Discovery of JTZ-951: A HIF Prolyl Hydroxylase Inhibitor for the Treatment of Renal Anemia
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Published in ACS medicinal chemistry letters (14.12.2017)
Published in ACS medicinal chemistry letters (14.12.2017)
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Novel N-substituted 2-phenyl-1-sulfonylamino-cyclopropane carboxylates as selective ADAMTS-5 (Aggrecanase-2) inhibitors
SHIOZAKI, Makoto, MAEDA, Katsuya, MIMURA, Takayuki, SHINOZAKI, Yuichi, YOSHIUCHI, Hiromi, INABA, Takashi, MIURA, Tomoya, OGOSHI, Yosuke, HAAS, Julia, FRYER, Andrew M, LAIRD, Ellen R, LITTMANN, Nicole M, ANDREWS, Steven W, JOSEY, John A
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
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Design, synthesis, and structure–activity relationship of new isobenzofuranone ligands of protein kinase C
Baba, Yoshiyasu, Ogoshi, Yosuke, Hirai, Go, Yanagisawa, Takeshi, Nagamatsu, Kumiko, Mayumi, Satoshi, Hashimoto, Yuichi, Sodeoka, Mikiko
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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6-ALKOXYPYRAZOLOPYRIMIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF
NISHIMARU, Tatsuya, OHBA, Yusuke, OGOSHI, Yosuke, ADACHI, Kaoru, SAKURAI, Kentaro
Year of Publication 29.08.2024
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Year of Publication 29.08.2024
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6-아미노피라졸로피리미딘 화합물 및 그 의약 용도
OHBA YUSUKE, SATO SHIMPEI, NISHIMARU TATSUYA, ADACHI KAORU, SAKURAI KENTARO, OGOSHI YOSUKE
Year of Publication 26.04.2024
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Year of Publication 26.04.2024
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Discovery of potent liver-selective stearoyl-CoA desaturase-1 (SCD1) inhibitors, thiazole-4-acetic acid derivatives, for the treatment of diabetes, hepatic steatosis, and obesity
Iida, Tetsuya, Ubukata, Minoru, Mitani, Ikuo, Nakagawa, Yuichi, Maeda, Katsuya, Imai, Hiroto, Ogoshi, Yosuke, Hotta, Takahiro, Sakata, Shohei, Sano, Ryuhei, Morinaga, Hisayo, Negoro, Tamotsu, Oshida, Shinichi, Tanaka, Masahiro, Inaba, Takashi
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
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테트라히드로벤조푸로디아제피논 화합물 및 그의 의약 용도
NAKAGAWA YUICHI, YAMAOKA NOBUTAKA, MACHIDA TAKUYA, INOUE MASAFUMI, HARADA KAZUHITO, OGOSHI YOSUKE, FURUKAWA TAKAYUKI, MITANI IKUO
Year of Publication 09.06.2023
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Year of Publication 09.06.2023
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6-AMINOPYRAZOLOPYRIMIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF
NISHIMARU, Tatsuya, OHBA, Yusuke, OGOSHI, Yosuke, ADACHI, Kaoru, SAKURAI, Kentaro, SATO, Shimpei
Year of Publication 09.03.2023
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Year of Publication 09.03.2023
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TRIAZOLOPYRIDINE COMPOUND AND ACTION THEREOF AS PROLYL HYDROXYLASE INHIBITOR AND ERYTHROPOIETIN PRODUCTION INDUCER
HOTTA TAKAHIRO, ABE HIROYUKI, OGOSHI YOSUKE, YOKOTA MASAHIRO, UEYAMA KAZUHITO, MATSUI TAKUYA, ITO TAKASHI, MOTODA DAI, TERASHITA MASAKAZU, MITANI IKUO
Year of Publication 05.12.2023
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Year of Publication 05.12.2023
