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Published in The Journal of pharmacology and experimental therapeutics (01.12.2018)
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Discovery of MK-7246, a selective CRTH2 antagonist for the treatment of respiratory diseases
Gallant, Michel, Beaulieu, Christian, Berthelette, Carl, Colucci, John, Crackower, Michael A., Dalton, Chad, Denis, Danielle, Ducharme, Yves, Friesen, Richard W., Guay, Daniel, Gervais, François G., Hamel, Martine, Houle, Robert, Krawczyk, Connie M., Kosjek, Birgit, Lau, Stephen, Leblanc, Yves, Lee, Ernest E., Levesque, Jean-François, Mellon, Christophe, Molinaro, Carmela, Mullet, Wayne, O’Neill, Gary P., O’Shea, Paul, Sawyer, Nicole, Sillaots, Susan, Simard, Daniel, Slipetz, Deborah, Stocco, Rino, Sørensen, Dan, Truong, Vouy Linh, Wong, Elizabeth, Wu, Jin, Zaghdane, Helmi, Wang, Zhaoyin
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Selective modulation of chemokinesis, degranulation, and apoptosis in eosinophils through the PGD2 receptors CRTH2 and DP
Gervais, Francois G., Cruz, Rani P.G., Chateauneuf, Anne, Gale, Stephen, Sawyer, Nicole, Nantel, Francois, Metters, Kathleen M., O'Neill, Gary P.
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Published in Journal of allergy and clinical immunology (01.12.2001)
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Quantification of In Vivo Target Engagement Using Microfluidic Activity-Based Protein Profiling
Reardon, Holly T., Herbst, Rachel A., Henry, Cassandra L., Herbst, Dylan M., Ngo, Nhi, Cisar, Justin S., Weber, Olivia D., Niphakis, Micah J., O’Neill, Gary P.
Published in SLAS technology (01.10.2019)
Published in SLAS technology (01.10.2019)
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Identification of ABX-1431, a Selective Inhibitor of Monoacylglycerol Lipase and Clinical Candidate for Treatment of Neurological Disorders
Cisar, Justin S, Weber, Olivia D, Clapper, Jason R, Blankman, Jacqueline L, Henry, Cassandra L, Simon, Gabriel M, Alexander, Jessica P, Jones, Todd K, Ezekowitz, R. Alan B, O’Neill, Gary P, Grice, Cheryl A
Published in Journal of medicinal chemistry (25.10.2018)
Published in Journal of medicinal chemistry (25.10.2018)
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Discovery of a receptor related to the galanin receptors
Lee, Dennis K, Nguyen, Tuan, O'Neill, Gary P, Cheng, Regina, Liu, Yang, Howard, Andrew D, Coulombe, Nathalie, Tan, Carina P, Tang-Nguyen, Anh-Thi, George, Susan R, O'Dowd, Brian F
Published in FEBS letters (05.03.1999)
Published in FEBS letters (05.03.1999)
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Expression of the cysteinyl leukotriene 1 receptor in normal human lung and peripheral blood leukocytes
FIGUEROA, David J, BREYER, Richard M, JONES, Thomas R, LYNCH, Kevin R, AUSTIN, Christopher P, EVANS, Jilly F, DEFOE, Stephanie K, KARGMAN, Stacia, DAUGHERTY, Bruce L, WALDBURGER, Kristine, QINGYUN LIU, CLEMENTS, Michelle, ZHIZEN ZENG, O'NEILL, Gary P
Published in American journal of respiratory and critical care medicine (2001)
Published in American journal of respiratory and critical care medicine (2001)
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Expression of prostaglandin D synthase and the prostaglandin D2 receptors DP and CRTH2 in human nasal mucosa
Nantel, François, Fong, Carolyn, Lamontagne, Sonia, Wright, D Hamish, Giaid, Adel, Desrosiers, Martin, Metters, Kathleen M, O'Neill, Gary P, Gervais, François G
Published in Prostaglandins & other lipid mediators (01.01.2004)
Published in Prostaglandins & other lipid mediators (01.01.2004)
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The C3a receptor antagonist SB 290157 has agonist activity
Mathieu, Marie-Claude, Sawyer, Nicole, Greig, Gillian M., Hamel, Martine, Kargman, Stacia, Ducharme, Yves, Lau, Cheuk K., Friesen, Richard W., O’Neill, Gary P., Gervais, Francois G., Therien, Alex G.
