Discovery of a Potent, Selective, and Orally Active Proteasome Inhibitor for the Treatment of Cancer
Dorsey, Bruce D, Iqbal, Mohamed, Chatterjee, Sankar, Menta, Ernesto, Bernardini, Raffaella, Bernareggi, Alberto, Cassarà, Paolo G, D’Arasmo, Germano, Ferretti, Edmondo, De Munari, Sergio, Oliva, Ambrogio, Pezzoni, Gabriella, Allievi, Cecilia, Strepponi, Ivan, Ruggeri, Bruce, Ator, Mark A, Williams, Michael, Mallamo, John P
Published in Journal of medicinal chemistry (28.02.2008)
Published in Journal of medicinal chemistry (28.02.2008)
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Journal Article
Selective Platination of Biologically Relevant Polyamines. Linear Coordinating Spermidine and Spermine as Amplifying Linkers in Dinuclear Platinum Complexes
Rauter, Holger, Di Domenico, Roberto, Menta, Ernesto, Oliva, Ambrogio, Qu, Yun, Farrell, Nicholas
Published in Inorganic chemistry (27.08.1997)
Published in Inorganic chemistry (27.08.1997)
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Journal Article
Synthesis and Antitumor Evaluation of 2,5-Disubstituted- Indazolo[4,3-g h]isoquinolin-6(2H)-ones (9-Aza-anthrapyrazoles)
Krapcho, A. Paul, Menta, Ernesto, Oliva, Ambrogio, Di Domenico, Roberto, Fiocchi, Luigi, Maresch, Martin E, Gallagher, Cynthia E, Hacker, Miles P, Beggiolin, Gino, Giuliani, Fernando C, Pezzoni, Gabriella, Spinelli, Silvano
Published in Journal of medicinal chemistry (31.12.1998)
Published in Journal of medicinal chemistry (31.12.1998)
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Journal Article
Physicochemical properties, cytotoxic activity and topoisomerase ii inhibition of 2,3-diaza-anthracenediones
De Isabella, Paola, Palumbo, Manlio, Sissi, Claudia, Carenini, Nives, Capranico, Giovanni, Menta, Emesto, Oliva, Ambrogio, Spinelli, Silvano, Krapcho, A.Paul, Giuliani, Fernando C., Zunino, Franco
Published in Biochemical pharmacology (24.01.1997)
Published in Biochemical pharmacology (24.01.1997)
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Journal Article
Pyrimidine-2,4,6-Triones: A New Effective and Selective Class of Matrix Metalloproteinase Inhibitors
Grams, Frank, Brandstetter, Hans, DAlò, Simonetta, Geppert, Dagmar, Krell, Hans-Willi, Leinert, Herbert, Livi, Valeria, Menta, Ernesto, Oliva, Ambrogio, Zimmermann, Gerd
Published in Biological chemistry (01.08.2001)
Published in Biological chemistry (01.08.2001)
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Journal Article
6,9-Bis[(aminoalkyl)amino]benzo[g]isoquinoline-5,10-diones. A Novel Class of Chromophore-Modified Antitumor Anthracene-9,10-diones: Synthesis and Antitumor Evaluations
Krapcho, A. Paul, Petry, Mary E, Getahun, Zelleka, Landi, John J, Stallman, John, Polsenberg, Johanna F, Gallagher, Cynthia E, Maresch, Martin J, Hacker, Miles P
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
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Journal Article
Topoisomerase II DNA cleavage stimulation, DNA binding activity, cytotoxicity, and physico-chemical properties of 2-aza- and 2-aza-oxide-anthracenedione derivatives
De Isabella, P, Palumbo, M, Sissi, C, Capranico, G, Carenini, N, Menta, E, Oliva, A, Spinelli, S, Krapcho, A P, Giuliani, F C
Published in Molecular pharmacology (01.07.1995)
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Published in Molecular pharmacology (01.07.1995)
Journal Article
N-tert-butoxycarbonyl-N-substituted hydrazines in SNAr displacements. Synthetic pathways to N-1-substituted anthrapyrazoles, aza-anthrapyrazoles and aza-benzothiopyranoindazoles
Oliva, A, Ellis, M, Fiocchi, L, Menta, E, Krapcho, AP
Published in Journal of heterocyclic chemistry (01.01.2000)
Published in Journal of heterocyclic chemistry (01.01.2000)
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Journal Article
Synthesis, DNA-damaging and cytotoxic properties of novel topoisomerase II-directed bisantrene analogues
Zagotto, Giuseppe, Oliva, Ambrogio, Guano, Fulvio, Menta, Ernesto, Capranico, Giovanni, Palumbo, Manlio
Published in Bioorganic & medicinal chemistry letters (20.01.1998)
Published in Bioorganic & medicinal chemistry letters (20.01.1998)
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Journal Article
Meltikornatálmar og aðferðir til að nota þá
D'Arasmo, Germano, De Munari, Sergio, Menta, Ernesto, Ferretti, Edmondo, G Cassara, Paolo, Bernareggi, Alberto, Chatterjee, Sankar, Bernardini, Raffaella, Iqbal, Mohamed, Oliva, Ambrogio, A. Messina McLaughlin, Patricia
Year of Publication 15.05.2019
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Year of Publication 15.05.2019
Patent
PROTEASOME INHIBITORS AND METHODS OF USING THE SAME
OLIVA, AMBROGIO, IQBAL, MOHAMED, BERNAREGGI, ALBERTO, CASSARA, PAOLO G, D'ARASMO, GERMANO, FERRETTI, EDMONDO, DE NUNARI, SERGIO, CHATTERJEE, SANKAR, MESSINA MCLAUGHLIN, PATRICIA A, BERNARDINI, RAFAELLA, MENTA, ERNESTO
Year of Publication 29.12.2017
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Year of Publication 29.12.2017
Patent
Inhibidores del proteasoma y procedimientos de uso de los mismos
FERRETTI, Edmondo, DE NUNARI, Sergio, CHATTERJEE, Sankar, MENTA, Ernesto, BERNAREGGI, ALberto, BERNARDINI, Rafaella, MESSINA MCLAUGHLIN, Patricia A, IQBAL, Mohamed, CASSARA, Paolo G, OLIVA, Ambrogio, D'ARASMO, Germano
Year of Publication 28.06.2017
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Year of Publication 28.06.2017
Patent