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Discovery of Selective Transforming Growth Factor β Type II Receptor Inhibitors as Antifibrosis Agents
Miwa, Shohei, Yokota, Masahiro, Ueyama, Yoshifumi, Maeda, Katsuya, Ogoshi, Yosuke, Seki, Noriyoshi, Ogawa, Naoki, Nishihata, Jun, Nomura, Akihiro, Adachi, Tsuyoshi, Kitao, Yuki, Nozawa, Keisuke, Ishikawa, Tomohiro, Ukaji, Yutaka, Shiozaki, Makoto
Published in ACS medicinal chemistry letters (13.05.2021)
Published in ACS medicinal chemistry letters (13.05.2021)
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TRIAZOLOPYRIDINE COMPOUND AND ACTION THEREOF AS PROLYL HYDROXYLASE INHIBITOR AND ERYTHROPOIETIN PRODUCTION INDUCER
HOTTA TAKAHIRO, ABE HIROYUKI, OGOSHI YOSUKE, YOKOTA MASAHIRO, UEYAMA KAZUHITO, MATSUI TAKUYA, ITO TAKASHI, MOTODA DAI, TERASHITA MASAKAZU, MITANI IKUO
Year of Publication 16.10.2019
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Year of Publication 16.10.2019
Patent
Asymmetric synthesis of isobenzofuranone derivatives and their unique character as protein kinase Cα (PKCα) activators
Hirai, Go, Ogoshi, Yosuke, Ohkubo, Megumi, Tamura, Yuki, Watanabe, Toru, Shimizu, Tadashi, Sodeoka, Mikiko
Published in Tetrahedron letters (01.07.2009)
Published in Tetrahedron letters (01.07.2009)
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TRIAZOLOPYRIDINE COMPOUND AND ACTION THEREOF AS PROLYL HYDROXYLASE INHIBITOR AND ERYTHROPOIETIN PRODUCTION INDUCER
HOTTA TAKAHIRO, ABE HIROYUKI, OGOSHI YOSUKE, YOKOTA MASAHIRO, UEYAMA KAZUHITO, MATSUI TAKUYA, ITO TAKASHI, MOTODA DAI, TERASHITA MASAKAZU, MITANI IKUO
Year of Publication 25.04.2018
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Year of Publication 25.04.2018
Patent
TRIAZOLOPYRIDINE COMPOUND AND ACTION THEREOF AS PROLYL HYDROXYLASE INHIBITOR AND ERYTHROPOIETIN PRODUCTION INDUCER
HOTTA TAKAHIRO, ABE HIROYUKI, OGOSHI YOSUKE, YOKOTA MASAHIRO, UEYAMA KAZUHITO, MATSUI TAKUYA, ITO TAKASHI, MOTODA DAI, TERASHITA MASAKAZU, MITANI IKUO
Year of Publication 15.02.2017
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Year of Publication 15.02.2017
Patent
Synthesis and SAR of 2-phenyl-1-sulfonylaminocyclopropane carboxylates as ADAMTS-5 (Aggrecanase-2) inhibitors
Shiozaki, Makoto, Imai, Hiroto, Maeda, Katsuya, Miura, Tomoya, Yasue, Katsutaka, Suma, Akira, Yokota, Masahiro, Ogoshi, Yosuke, Haas, Julia, Fryer, Andrew M., Laird, Ellen R., Littmann, Nicole M., Andrews, Steven W., Josey, John A., Mimura, Takayuki, Shinozaki, Yuichi, Yoshiuchi, Hiromi, Inaba, Takashi
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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2- DIHYDROPYRIMIDINE-2-ONE COMPOUNDS AND MEDICINAL USES THEREOF
FUJIOKA SHINGO, SHIOZAKI MAKOTO, IKENOGAMI TAKU, NOGUCHI MASATO, MAEDA KATSUYA, SUWA KATSUNORI, YOKOTA MASAHIRO, OGOSHI YOSUKE, WATANABE EIICHI, SEKI NORIYOSHI, SAKAI TAKAYUKI
Year of Publication 07.08.2017
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Year of Publication 07.08.2017
Patent
DIHYDROPYRIMIDINE-2-ONE COMPOUNDS AND MEDICINAL USES THEREOF
MAEDA, KATSUYA, YOKOTA, MASAHIRO, IKENOGAMI, TAKU, SEKI, NORIYOSHI, SAKAI, TAKAYUKI, OGOSHI, YOSUKE, SUWA, KATSUNORI, SHIOZAKI, MAKOTO, WATANABE, EIICHI, NOGUCHI, MASATO, FUJIOKA, SHINGO
Year of Publication 16.06.2016
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Year of Publication 16.06.2016
Patent