Published in Immunology Letters (15.09.2005)
Published in Immunology Letters (15.09.2005)
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Identification of a Potent and Selective Synthetic Agonist at the CRTH2 Receptor
Gervais, François G, Morello, Jean-Pierre, Beaulieu, Christian, Sawyer, Nicole, Denis, Danielle, Greig, Gillian, Malebranche, A Daniel, O'Neill, Gary P
Published in Molecular pharmacology (01.06.2005)
Published in Molecular pharmacology (01.06.2005)
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Pharmacological characterization of MK-7246, a potent and selective CRTH2 (chemoattractant receptor-homologous molecule expressed on T-helper type 2 cells) antagonist
Gervais, Francois G, Sawyer, Nicole, Stocco, Rino, Hamel, Martine, Krawczyk, Connie, Sillaots, Susan, Denis, Danielle, Wong, Elizabeth, Wang, Zhaoyin, Gallant, Michel, Abraham, William M, Slipetz, Deborah, Crackower, Michael A, O'Neill, Gary P
Published in Molecular pharmacology (01.01.2011)
Published in Molecular pharmacology (01.01.2011)
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Structure-Function Relationships in the Neuropeptide S Receptor: MOLECULAR CONSEQUENCES OF THE ASTHMA-ASSOCIATED MUTATION N107I
Bernier, Virginie, Stocco, Rino, Bogusky, Michael J, Joyce, Joseph G, Parachoniak, Christine, Grenier, Karl, Arget, Michael, Mathieu, Marie-Claude, O'Neill, Gary P, Slipetz, Deborah, Crackower, Michael A, Tan, Christopher M, Therien, Alex G
Published in The Journal of biological chemistry (25.08.2006)
Published in The Journal of biological chemistry (25.08.2006)
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Molecular pharmacology of the human prostaglandin D 2 receptor, CRTH2
Sawyer, Nicole, Cauchon, Elizabeth, Chateauneuf, Anne, Cruz, Rani P G, Nicholson, Donald W, Metters, Kathleen M, O'Neill, Gary P, Gervais, Francois G
Published in British journal of pharmacology (01.12.2002)
Published in British journal of pharmacology (01.12.2002)
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Expression of prostaglandin G/H synthase-1 and -2 protein in human colon cancer
KARGMAN, S. L, O'NEILL, G. P, VICKERS, P. J, EVANS, J. F, MANCINI, J. A, JOTHY, S
Published in Cancer research (Chicago, Ill.) (15.06.1995)
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Published in Cancer research (Chicago, Ill.) (15.06.1995)
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Comparative analysis of the effects of antimuscarinic agents on bladder functions in both nonhuman primates and rodents
Nagabukuro, Hiroshi, Villa, Katherine L, Wickham, L Alexandra, Kulick, Alison A, Gichuru, Loise, Donnelly, Marcie J, Voronin, Gregory O, Pereira, Tony, Tong, Xinchun, Nichols, Andrew, Alves, Stephen E, O'Neill, Gary P, Johnson, Christopher V, Hickey, Emily J
Published in The Journal of pharmacology and experimental therapeutics (01.07.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2011)
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Adenovirus IL-13-Induced Airway Disease in Mice: A Corticosteroid-Resistant Model of Severe Asthma
Therien, Alex G, Bernier, Virginie, Weicker, Sean, Tawa, Paul, Falgueyret, Jean-Pierre, Mathieu, Marie-Claude, Honsberger, Jeanne, Pomerleau, Veronique, Robichaud, Annette, Stocco, Rino, Dufresne, Lynn, Houshyar, Hani, Lafleur, Josiane, Ramachandran, Chidambaram, O'Neill, Gary P, Slipetz, Deborah, Tan, Christopher M
Published in American journal of respiratory cell and molecular biology (01.07.2008)
Published in American journal of respiratory cell and molecular biology (01.07.2008)
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Characterization of the cloned guinea pig leukotriene B4 receptor: comparison to its human orthologue
BOIE, Y, STOCCO, R, ABRAMOVITZ, M, SAWYER, N, GREIG, G. M, KARGMAN, S, SLIPETZ, D. M, O'NEILL, G. P, SHIMIZU, T, YOKOMIZO, T, METTERS, K. M
Published in European journal of pharmacology (10.09.1999)
Published in European journal of pharmacology (10.09.1999)
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Identification of Distinct Plasma Biomarker Signatures in Patients with Rapid and Slow Declining Forms of COPD
Devanarayan, Viswanath, Scholand, Mary-Beth, Hoidal, John, Leppert, Mark F., Crackower, Michael A., O'Neill, Gary P., Gervais, Francois G.
Published in Chronic obstructive pulmonary disease (01.02.2011)
Published in Chronic obstructive pulmonary disease (01.02.2011)
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Arginine 120 of Prostaglandin G/H Synthase-1 Is Required for the Inhibition by Nonsteroidal Anti-inflammatory Drugs Containing a Carboxylic Acid Moiety
Mancini, J A, Riendeau, D, Falgueyret, J P, Vickers, P J, O'Neill, G P
Published in The Journal of biological chemistry (08.12.1995)
Published in The Journal of biological chemistry (08.12.1995)
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