Discovery and Structure–Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials
Laleu, Benoît, Akao, Yuichiro, Ochida, Atsuko, Duffy, Sandra, Lucantoni, Leonardo, Shackleford, David M, Chen, Gong, Katneni, Kasiram, Chiu, Francis C. K, White, Karen L, Chen, Xue, Sturm, Angelika, Dechering, Koen J, Crespo, Benigno, Sanz, Laura M, Wang, Binglin, Wittlin, Sergio, Charman, Susan A, Avery, Vicky M, Cho, Nobuo, Kamaura, Masahiro
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Synthesis, Properties, and Catalytic Applications of Caged, Compact Trialkylphosphine 4-Phenyl-1-phospha-4-silabicyclo[2.2.2]octane
Ochida, Atsuko, Hamasaka, Go, Yamauchi, Yoshihiro, Kawamorita, Soichiro, Oshima, Naoya, Hara, Kenji, Ohmiya, Hirohisa, Sawamura, Masaya
Published in Organometallics (10.11.2008)
Published in Organometallics (10.11.2008)
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Nonvolatile Me3P-like P-Donor Ligand: Synthesis and Properties of 4-Phenyl-1-phospha-4-silabicyclo[2.2.2]octane
Ochida, Atsuko, Hara, Kenji, Ito, Hajime, Sawamura, Masaya
Published in Organic letters (24.07.2003)
Published in Organic letters (24.07.2003)
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Synthesis and properties of SMAPs 1-phospha-4-silabicyclo[2.2.2]octane derivatives
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Partnership Activity for Neglected Tropical Diseases
Akao, Yuichiro, Ochida, Atsuko, Muranishi, Hiroya, Nomura, Izumi, Ichikawa, Takashi
Published in YAKUGAKU ZASSHI (01.07.2022)
Published in YAKUGAKU ZASSHI (01.07.2022)
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Pharmacological inhibitory profile of TAK-828F, a potent and selective orally available RORγt inverse agonist
Shibata, Akira, Uga, Keiko, Sato, Takayuki, Sagara, Masaki, Igaki, Keiko, Nakamura, Yoshiki, Ochida, Atsuko, Kono, Mitsunori, Shirai, Junya, Yamamoto, Satoshi, Yamasaki, Masashi, Tsuchimori, Noboru
Published in Biochemical pharmacology (01.04.2018)
Published in Biochemical pharmacology (01.04.2018)
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Discovery of (ITcisIT-3-({(5ITRIT)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro-1ITHIT-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5ITHIT)-yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor gamma t Inverse Agonist
Kono, Mitsunori, Ochida, Atsuko, Oda, Tsuneo, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Masada, Shinichi, Kawamoto, Tetsuji, Yonemori, Kazuko, Nara, Yoshi, Fukase, Yoshiyuki, Yukawa, Tomoya, Tokuhara, Hidekazu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac D., Snell, Gyorgy P., Uga, Keiko, Shibata, Akira, Igaki, Keiko, Nakamura, Yoshiki, Nakagawa, Hideyuki, Tsuchimori, Noboru, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Discovery of [cis-3-({(5R)‑5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro‑1H‑inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5H)‑yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor γt Inverse Agonist
Kono, Mitsunori, Ochida, Atsuko, Oda, Tsuneo, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Masada, Shinichi, Kawamoto, Tetsuji, Yonemori, Kazuko, Nara, Yoshi, Fukase, Yoshiyuki, Yukawa, Tomoya, Tokuhara, Hidekazu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac D, Snell, Gyorgy P, Uga, Keiko, Shibata, Akira, Igaki, Keiko, Nakamura, Yoshiki, Nakagawa, Hideyuki, Tsuchimori, Noboru, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Nonbisphosphonate inhibitors of Plasmodium falciparum FPPS/GGPPS
Kabeche, Stephanie, Aida, Jumpei, Akther, Thamina, Ichikawa, Takashi, Ochida, Atsuko, Pulkoski-Gross, Michael J., Smith, Mark, Humphries, Paul S., Yeh, Ellen
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Collaborative Virtual Screening Identifies a 2‑Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection
Tawaraishi, Taisuke, Ochida, Atsuko, Akao, Yuichiro, Itono, Sachiko, Kamaura, Masahiro, Akther, Thamina, Shimada, Mitsuyuki, Canan, Stacie, Chowdhury, Sanjoy, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Francisco, Amanda, Ghosh, Sunil, Kaki, Rina, Kelly, John M., Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shum, David, Watanabe, Nao-aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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Identification of novel quinazolinedione derivatives as RORγt inverse agonist
Fukase, Yoshiyuki, Sato, Ayumu, Tomata, Yoshihide, Ochida, Atsuko, Kono, Mitsunori, Yonemori, Kazuko, Koga, Keiko, Okui, Toshitake, Yamasaki, Masashi, Fujitani, Yasushi, Nakagawa, Hideyuki, Koyama, Ryoukichi, Nakayama, Masaharu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac, Shirai, Junya, Yamamoto, Satoshi
Published in Bioorganic & medicinal chemistry (01.02.2018)
Published in Bioorganic & medicinal chemistry (01.02.2018)
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Optimization of Methionyl tRNA-Synthetase Inhibitors for Treatment of Cryptosporidium Infection
Buckner, Frederick S, Ranade, Ranae M, Gillespie, J Robert, Shibata, Sayaka, Hulverson, Matthew A, Zhang, Zhongsheng, Huang, Wenlin, Choi, Ryan, Verlinde, Christophe L M J, Hol, Wim G J, Ochida, Atsuko, Akao, Yuichiro, Choy, Robert K M, Van Voorhis, Wesley C, Arnold, Sam L M, Jumani, Rajiv S, Huston, Christopher D, Fan, Erkang
Published in Antimicrobial agents and chemotherapy (01.04.2019)
Published in Antimicrobial agents and chemotherapy (01.04.2019)
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Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivatives
Kono, Mitsunori, Oda, Tsuneo, Tawada, Michiko, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Kawamoto, Tetsuji, Tokuhara, Hidekazu, Tomata, Yoshihide, Ishii, Naoki, Ochida, Atsuko, Fukase, Yoshiyuki, Yukawa, Tomoya, Fukumoto, Shoji, Watanabe, Hiroyuki, Uga, Keiko, Shibata, Akira, Nakagawa, Hideyuki, Shirasaki, Mikio, Fujitani, Yasushi, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi
Published in Bioorganic & medicinal chemistry (15.01.2018)
Published in Bioorganic & medicinal chemistry (15.01.2018)
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