Discovery of the First Non-Peptide Full Agonists for the Human Bradykinin B2 Receptor Incorporating 4-(2-Picolyloxy)quinoline and 1-(2-Picolyl)benzimidazole Frameworks
Sawada, Yuki, Kayakiri, Hiroshi, Abe, Yoshito, Mizutani, Tsuyoshi, Inamura, Noriaki, Asano, Masayuki, Hatori, Chie, Aramori, Ichiro, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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Pharmacological characteristics of a novel nonthiazolidinedione insulin sensitizer, FK614
Minoura, Hideaki, Takeshita, Shigeru, Ita, Makoto, Hirosumi, Jiro, Mabuchi, Miyuki, Kawamura, Ikuo, Nakajima, Satoko, Nakayama, Osamu, Kayakiri, Hiroshi, Oku, Teruo, Ohkubo-Suzuki, Akiko, Fukagawa, Masao, Kojo, Hitoshi, Hanioka, Kenichi, Yamasaki, Noritsugu, Imoto, Takafumi, Kobayashi, Yoshinori, Mutoh, Seitaro
Published in European journal of pharmacology (28.06.2004)
Published in European journal of pharmacology (28.06.2004)
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A Novel Class of Orally Active Non-Peptide Bradykinin B2 Receptor Antagonists. 1. Construction of the Basic Framework
Abe, Yoshito, Kayakiri, Hiroshi, Satoh, Shigeki, Inoue, Takayuki, Sawada, Yuki, Imai, Keisuke, Inamura, Noriaki, Asano, Masayuki, Hatori, Chie, Katayama, Akira, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (12.02.1998)
Published in Journal of medicinal chemistry (12.02.1998)
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A Novel Class of Orally Active Non-Peptide Bradykinin B2 Receptor Antagonists. 3. Discovering Bioisosteres of the Imidazo[1,2-a]pyridine Moiety
Abe, Yoshito, Kayakiri, Hiroshi, Satoh, Shigeki, Inoue, Takayuki, Sawada, Yuki, Inamura, Noriaki, Asano, Masayuki, Aramori, Ichiro, Hatori, Chie, Sawai, Hiroe, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (08.10.1998)
Published in Journal of medicinal chemistry (08.10.1998)
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The identification of an orally active, nonpeptide bradykinin B2 receptor antagonist, FR173657
Asano, Masayuki, Inamura, Noriaki, Hatori, Chie, Sawai, Hiroe, Fujiwara, Tatsujiro, Katayama, Akira, Kayakiri, Hiroshi, Satoh, Shigeki, Abe, Yoshito, Inoue, Takayuki, Sawada, Yuki, Nakahara, Kunio, Oku, Teruo, Okuhara, Masakuni
Published in British journal of pharmacology (01.02.1997)
Published in British journal of pharmacology (01.02.1997)
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A Novel Class of Orally Active Non-Peptide Bradykinin B2 Receptor Antagonists. 4. Discovery of Novel Frameworks Mimicking the Active Conformation
Abe, Yoshito, Kayakiri, Hiroshi, Satoh, Shigeki, Inoue, Takayuki, Sawada, Yuki, Inamura, Noriaki, Asano, Masayuki, Aramori, Ichiro, Hatori, Chie, Sawai, Hiroe, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (05.11.1998)
Published in Journal of medicinal chemistry (05.11.1998)
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A Novel Class of Orally Active Non-Peptide Bradykinin B2 Receptor Antagonists. 2. Overcoming the Species Difference between Guinea Pig and Man
Abe, Yoshito, Kayakiri, Hiroshi, Satoh, Shigeki, Inoue, Takayuki, Sawada, Yuki, Inamura, Noriaki, Asano, Masayuki, Hatori, Chie, Sawai, Hiroe, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (08.10.1998)
Published in Journal of medicinal chemistry (08.10.1998)
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Nonpeptide Mimic of Bradykinin with Long-Acting Properties at the Bradykinin B2 Receptor
Aramori, I, Zenkoh, J, Morikawa, N, Asano, M, Hatori, C, Sawai, H, Kayakiri, H, Satoh, S, Inoue, T, Abe, Y, Sawada, Y, Mizutani, T, Inamura, N, Nakahara, K, Kojo, H, Oku, T, Notsu, Y
Published in Molecular pharmacology (01.07.1997)
Published in Molecular pharmacology (01.07.1997)
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Pharmacological characterization of a nonpeptide bradykinin B2 receptor antagonist, FR165649, and agonist, FR190997
