Xanomeline: a novel muscarinic receptor agonist with functional selectivity for M1 receptors
Shannon, H E, Bymaster, F P, Calligaro, D O, Greenwood, B, Mitch, C H, Sawyer, B D, Ward, J S, Wong, D T, Olesen, P H, Sheardown, M J, Swedberg, M D, Suzdak, P D, Sauerberg, P
Published in The Journal of pharmacology and experimental therapeutics (01.04.1994)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1994)
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Improving the Nicotinic Pharmacophore with a Series of (Isoxazole)methylene-1-azacyclic Compounds: Synthesis, Structure−Activity Relationship, and Molecular Modeling
Tønder, Janne E, Hansen, John Bondo, Begtrup, Mikael, Pettersson, Ingrid, Rimvall, Karin, Christensen, Birgitte, Ehrbar, Ulrich, Olesen, Preben H
Published in Journal of medicinal chemistry (02.12.1999)
Published in Journal of medicinal chemistry (02.12.1999)
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Neurochemical effects of the M1 muscarinic agonist xanomeline (LY246708/NNC11-0232)
BYMASTER, F. P, WONG, D. T, SWEDBERG, D. B, SAUERBERG, P, MITCH, C. H, WARD, J. S, CALLIGARO, D. O, SCHOEPP, D. D, SHANNON, H. E, DHEARDOWN, M. J, OLESEN, P. H, ZUZDAK, P. D
Published in The Journal of pharmacology and experimental therapeutics (01.04.1994)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1994)
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Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5 R,6 R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane
Bymaster, Frank P, Shannon, Harlan E, Rasmussen, Kurt, Delapp, Neil W, Mitch, Charles H, Ward, John S, Calligaro, David O, Ludvigsen, Thomas S, Sheardown, Malcolm J, Olesen, Preben H, Swedberg, Michael D.B, Sauerberg, Per, Fink-Jensen, Anders
Published in European journal of pharmacology (04.09.1998)
Published in European journal of pharmacology (04.09.1998)
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Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3-(1,2,5-thiadiazolyl)-1,2,5,6-tetrahydro-1-methylpyridines
Sauerberg, Per, Olesen, Preben H, Nielsen, Susanne, Treppendahl, Svend, Sheardown, Malcolm J, Honore, Tage, Mitch, Charles H, Ward, John S, Pike, Andrew J
Published in Journal of medicinal chemistry (01.06.1992)
Published in Journal of medicinal chemistry (01.06.1992)
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Muscarinic Agonists with Antipsychotic-like Activity: Structure−Activity Relationships of 1,2,5-Thiadiazole Analogues with Functional Dopamine Antagonist Activity
Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Rasmussen, Thøger, Swedberg, Michael D. B, Sheardown, Malcolm J, Fink-Jensen, Anders, Thomsen, Christian, Thøgersen, Henning, Rimvall, Karin, Ward, John S, Calligaro, David O, DeLapp, Neil W, Bymaster, Frank P, Shannon, Harlan E
Published in Journal of medicinal chemistry (22.10.1998)
Published in Journal of medicinal chemistry (22.10.1998)
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Fate of circulating amino-terminal propeptide of type III procollagen in conscious pigs
Jensen, L T, Henriksen, J H, Risteli, J, Olesen, H P, Nielsen, M D, Lorenzen, I
Published in The American journal of physiology (01.07.1993)
Published in The American journal of physiology (01.07.1993)
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Muscarinic Analgesics with Potent and Selective Effects on the Gastrointestinal Tract: Potential Application for the Treatment of Irritable Bowel Syndrome
Mitch, Charles H, Brown, Thomas J, Bymaster, Frank P, Calligaro, David O, Dieckman, Donna, Merrit, Leander, Peters, Steven C, Quimby, Steven J, Shannon, Harlan E, Shipley, Lisa A, Ward, John S, Hansen, Kristian, Olesen, Preben H, Sauerberg, Per, Sheardown, Malcolm J, Swedberg, Michael D. B, Suzdak, Peter, Greenwood, Beverley
Published in Journal of medicinal chemistry (14.02.1997)
Published in Journal of medicinal chemistry (14.02.1997)
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Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic M1 receptor activation
Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Sheardown, Malcolm J, Fink-Jensen, Anders, Rasmussen, Thøger, Rimvall, Karin, Shannon, Harlan E, Bymaster, Frank P, DeLapp, Neil W, Calligaro, Dave O, Ward, John S, Whitesitt, Celia A, Thomsen, Christian
Published in Bioorganic & medicinal chemistry letters (20.10.1998)
Published in Bioorganic & medicinal chemistry letters (20.10.1998)
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Identification of novel (isoxazole)methylene-1-azabicyclic compounds with high affinity for the central nicotinic cholinergic receptor
Olesen, P.H., Swedberg, M.D.B., Eskesen, K., Judge, M.E., Egebjerg, J., Tønder, J.E., Rasmussen, T., Sheardown, M.J., Rimvall, K.
Published in Bioorganic & medicinal chemistry letters (05.08.1997)
Published in Bioorganic & medicinal chemistry letters (05.08.1997)
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3-(3-Alkylthio-1,2,5-thiadiazol-4-yl)-1-azabicycles. Structure—activity relationships for antinociception mediated by central muscarinic receptors
Olesen, PH, Sauerberg, P, Treppendahl, S, Larsson, O, Sheardown, MJ, Suzdak, PD, Mitch, CH, Ward, JS, Bymaster, FP, Shannon, HE, Swedberg, MDB
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Autologous fibrin sealant in reconstructive rabbit oviduct microsurgery
Weis-Fogh, Ulla Sivertsen, Schroeder, Erik, Olesen, Henning Peter, Sørensen, Søren Stampe
Published in Fertility and sterility (01.07.1990)
Published in Fertility and sterility (01.07.1990)
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Histomorphological evaluation of wound healing of rabbit oviduct after microsurgical reanastomosis with the use of autologous fibrin adhesive, human fibrin adhesive or poly-glycolic acid suture
Weis-Fogh, U S, Pedersen, H, Schroeder, E, Sørensen, S S, Olesen, H P
Published in European surgical research (1993)
Published in European surgical research (1993)
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