Splicing factor SF3b as a target of the antitumor natural product pladienolide
Mizui, Yoshiharu, Kotake, Yoshihiko, Sagane, Koji, Owa, Takashi, Mimori-Kiyosue, Yuko, Shimizu, Hajime, Uesugi, Mai, Ishihama, Yasushi, Iwata, Masao
Published in Nature chemical biology (01.09.2007)
Published in Nature chemical biology (01.09.2007)
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Anticancer and Antiviral Sulfonamides
SCOZZAFAVA, Andrea, OWA, Takashi, MASTROLORENZO, Antonio, SUPURAN, Claudiu T
Published in Current medicinal chemistry (01.06.2003)
Published in Current medicinal chemistry (01.06.2003)
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A landmark in drug discovery based on complex natural product synthesis
Kawano, Satoshi, Ito, Ken, Yahata, Kenzo, Kira, Kazunobu, Abe, Takanori, Akagi, Tsuyoshi, Asano, Makoto, Iso, Kentaro, Sato, Yuki, Matsuura, Fumiyoshi, Ohashi, Isao, Matsumoto, Yasunobu, Isomura, Minetaka, Sasaki, Takeo, Fukuyama, Takashi, Miyashita, Yusuke, Kaburagi, Yosuke, Yokoi, Akira, Asano, Osamu, Owa, Takashi, Kishi, Yoshito
Published in Scientific reports (17.06.2019)
Published in Scientific reports (17.06.2019)
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Enhancement of Soft Tissue Sarcoma Response to Gemcitabine through Timed Administration of a Short-Acting Anti-Angiogenic Agent
Cheng, Jin, Fuller, John, Feldman, Regina, Tap, William, Owa, Takashi, Fuks, Zvi, Kolesnick, Richard
Published in Cellular physiology and biochemistry (29.07.2020)
Published in Cellular physiology and biochemistry (29.07.2020)
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Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX
Abbate, Francesco, Casini, Angela, Owa, Takashi, Scozzafava, Andrea, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
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A molecular glue RBM39-degrader induces synthetic lethality in cancer cells with homologous recombination repair deficiency
Kohsaka, Shinji, Yagishita, Shigehiro, Shirai, Yukina, Matsuno, Yusuke, Ueno, Toshihide, Kojima, Shinya, Ikeuchi, Hiroshi, Ikegami, Masachika, Kitada, Rina, Yoshioka, Ken-ichi, Toshimitsu, Kohta, Tabata, Kimiyo, Yokoi, Akira, Doi, Toshihiko, Yamamoto, Noboru, Owa, Takashi, Hamada, Akinobu, Mano, Hiroyuki
Published in NPJ precision oncology (24.05.2024)
Published in NPJ precision oncology (24.05.2024)
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Quantitative Chemical Proteomics for Identifying Candidate Drug Targets
Oda, Yoshiya, Owa, Takashi, Sato, Toshitaka, Boucher, Brian, Daniels, Scott, Yamanaka, Hidenori, Shinohara, Yasuhiro, Yokoi, Akira, Kuromitsu, Junro, Nagasu, Takeshi
Published in Analytical chemistry (Washington) (01.05.2003)
Published in Analytical chemistry (Washington) (01.05.2003)
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Discovery of Novel Antitumor Sulfonamides Targeting G1 Phase of the Cell Cycle
Owa, Takashi, Yoshino, Hiroshi, Okauchi, Tatsuo, Yoshimatsu, Kentaro, Ozawa, Yoichi, Sugi, Naoko Hata, Nagasu, Takeshi, Koyanagi, Nozomu, Kitoh, Kyosuke
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
A Role for Histone Deacetylase Activity in HDAC1-Mediated Transcriptional Repression
Hassig, Christian A., Tong, Jeffrey K., Fleischer, Tracey C., Owa, Takashi, Grable, Phyllis G., Ayer, Donald E., Schreiber, Stuart L.
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.1998)
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Journal Article
Depudecin Induces Morphological Reversion of Transformed Fibroblasts via the Inhibition of Histone Deacetylase
Kwon, Ho Jeong, Owa, Takashi, Hassig, Christian A., Shimada, Junichi, Schreiber, Stuart L.
