Synthesis of the Methyl Analog of 2′‑O,4′‑C‑Ethylene-Bridged 5‑Methyluridine via Intramolecular Radical Cyclization and Properties of Modified Oligonucleotides
Ito, Yuta, Tsutsui, Norika, Osawa, Takashi, Hari, Yoshiyuki
Published in Journal of organic chemistry (19.07.2019)
Published in Journal of organic chemistry (19.07.2019)
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Journal Article
Synthesis, Duplex-Forming Ability, and Nuclease Resistance of Oligonucleotides Containing a Thymidine Derivative with a 1-Oxaspiro[4.5]decane Skeleton
Osawa, Takashi, Yano, Natsumi, Aoyama, Hiroshi, Obika, Satoshi
Published in Chemical & pharmaceutical bulletin (01.10.2022)
Published in Chemical & pharmaceutical bulletin (01.10.2022)
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Journal Article
New Cleavable Spacers for Tandem Synthesis of Multiple Oligo-nucleotides
Yamamoto, Kazuki, Fuchi, Yasufumi, Okabe, Masaya, Osawa, Takashi, Ito, Yuta, Hari, Yoshiyuki
Published in Synthesis (Stuttgart) (01.12.2021)
Published in Synthesis (Stuttgart) (01.12.2021)
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Journal Article
Synthesis and Properties of 2′‑O,4′‑C‑Ethyleneoxy Bridged 5‑Methyluridine
Hari, Yoshiyuki, Morikawa, Tomohiko, Osawa, Takashi, Obika, Satoshi
Published in Organic letters (19.07.2013)
Published in Organic letters (19.07.2013)
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Journal Article
Post-synthetic modification of oligonucleotides containing 5-trifluoromethylpyrimidine bases
Ito, Yuta, Matsuo, Misaki, Yamamoto, Kazuki, Yamashita, Wakana, Osawa, Takashi, Hari, Yoshiyuki
Published in Tetrahedron (22.11.2018)
Published in Tetrahedron (22.11.2018)
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Journal Article
Synthesis of Oligonucleotides Containing 2'- N -alkylaminocarbonyl-2'-amino-LNA (2'-urea-LNA) Moieties Using Post-Synthetic Modification Strategy
Yamashita, Shoko, Nishida, Kodai, Osawa, Takashi, Nakanishi, Ayumi, Ito, Yuta, Hari, Yoshiyuki
Published in Molecules (Basel, Switzerland) (15.01.2020)
Published in Molecules (Basel, Switzerland) (15.01.2020)
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Journal Article
Synthesis of 2′‑C,4′‑C‑Methyleneoxy-Bridged Thymidine Derivatives and Properties of Modified Oligonucleotides
Osawa, Takashi, Kim, Han, Shoji, Misa, Saijo, Miku, Dohi, Masakazu, Ito, Yuta, Obika, Satoshi, Hari, Yoshiyuki
Published in Journal of organic chemistry (01.11.2019)
Published in Journal of organic chemistry (01.11.2019)
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Journal Article
Synthesis of Sugar and Nucleoside Analogs and Evaluation of Their Anticancer and Analgesic Potentials
Hussain, Fahad, Rahman, Fahad Imtiaz, Saha, Poushali, Mikami, Atsushi, Osawa, Takashi, Obika, Satoshi, Rahman, S M Abdur
Published in Molecules (Basel, Switzerland) (29.05.2022)
Published in Molecules (Basel, Switzerland) (29.05.2022)
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Journal Article
Amido-Bridged Nucleic Acids (AmNAs): Synthesis, Duplex Stability, Nuclease Resistance, and in Vitro Antisense Potency
Yahara, Aiko, Shrestha, Ajaya Ram, Yamamoto, Tsuyoshi, Hari, Yoshiyuki, Osawa, Takashi, Yamaguchi, Masaki, Nishida, Masaru, Kodama, Tetsuya, Obika, Satoshi
Published in Chembiochem : a European journal of chemical biology (26.11.2012)
Published in Chembiochem : a European journal of chemical biology (26.11.2012)
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Journal Article
Synthesis, duplex-forming ability, enzymatic stability, and in vitro antisense potency of oligonucleotides including 2'-C,4'-C-ethyleneoxy-bridged thymidine derivatives
Osawa, Takashi, Sawamura, Motoki, Wada, Fumito, Yamamoto, Tsuyoshi, Obika, Satoshi, Hari, Yoshiyuki
Published in Organic & biomolecular chemistry (2017)
Published in Organic & biomolecular chemistry (2017)
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Journal Article
Present and Future Impact of Pharmaceuticals on Medical Economy
Hashida, Tohru, Osawa, Takashi
Published in Journal of Pharmaceutical Science and Technology, Japan (2020)
Published in Journal of Pharmaceutical Science and Technology, Japan (2020)
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Journal Article
Blood distribution of subcutaneous bortezomib and its kinetics in multiple myeloma patients
Osawa, Takashi, Naito, Takafumi, Mino, Yasuaki, Kawakami, Junichi
Published in Drug metabolism and pharmacokinetics (01.01.2017)
Published in Drug metabolism and pharmacokinetics (01.01.2017)
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