Health Utility Analysis of Tepotinib in Patients With Non-Small Cell Lung Cancer Harboring MET Exon 14 Skipping
Yang, Mo, Vioix, Helene, Hook, Emma S., Hatswell, Anthony J., Batteson, Rachael L., Gaumond, Bruce R., O’Brate, Aurora, Popat, Sanjay, Paik, Paul K.
Published in Value in health (01.08.2023)
Published in Value in health (01.08.2023)
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Tepotinib Treatment in Patients With MET Exon 14-Skipping Non-Small Cell Lung Cancer: Long-term Follow-up of the VISION Phase 2 Nonrandomized Clinical Trial
Mazieres, Julien, Paik, Paul K, Garassino, Marina C, Le, Xiuning, Sakai, Hiroshi, Veillon, Remi, Smit, Egbert F, Cortot, Alexis B, Raskin, Jo, Viteri, Santiago, Wu, Yi-Long, Yang, James C H, Ahn, Myung-Ju, Ma, Rui, Zhao, Jun, O'Brate, Aurora, Berghoff, Karin, Bruns, Rolf, Otto, Gordon, Johne, Andreas, Felip, Enriqueta, Thomas, Michael
Published in JAMA oncology (01.09.2023)
Published in JAMA oncology (01.09.2023)
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Brief Report: Clinical Response, Toxicity, and Resistance Mechanisms to Osimertinib Plus MET Inhibitors in Patients With EGFR-Mutant MET-Amplified NSCLC
Wang, Kaiwen, Du, Robyn, Roy-Chowdhuri, Sinchita, Li, Ziping T., Hong, Lingzhi, Vokes, Natalie, Elamin, Yasir Y., Hume, Celyne Bueno, Skoulidis, Ferdinandos, Gay, Carl M., Blumenschein, George, Fossella, Frank V., Tsao, Anne, Zhang, Jianjun, Karachaliou, Niki, O’Brate, Aurora, Gann, Claudia-Nanette, Lewis, Jeff, Rinsurongkawong, Waree, Lee, Jack, Gibbons, Don Lynn, Vaporciyan, Ara A., Heymach, John V., Altan, Mehmet, Le, Xiuning
Published in JTO clinical and research reports (01.08.2023)
Published in JTO clinical and research reports (01.08.2023)
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Chemistry and Biology of Diazonamide A: Second Total Synthesis and Biological Investigations
Nicolaou, K. C, Hao, Junliang, Reddy, Mali V, Rao, Paraselli Bheema, Rassias, Gerasimos, Snyder, Scott A, Huang, Xianhai, Chen, David Y.-K, Brenzovich, William E, Giuseppone, Nicolas, Giannakakou, Paraskevi, O'Brate, Aurora
Published in Journal of the American Chemical Society (13.10.2004)
Published in Journal of the American Chemical Society (13.10.2004)
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The synergistic combination of the farnesyl transferase inhibitor lonafarnib and paclitaxel enhances tubulin acetylation and requires a functional tubulin deacetylase
MARCUS, Adam I, JUN ZHOU, O'BRATE, Aurora, HAMEL, Ernest, JASON WONG, NIVENS, Michael, EL-NAGGAR, Adel, YAO, Tso-Pang, KHURI, Fadlo R, GIANNAKAKOU, Paraskevi
Published in Cancer research (Chicago, Ill.) (01.05.2005)
Published in Cancer research (Chicago, Ill.) (01.05.2005)
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Enhanced Microtubule-Dependent Trafficking and p53 Nuclear Accumulation by Suppression of Microtubule Dynamics
Giannakakou, Paraskevi, Nakano, Michel, Nicolaou, Kyriacos C., O'Brate, Aurora, Yu, Jian, Blagosklonny, Mikhail V., Greber, Urs F., Fojo, Tito
Published in Proceedings of the National Academy of Sciences - PNAS (06.08.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (06.08.2002)
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Farnesyltransferase inhibitors reverse taxane resistance
MARCUS, Adam I, O'BRATE, Aurora M, BUEY, Ruben M, JUN ZHOU, THOMAS, Shala, KHURI, Fadlo R, ANDREU, Jose Manuel, DIAZ, Fernando, GIANNAKAKOU, Paraskevi
Published in Cancer research (Chicago, Ill.) (01.09.2006)
Published in Cancer research (Chicago, Ill.) (01.09.2006)
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Detection of MET amplification ( MET amp) in patients with EGFR mutant (m) NSCLC after first-line (1L) osimertinib
Yu, Helena Alexandra, Kerr, Keith, Rolfo, Christian Diego, Fang, Jian, Finocchiaro, Giovanna, Wong, Kam-Hung, Veillon, Remi, Kato, Terufumi, Yang, James Chih-Hsin, Nadal, Ernest, Raskin, Jo, Le, Xiuning, Karachaliou, Niki, Ellers-Lenz, Barbara, OBrate, Aurora, Stroh, Christopher, Piske, Nadine, Boesler, Carsten, Yang, Jinji, Mazieres, Julien
Published in Journal of clinical oncology (01.06.2023)
Published in Journal of clinical oncology (01.06.2023)
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Intracranial activity of tepotinib in patients (pts) with MET exon 14 ( MET ex14) skipping NSCLC enrolled in VISION
Patel, Jyoti D., Le, Xiuning, Veillon, Remi, Anderson, Ian Churchill, Bestvina, Christine M., Demedts, Ingel, Garassino, Marina Chiara, Mazieres, Julien, Morise, Masahiro, Smit, Egbert F., Eggleton, S. Peter, OBrate, Aurora, Otto, Gordon, Bruns, Rolf, Schumacher, Karl-Maria, Paik, Paul K.