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (31.03.1998)
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Journal Article
Profiling Novel Sulfonamide Antitumor Agents with Cell-based Phenotypic Screens and Array-based Gene Expression Analysis
Yokoi, Akira, Kuromitsu, Junro, Kawai, Takatoshi, Nagasu, Takeshi, Sugi, Naoko Hata, Yoshimatsu, Kentaro, Yoshino, Hiroshi, Owa, Takashi
Published in Molecular cancer therapeutics (01.02.2002)
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Published in Molecular cancer therapeutics (01.02.2002)
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Microarray-based transcriptional profiling of renieramycin M and jorunnamycin C, isolated from Thai marine organisms
Charupant, Kornvika, Suwanborirux, Khanit, Daikuhara, Naomi, Yokoya, Masashi, Ushijima-Sugano, Rie, Kawai, Takatoshi, Owa, Takashi, Saito, Naoki
Published in Marine drugs (19.10.2009)
Published in Marine drugs (19.10.2009)
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Journal Article
Selective degradation of splicing factor CAPERα by anticancer sulfonamides
Uehara, Taisuke, Minoshima, Yukinori, Sagane, Koji, Sugi, Naoko Hata, Mitsuhashi, Kaoru Ogawa, Yamamoto, Noboru, Kamiyama, Hiroshi, Takahashi, Kentaro, Kotake, Yoshihiko, Uesugi, Mai, Yokoi, Akira, Inoue, Atsushi, Yoshida, Taku, Mabuchi, Miyuki, Tanaka, Akito, Owa, Takashi
Published in Nature chemical biology (01.06.2017)
Published in Nature chemical biology (01.06.2017)
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Journal Article
Tazemetostat, an EZH2 inhibitor, in relapsed or refractory B-cell non-Hodgkin lymphoma and advanced solid tumours: a first-in-human, open-label, phase 1 study
Italiano, Antoine, Soria, Jean-Charles, Toulmonde, Maud, Michot, Jean-Marie, Lucchesi, Carlo, Varga, Andrea, Coindre, Jean-Michel, Blakemore, Stephen J, Clawson, Alicia, Suttle, Benjamin, McDonald, Alice A, Woodruff, Mark, Ribich, Scott, Hedrick, Eric, Keilhack, Heike, Thomson, Blythe, Owa, Takashi, Copeland, Robert A, Ho, Peter T C, Ribrag, Vincent
Published in The lancet oncology (01.05.2018)
Published in The lancet oncology (01.05.2018)
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A focused compound library of novel N-(7-indolyl)benzenesulfonamides for the discovery of potent cell cycle inhibitors
OWA, T, OKAUCHI, T, YOSHIMATSU, K, SUGI, N. H, OZAWA, Y, NAGASU, T, KOYANAGI, N, OKABE, T, KITOH, K, YOSHINO, H
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
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Final results of a phase 2, open‐label study of indisulam, idarubicin, and cytarabine in patients with relapsed or refractory acute myeloid leukemia and high‐risk myelodysplastic syndrome
Assi, Rita, Kantarjian, Hagop M., Kadia, Tapan M., Pemmaraju, Naveen, Jabbour, Elias, Jain, Nitin, Daver, Naval, Estrov, Zeev, Uehara, Taisuke, Owa, Takashi, Cortes, Jorge E., Borthakur, Gautam
Published in Cancer (01.07.2018)
Published in Cancer (01.07.2018)
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NF-κB suppression synergizes with E7386, an inhibitor of CBP/β-catenin interaction, to block proliferation of patient-derived colon cancer spheroids
Kanda, Yusuke, Ohata, Hirokazu, Miyazaki, Toshiaki, Sakai, Hiroaki, Mori, Yutaro, Shiokawa, Daisuke, Yokoi, Akira, Owa, Takashi, Ochiai, Atsushi, Okamoto, Koji
Published in Biochemical and biophysical research communications (01.01.2022)
Published in Biochemical and biophysical research communications (01.01.2022)
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