A Purification Strategy Utilizing Hydrophobic Interaction Chromatography to Obtain Homogeneous Species from a Site-Specific Antibody Drug Conjugate Produced by AJICAP™ First Generation
Matsuda, Yutaka, Leung, Monica, Okuzumi, Tatsuya, Mendelsohn, Brian
Published in Antibodies (Basel) (18.05.2020)
Published in Antibodies (Basel) (18.05.2020)
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Biological Evaluation of Maytansinoid-Based Site-Specific Antibody-Drug Conjugate Produced by Fully Chemical Conjugation Approach: AJICAP
Seki, Takuya, Yamada, Kei, Ooba, Yuri, Fujii, Tomohiro, Narita, Takahiro, Nakayama, Akira, Kitahara, Yoshiro, Mendelsohn, Brian A., Matsuda, Yutaka, Okuzumi, Tatsuya
Published in Frontiers in bioscience (Landmark. Print) (05.08.2022)
Published in Frontiers in bioscience (Landmark. Print) (05.08.2022)
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Chromatographic analysis of site-specific antibody-drug conjugates produced by AJICAP first-generation technology using a recombinant FcγIIIa receptor-ligand affinity column
Matsuda, Yutaka, Chakrabarti, Atis, Takahashi, Kazutoshi, Yamada, Kei, Nakata, Kunio, Okuzumi, Tatsuya, Mendelsohn, Brian A.
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.07.2021)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.07.2021)
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AJICAP Second Generation: Improved Chemical Site-Specific Conjugation Technology for Antibody–Drug Conjugate Production
Fujii, Tomohiro, Matsuda, Yutaka, Seki, Takuya, Shikida, Natsuki, Iwai, Yusuke, Ooba, Yuri, Takahashi, Kazutoshi, Isokawa, Muneki, Kawaguchi, Sayaka, Hatada, Noriko, Watanabe, Tomohiro, Takasugi, Rika, Nakayama, Akira, Shimbo, Kazutaka, Mendelsohn, Brian A., Okuzumi, Tatsuya, Yamada, Kei
Published in Bioconjugate chemistry (09.03.2023)
Published in Bioconjugate chemistry (09.03.2023)
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Chemical Site-Specific Conjugation Platform to Improve the Pharmacokinetics and Therapeutic Index of Antibody–Drug Conjugates
Matsuda, Yutaka, Seki, Takuya, Yamada, Kei, Ooba, Yuri, Takahashi, Kazutoshi, Fujii, Tomohiro, Kawaguchi, Sayaka, Narita, Takahiro, Nakayama, Akira, Kitahara, Yoshiro, Mendelsohn, Brian A, Okuzumi, Tatsuya
Published in Molecular pharmaceutics (01.11.2021)
Published in Molecular pharmaceutics (01.11.2021)
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Inhibitor hijacking of Akt activation
Shokat, Kevan M, Okuzumi, Tatsuya, Fiedler, Dorothea, Zhang, Chao, Gray, Daniel C, Aizenstein, Brian, Hoffman, Randy
Published in Nature Chemical Biology (01.07.2009)
Published in Nature Chemical Biology (01.07.2009)
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AJICAP-M: Traceless Affinity Peptide Mediated Conjugation Technology for Site-Selective Antibody–Drug Conjugate Synthesis
Matsuda, Yutaka, Shikida, Natsuki, Hatada, Noriko, Yamada, Kei, Seki, Takuya, Nakahara, Yuichi, Endo, Yuta, Shimbo, Kazutaka, Takahashi, Kazutoshi, Nakayama, Akira, Mendelsohn, Brian A., Fujii, Tomohiro, Okuzumi, Tatsuya, Hirasawa, Shigeo
Published in Organic letters (12.07.2024)
Published in Organic letters (12.07.2024)
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Journal Article
Synthesis and evaluation of indazole based analog sensitive Akt inhibitors
Okuzumi, Tatsuya, Ducker, Gregory S, Zhang, Chao, Aizenstein, Brian, Hoffman, Randy, Shokat, Kevan M
Published in Molecular bioSystems (01.08.2010)
Published in Molecular bioSystems (01.08.2010)
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HETEROCYCLIC SULFONAMIDE DERIVATIVE AND MEDICINE COMPRISING SAME
KAWAHIRA MIZUKI, OHSUMI KOJI, KOBAYASHI KAORI, SUGIKI MASAYUKI, SUZUKI TAMOTSU, FUJII TOMOHIRO, OKUZUMI TATSUYA
Year of Publication 25.11.2016
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Year of Publication 25.11.2016
Patent
HETEROCYCLIC AMIDE DERIVATIVE AND PHARMACEUTICAL PRODUCT CONTAINING SAME
KOBAYASHI, KAORI, SHIRAISHI, SEIJI, ASARI, SAYAKA, SUZUKI, TAMOTSU, OKUZUMI, TATSUYA
Year of Publication 25.07.2013
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Year of Publication 25.07.2013
Patent
Synthesis and evaluation of indazole based analog sensitive Akt inhibitorsElectronic supplementary information (ESI) available: Supplementary Table 1. See DOI: 10.1039/c003917aThis article is part of a Molecular BioSystems themed issue on Chemical Genomics
Okuzumi, Tatsuya, Ducker, Gregory S, Zhang, Chao, Aizenstein, Brian, Hoffman, Randy, Shokat, Kevan M
Year of Publication 12.07.2010
Year of Publication 12.07.2010
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Journal Article
HETEROCYCLIC SULFONAMIDE DERIVATIVE AND MEDICINE COMPRISING SAME
KOBAYASHI, KAORI, FUJII, TOMOHIRO, OHSUMI, KOJI, KAWAHIRA, MIZUKI, SUZUKI, TAMOTSU, SUGIKI, MASAYUKI, OKUZUMI, TATSUYA
Year of Publication 06.08.2015
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Year of Publication 06.08.2015
Patent
Efficient solid-phase synthesis of diverse 1,2,3-benzotriazin-4-ones using tert-butyl nitrite
Okuzumi, Tatsuya, Nakanishi, Eiji, Tsuji, Takashi, Makino, Shingo
Published in Tetrahedron letters (14.07.2003)
Published in Tetrahedron letters (14.07.2003)
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