS, RDCS, Qi, Yue, MD, Kaufmann, Beat A., MD, Xie, Aris, BS, Bullens, Sherry, BA, Morgan, Terry K., MD, PhD, Bagby, Susan P., MD, Kolumam, Ganesh, PhD, Kowalski, Joe, BS, Oyer, Jon A., PhD, Bunting, Stuart, PhD, Lindner, Jonathan R., MD
Published in Journal of the American College of Cardiology (14.08.2012)
Published in Journal of the American College of Cardiology (14.08.2012)
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Cardiovascular and Systemic Microvascular Effects of Anti-Vascular Endothelial Growth Factor Therapy for Cancer
BELCIK, J. Todd, YUE QI, BUNTING, Stuart, LINDNER, Jonathan R, KAUFMANN, Beat A, XIE, Aris, BULLENS, Sherry, MORGAN, Terry K, BAGBY, Susan P, KOLUMAM, Ganesh, KOWALSKI, Joe, OYER, Jon A
Published in Journal of the American College of Cardiology (14.08.2012)
Published in Journal of the American College of Cardiology (14.08.2012)
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Abstract 330: Engineering electrophile-sensitive kinase mutants to accelerate oncology target validation
Oyer, Jon A., Johnson, Ted W., Wang, Andrew C., Maestre, Michael F., Flores-Bojorquez, Ana, Melnychuk, Roksolana, Timofeevski, Sergei, Niessen, Sherry, Wang, Zhenxiong, Li, Jian, Diehl, Wade C., Eisele, Koleen J., Lee, Nathan V., Zou, Aihua, Davis, Carl, Greenwald, Eric C., DeForest, Jacob, Ornelas, Martha, Li, Bryan, Scales, Stephanie, Khamphavong, Penney L., Ambler, Catherine M., Huang, Yun, Salomon-Ferrer, Romelia, Greasley, Samantha E., Bolanos, Ben, Grodsky, Neil, Lum, Lawrence, VanArsdale, Todd L., McAlpine, Indrawan J.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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