Structure−Activity Relationship for Thiohydantoin Androgen Receptor Antagonists for Castration-Resistant Prostate Cancer (CRPC)
Jung, Michael E, Ouk, Samedy, Yoo, Dongwon, Sawyers, Charles L, Chen, Charlie, Tran, Chris, Wongvipat, John
Published in Journal of medicinal chemistry (08.04.2010)
Published in Journal of medicinal chemistry (08.04.2010)
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Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer
Tran, Chris, Ouk, Samedy, Clegg, Nicola J, Chen, Yu, Watson, Philip A, Arora, Vivek, Wongvipat, John, Smith-Jones, Peter M, Yoo, Dongwon, Kwon, Andrew, Wasielewska, Teresa, Welsbie, Derek, Chen, Charlie Degui, Higano, Celestia S, Beer, Tomasz M, Hung, David T, Scher, Howard I, Jung, Michael E, Sawyers, Charles L
Published in Science (American Association for the Advancement of Science) (08.05.2009)
Published in Science (American Association for the Advancement of Science) (08.05.2009)
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Targeting metabolism and survival in chronic lymphocytic leukemia and Richter syndrome cells by a novel NF-κB inhibitor
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Published in Haematologica (Roma) (01.11.2017)
Published in Haematologica (Roma) (01.11.2017)
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ARN-509: A Novel Antiandrogen for Prostate Cancer Treatment
CLEGG, Nicola J, WONGVIPAT, John, APARICIO, Anna, DOROW, Steven, ARORA, Vivek, GANG SHAO, JING QIAN, HONG ZHAO, GUANGBIN YANG, CHUNYAN CAO, SENSINTAFFAR, John, WASIELEWSKA, Teresa, JOSEPH, James D, HERBERT, Mark R, BONNEFOUS, Celine, DARIMONT, Beatrice, SCHER, Howard I, SMITH-JONES, Peter, KLANG, Mark, SMITH, Nicholas D, DE STANCHINA, Elisa, NIAN WU, OUERFELLI, Ouathek, TRAN, Chris, RIX, Peter J, HEYMAN, Richard A, JUNG, Michael E, SAWYERS, Charles L, HAGER, Jeffrey H, OUK, Samedy, DILHAS, Anna, YU CHEN, GRILLOT, Kate, BISCHOFF, Eric D, LING CAI
Published in Cancer research (Chicago, Ill.) (15.03.2012)
Published in Cancer research (Chicago, Ill.) (15.03.2012)
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Targeted Nanotherapy of Hematologic Malignancies Using Gold Nanoframework-Based Delivery of a Novel NF-Kb Inhibitor
Bariana, Manpreet, Zhang, Beilu, Sun, Jingyu, Cassella, Elena, Rateshwar, Janice, Tan, Ming Tony, Wang, Weiwei, Wang, Jinping, Feinman, Rena, Siegel, David, Liou, Hsiou-Chi, Ouk, Samedy, Mondello, Patrizia, Wang, Hongjun, Zakrzewski, Johannes
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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Targeted Lymphoma Therapy Using a Gold Nanoframework-Based Drug Delivery System
Bariana, Manpreet, Zhang, Beilu, Sun, Jingyu, Wang, Weiwei, Wang, Jinping, Cassella, Elena, Myint, Faith, Anuncio, Shaina A., Ouk, Samedy, Liou, Hsiou-Chi, Tan, Ming, Wang, Hongjun, Zakrzewski, Johannes L.
Published in ACS applied materials & interfaces (08.02.2023)
Published in ACS applied materials & interfaces (08.02.2023)
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Inhibition of NF-κB DNA Binding Suppresses Myeloma Growth via Intracellular Redox and Tumor Microenvironment Modulation
Bariana, Manpreet, Cassella, Elena, Rateshwar, Janice, Ouk, Samedy, Liou, Hsiou-Chi, Heller, Claudia, Colorado, Iriana, Feinman, Rena, Makhdoom, Ali, Siegel, David S, Heller, Glenn, Tuckett, Andrea, Mondello, Patrizia, Zakrzewski, Johannes L
Published in Molecular cancer therapeutics (02.12.2022)
Published in Molecular cancer therapeutics (02.12.2022)
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Characterization of a c-Rel Inhibitor That Mediates Anticancer Properties in Hematologic Malignancies by Blocking NF-κB-Controlled Oxidative Stress Responses
Shono, Yusuke, Tuckett, Andrea Z, Liou, Hsiou-Chi, Doubrovina, Ekaterina, Derenzini, Enrico, Ouk, Samedy, Tsai, Jennifer J, Smith, Odette M, Levy, Emily R, Kreines, Fabiana M, Ziegler, Carly G K, Scallion, Mary I, Doubrovin, Mikhail, Heller, Glenn, Younes, Anas, O'Reilly, Richard J, van den Brink, Marcel R M, Zakrzewski, Johannes L
Published in Cancer research (Chicago, Ill.) (15.01.2016)
Published in Cancer research (Chicago, Ill.) (15.01.2016)
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DIARYLHYDANTOIN COMPOUNDS
YOO DONGWON, WONGVIPAT JOHN, SAWYERS CHARLES L, WELSBIE DEREK, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E, CHEN CHARLIE D
Year of Publication 05.01.2023
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Year of Publication 05.01.2023
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Targeting Cellular Metabolism and Survival in Chronic Lymphocytic Leukemia and Richter Syndrome Cells By a Novel NF-Kb Inhibitor
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Published in Blood (02.12.2016)
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A small-molecule c-Rel inhibitor reduces alloactivation of T cells without compromising antitumor activity
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Published in Cancer discovery (01.05.2014)
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ANDROGEN RECEPTOR MODULATOR FOR TREATMENT OF PROSTATE CANCER AND ANDROGEN RECEPTOR-ASSOCIATED DISEASES
WONGVIPAT JOHN, SAWYERS CHARLES L, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E
Year of Publication 03.12.2020
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Year of Publication 03.12.2020
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DIARYLHYDANTOIN COMPOUNDS
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Year of Publication 04.03.2021
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Year of Publication 04.03.2021
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Targeted Therapy of B Cell Lymphoma with a Direct Inhibitor of the NF-κB Subunit c-Rel
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Published in Blood (06.12.2014)
Published in Blood (06.12.2014)
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ANDROGEN RECEPTOR MODULATOR FOR TREATMENT OF PROSTATE CANCER AND ANDROGEN RECEPTOR-ASSOCIATED DISEASES
WONGVIPAT JOHN, SAWYERS CHARLES L, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E
Year of Publication 30.05.2019
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Year of Publication 30.05.2019
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DIARYLHYDANTOIN COMPOUNDS
YOO DONGWON, WONGVIPAT JOHN, SAWYERS CHARLES L, WELSBIE DEREK, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E, CHEN CHARLIE D
Year of Publication 26.12.2019
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Year of Publication 26.12.2019
Patent
DIARYLHYDANTOIN COMPOUNDS
YOO DONGWON, WONGVIPAT JOHN, SAWYERS CHARLES L, WELSBIE DEREK, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E, CHEN CHARLIE D
Year of Publication 06.09.2019
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Year of Publication 06.09.2019
Patent
ANDROGEN RECEPTOR MODULATOR FOR TREATMENT OF PROSTATE CANCER AND ANDROGEN RECEPTOR-ASSOCIATED DISEASES
WONGVIPAT JOHN, SAWYERS CHARLES L, OUK SAMEDY, TRAN CHRIS, JUNG MICHAEL E
Year of Publication 26.04.2018
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Year of Publication 26.04.2018
Patent