Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) Antagonists
Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M
Published in Journal of medicinal chemistry (08.12.2011)
Published in Journal of medicinal chemistry (08.12.2011)
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(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor
Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Okun, Ilya M, Tkachenko, Sergey E, Vorobiev, Anton A
Published in Journal of medicinal chemistry (22.07.2010)
Published in Journal of medicinal chemistry (22.07.2010)
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Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists
IVACHTCHENKO, Alexandre V, FROLOV, Eugene B, MITKIN, Oleg D, KYSIL, Volodymyr M, KHVAT, Alexander V, OKUN, Ilya M, TLCACHENKO, Sergey E
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Journal Article
Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6 receptor antagonists
IVACHTCHENKO, Alexandre V, DMITRIEV, Dmitri E, VOROBIOV, Anton A, GOLOVINA, Elena S, DUBROVSKAYA, Elena S, KADIEVA, Madina G, KORYAKOVA, Angela G, KYSIL, Volodymyr M, MITKIN, Oleg D, TKACHENKO, Sergey E, OKUN, Ilya M
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indoles
Ivachtchenko, Alexandre V, Frolov, Eugen B, Mitkin, Oleg D, Tkachenko, Sergei E, Okun, Ilya M, Khvat, Alex V
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists
Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kovalenko, Sergiy M., Mitkin, Oleg D., Okun, Ilya M., Ravnyeyko, Irina M., Tkachenko, Sergey E., Zaremba, Oleg V.
Published in Bioorganic & medicinal chemistry (15.07.2010)
Published in Bioorganic & medicinal chemistry (15.07.2010)
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Synthesis and Structure−Activity Relationship of 4-Substituted 2-(2-Acetyloxyethyl)-8-(morpholine- 4-sulfonyl)pyrrolo[3,4-c]quinoline- 1,3-diones as Potent Caspase-3 Inhibitors
Kravchenko, Dmitri V, Kuzovkova, Yulia A, Kysil, Volodymyr M, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Balakin, Konstantin V, Ivachtchenko, Alexandre V
Published in Journal of medicinal chemistry (02.06.2005)
Published in Journal of medicinal chemistry (02.06.2005)
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Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. Synthesis and SAR of 2-substituted 4-methyl-8-(morpholine-4-sulfonyl)-pyrrolo[3,4- c]quinoline-1,3-diones
Kravchenko, Dmitri V., Kysil, Volodymyr M., Tkachenko, Sergey E., Maliarchouk, Sergey, Okun, Ilya M., Ivachtchenko, Alexandre V.
Published in European journal of medicinal chemistry (01.12.2005)
Published in European journal of medicinal chemistry (01.12.2005)
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1,3-Dioxo-4-methyl-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines as potent caspase-3 inhibitors
Kravchenko, Dmitri V, Kysil, Vladimir V, Ilyn, Alexey P, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Ivachtchenko, Alexandre V
Published in Bioorganic & medicinal chemistry letters (01.04.2005)
Published in Bioorganic & medicinal chemistry letters (01.04.2005)
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Journal Article
Synthesis and caspase-3 inhibitory activity of 8-sulfonyl-1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines
Kravchenko, Dmitri V, Kysil, Volodymyr M, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Ivachtchenko, Alexandre V
Published in Farmaco (Società chimica italiana : 1989) (01.10.2005)
Published in Farmaco (Società chimica italiana : 1989) (01.10.2005)
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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5- a ]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT 6 Receptor (5-HT 6 R) Antagonists
Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya M.
Published in Journal of medicinal chemistry (08.12.2011)
Published in Journal of medicinal chemistry (08.12.2011)
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Journal Article
Solution Phase Parallel Synthesis of Substituted 3-Phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: Selective Serotonin 5-HT6 Receptor Antagonists
Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kovalenko, Sergiy M, Mitkin, Oleg D, Okun, Ilya M, Ravnyeyko, Irina M, Tkachenko, Sergey E, Zaremba, Oleg V
Published in Journal of combinatorial chemistry (12.07.2010)
Published in Journal of combinatorial chemistry (12.07.2010)
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Journal Article
Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1 H-pyrido[4,3- b]indoles
Ivachtchenko, Alexandre V., Frolov, Eugen B., Mitkin, Oleg D., Tkachenko, Sergei E., Okun, Ilya M., Khvat, Alex V.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
(3-Phenylsulfonylcycloalkano[ e and d ]pyrazolo[1,5- a ]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT 6 Receptor
Ivachtchenko, Alexandre V., Dmitriev, Dmitri E., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kysil, Volodymyr M., Mitkin, Oleg D., Okun, Ilya M., Tkachenko, Sergey E., Vorobiev, Anton A.
Published in Journal of medicinal chemistry (22.07.2010)
Published in Journal of medicinal chemistry (22.07.2010)
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Journal Article
Synthesis and biological evaluation of novel [gamma]-carboline analogues of Dimebon as potent 5-HT[sub]6 receptor antagonists
Ivachtchenko, Alexandre V, Frolov, Eugene B, Mitkin, Oleg D, Kysil, Volodymyr M, Khvat, Alexander V, Okun, Ilya M, Tkachenko, Sergey E
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Journal Article
Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT sub(6) receptor antagonists
Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Dubrovskaya, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M, Vorobiov, Anton A
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Journal Article
Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5- a]pyrimidines and their evaluation as 5-HT 6 receptor antagonists
Ivachtchenko, Alexandre V., Dmitriev, Dmitri E., Golovina, Elena S., Dubrovskaya, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya M., Vorobiov, Anton A.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
Get full text
Journal Article
Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT 6 receptor antagonists
Ivachtchenko, Alexandre V., Frolov, Eugene B., Mitkin, Oleg D., Kysil, Volodymyr M., Khvat, Alexander V., Okun, Ilya M., Tkachenko, Sergey E.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article