Published in Journal of clinical oncology (20.05.2021)
Published in Journal of clinical oncology (20.05.2021)
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Paclitaxel Resistance in Non–Small-Cell Lung Cancer Associated With Beta-Tubulin Gene Mutations
Monzó, M, Rosell, R, Sánchez, J J, Lee, J S, O'Brate, A, González-Larriba, J L, Alberola, V, Lorenzo, J C, Núñez, L, Ro, J Y, Martín, C
Published in Journal of clinical oncology (01.06.1999)
Published in Journal of clinical oncology (01.06.1999)
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Discovery of a Biologically Active Thiostrepton Fragment
Nicolaou, K. C, Zak, Mark, Rahimipour, Shai, Estrada, Anthony A, Lee, Sang Hyup, O'Brate, Aurora, Giannakakou, Paraskevi, Ghadiri, M. Reza
Published in Journal of the American Chemical Society (02.11.2005)
Published in Journal of the American Chemical Society (02.11.2005)
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Microtubule disruption targets HIF-1α mRNA to cytoplasmic P-bodies for translational repression
Carbonaro, Marisa, O'Brate, Aurora, Giannakakou, Paraskevi
Published in The Journal of cell biology (10.01.2011)
Published in The Journal of cell biology (10.01.2011)
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Microtubules regulate hypoxia-inducible factor-1α protein trafficking and activity: implications for taxane therapy
Carbonaro, Marisa, Escuin, Daniel, O'Brate, Aurora, Thadani-Mulero, Maria, Giannakakou, Paraskevi
Published in The Journal of biological chemistry (06.04.2012)
Published in The Journal of biological chemistry (06.04.2012)
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PP01.84 Tepotinib + Osimertinib in EGFR-mutant NSCLC with MET Amplification Following 1L Osimertinib: INSIGHT 2 Primary Analysis
Kim, Tae Min, Guarneri, Valentina, Voon, Pei Jye, Lim, Boon Khaw, Yang, Jin-ji, Wislez, Marie, Huang, Cheng, Liam, Chong Kin, Mazieres, Julien, Tho, ye Mun, Hayashi, Hidetoshi, Nguyen, Nhung, Chia, Puey Ling, de Marinis, Filippo, Raskin, Jo, Zhou, Qinghua, Finocchiaro, Giovanna, Le, Xiuning, Tan, Daniel, O’Hara, Richard M., Brutlach, Sabine, O’Brate, Aurora, Adrian, Svenja, Berghoff, Karin, Ellers-Lenz, Barbara, Karachaliou, Niki, Wu, Yi-Long
Published in Journal of thoracic oncology (01.07.2024)
Published in Journal of thoracic oncology (01.07.2024)
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Activity of tepotinib in hepatocellular carcinoma (HCC) with high-level MET amplification ( MET amp): Preclinical and clinical evidence
Faivre, Sandrine J., Blanc, Jean-frederic, Pan, Hongming, Grando, Véronique, Lim, Ho Yeong, Cubillo Gracián, Antonio, Isambert, Nicolas, Johne, Andreas, Schumacher, Karl, Stroh, Christopher, Friese-Hamim, Manja, O'Brate, Aurora, Zhou, Dongli, Qin, Shukui
Published in Journal of clinical oncology (20.01.2021)
Published in Journal of clinical oncology (20.01.2021)
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Tepotinib plus osimertinib in patients with EGFR-mutated non-small-cell lung cancer with MET amplification following progression on first-line osimertinib (INSIGHT 2): a multicentre, open-label, phase 2 trial
Wu, Yi-Long, Guarneri, Valentina, Voon, Pei Jye, Lim, Boon Khaw, Yang, Jin-Ji, Wislez, Marie, Huang, Cheng, Liam, Chong Kin, Mazieres, Julien, Tho, Lye Mun, Hayashi, Hidetoshi, Nhung, Nguyen Viet, Chia, Puey Ling, de Marinis, Filippo, Raskin, Jo, Zhou, Qinghua, Finocchiaro, Giovanna, Le, Anh Tuan, Wang, Jialei, Dooms, Christophe, Kato, Terufumi, Nadal, Ernest, Hin, How Soon, Smit, Egbert F, Wermke, Martin, Tan, Daniel, Morise, Masahiro, O'Brate, Aurora, Adrian, Svenja, Pfeiffer, Boris M, Stroh, Christopher, Juraeva, Dilafruz, Strotmann, Rainer, Goteti, Kosalaram, Berghoff, Karin, Ellers-Lenz, Barbara, Karachaliou, Niki, Le, Xiuning, Kim, Tae Min
Published in The lancet oncology (01.08.2024)
Published in The lancet oncology (01.08.2024)
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