Asano, Masayuki, Hatori, Chie, Sawai, Hiroe, Johki, Shigeru, Inamura, Noriaki, Kayakiri, Hiroshi, Satoh, Shigeki, Abe, Yoshito, Inoue, Takayuki, Sawada, Yuki, Mizutani, Tsuyoshi, Oku, Teruo, Nakahara, Kunio
Published in British journal of pharmacology (01.06.1998)
Published in British journal of pharmacology (01.06.1998)
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Journal Article
The identification of an orally active, nonpeptide bradykinin B 2 receptor antagonist, FR173657
Asano, Masayuki, Inamura, Noriaki, Hatori, Chie, Sawai, Hiroe, Fujiwara, Tatsujiro, Katayama, Akira, Kayakiri, Hiroshi, Satoh, Shigeki, Abe, Yoshito, Inoue, Takayuki, Sawada, Yuki, Nakahara, Kunio, Oku, Teruo, Okuhara, Masakuni
Published in British journal of pharmacology (10.02.2009)
Published in British journal of pharmacology (10.02.2009)
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Pharmacological characterization of a novel, orally active, nonpeptide bradykinin B2 receptor antagonist, FR167344
INAMURA, N, ASANO, M, SAWADA, Y, OKU, T, NAKAHARA, K, HATORI, C, SAWAI, H, HIROSUMI, J, FUJIWARA, T, KAYAKIRI, H, SATOH, S, ABE, Y, INOUE, T
Published in European journal of pharmacology (20.08.1997)
Published in European journal of pharmacology (20.08.1997)
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Discovery of the first non-peptide full agonists for the human bradykinin B-2 receptor incorporating 4-(2-picolyloxy)quinoline and 1-(2-picolyl)benzimidazole frameworks
Sawada, Y, Kayakiri, H, Abe, Y, Mizutani, T, Inamura, N, Asano, M, Hatori, C, Aramori, Oku, T, Tanaka, H
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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Studies on 5-Lipoxygenase Inhibitors. II. Discovery, Optical Resolution and Enantioselective Synthesis of FR110302, a Highly Potent Non-redox Type-5-Lipoxygenase Inhibitor
YATABE, Takumi, KAYAKIRI, Hiroshi, KAWAI, Yoshio, OKU, Teruo, TANAKA, Hirokazu
Published in Chemical & pharmaceutical bulletin (1998)
Published in Chemical & pharmaceutical bulletin (1998)
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Journal Article
Pharmacological characterization of a nonpeptide bradykinin B 2 receptor antagonist, FR165649, and agonist, FR190997
Asano, Masayuki, Hatori, Chie, Sawai, Hiroe, Johki, Shigeru, Inamura, Noriaki, Kayakiri, Hiroshi, Satoh, Shigeki, Abe, Yoshito, Inoue, Takayuki, Sawada, Yuki, Mizutani, Tsuyoshi, Oku, Teruo, Nakahara, Kunio
Published in British journal of pharmacology (03.02.2009)
Published in British journal of pharmacology (03.02.2009)
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A New Series of Highly Potent Non-Peptide Bradykinin B2 Receptor Antagonists Incorporating the 4-Heteroarylquinoline Framework. Improvement of Aqueous Solubility and New Insights into Species Difference
Sawada, Yuki, Kayakiri, Hiroshi, Abe, Yoshito, Imai, Keisuke, Mizutani, Tsuyoshi, Inamura, Noriaki, Asano, Masayuki, Aramori, Ichiro, Hatori, Chie, Katayama, Akira, Oku, Teruo, Tanaka, Hirokazu
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
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Synthesis 8-epi-Kifunensine
KAYAKIRI, Hiroshi, OKU, Teruo, HASHIMOTO, Masashi
Published in Chemical & pharmaceutical bulletin (1991)
Published in Chemical & pharmaceutical bulletin (1991)
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A new series of highly potent non-peptide bradykinin B-2 receptor antagonists incorporating the 4-heteroarylquinoline framework. Improvement of aqueous solubility and new insights into species difference
Sawada, Y, Kayakiri, H, Abe, Y, Imai, K, Mizutani, T, Inamura, N, Asano, M, Aramori, Hatori, C, Katayama, A, Oku, T, Tanaka, H
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
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SYNTHESIS OF 8-EPI-KIFUNENSINE
KAYAKIRI, Hiroshi, OKU, Teruo, HASHIMOTO, Masashi
Published in Chemical & pharmaceutical bulletin (01.01.1990)
Published in Chemical & pharmaceutical bulletin (01.01.1990)
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