Antimicrobial Properties and Mode of Action of the Pyrrothine Holomycin
OLIVA, Brunello, O'NEILL, Alexander, WILSON, Jenny M, O'HANLON, Peter J, CHOPRA, Ian
Published in Antimicrobial Agents and Chemotherapy (01.02.2001)
Published in Antimicrobial Agents and Chemotherapy (01.02.2001)
Get full text
Journal Article
Variable Sensitivity to Bacterial Methionyl-tRNA Synthetase Inhibitors Reveals Subpopulations of Streptococcus pneumoniae with Two Distinct Methionyl-tRNA Synthetase Genes
GENTRY, Daniel R, INGRAHAM, Karen A, STANHOPE, Michael J, RITTENHOUSE, Stephen, JARVEST, Richard L, O'HANLON, Peter J, BROWN, James R, HOLMES, David J
Published in Antimicrobial Agents and Chemotherapy (01.06.2003)
Published in Antimicrobial Agents and Chemotherapy (01.06.2003)
Get full text
Journal Article
Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase
BERGE, JOHN M., BROOM, NIGEL J. P., HOUGE-FRYDRYCH, CATHERINE S. V., JARVEST, RICHARD L., MENSAH, LUCY, MCNAIR, DAVID J., O'HANLON, PETER J., POPE, ANDREW J., RITTENHOUSE, STEPHEN
Published in Journal of antibiotics (01.11.2000)
Published in Journal of antibiotics (01.11.2000)
Get full text
Journal Article
The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
Brown, Murray J., Carter, Paul S., Fenwick, Ashley E., Fosberry, Andrew P., Hamprecht, Dieter W., Hibbs, Martin J., Jarvest, Richard L., Mensah, Lucy, Milner, Peter H., O'Hanlon, Peter J., Pope, Andrew J., Richardson, Christine M., West, Andrew, Witty, David R.
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Get full text
Journal Article
Seven-Membered Lactams as Constraints for Amide Self-Recognition
Nadin, Alan, Derrer, Sam, McGeary, Ross P, Goodman, Jonathan M, Raithby, Paul R, Holmes, Andrew B, O'Hanlon, Peter J, Pearson, Neil D
Published in Journal of the American Chemical Society (01.09.1995)
Published in Journal of the American Chemical Society (01.09.1995)
Get full text
Journal Article
Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens
JARVEST, Richard L., BERGE, John M., BERRY, Valerie, BOYD, Helen F., BROWN, Murray J., ELDER, John S., FORREST, Andrew K., FOSBERRY, Andrew P., GENTRY, Daniel R., HIBBS, Martin J., JAWORSKI, Deborah D., O'HANLON, Peter J., POPE, Andrew J., RITTENHOUSE, Stephen, SHEPPARD, Robert J., SLATER-RADOSTI, Courtney, WORBY, Angela
Published in Journal of medicinal chemistry (09.05.2002)
Published in Journal of medicinal chemistry (09.05.2002)
Get full text
Journal Article
SAR of biphenyl carboxamide ligands of the human melanin-concentrating hormone receptor 1 (MCH R1): Discovery of antagonist SB-568849
Witty, David R., Bateson, John H., Hervieu, Guillaume J., Jeffrey, Phillip, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin M., Wilson, Shelagh, Winborn, Kim Y.
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Get full text
Journal Article
Thiocarbonyl-based 1,3-dipolarophiles for the synthesis of C(2)-unsubstituted penems
Gallagher, Timothy, Sanchez, Sylvie, Bateson, John H., O'Hanlon, Peter J.
Published in Pure and applied chemistry (01.12.2005)
Published in Pure and applied chemistry (01.12.2005)
Get full text
Journal Article
S-Alkyl Dithioformates as 1,3-Dipolarophiles. Generation of C(2)-Unsubstituted Penems
Sanchez, Sylvie, Bateson, John H, O'Hanlon, Peter J, Gallagher, Timothy
Published in Organic letters (05.08.2004)
Published in Organic letters (05.08.2004)
Get full text
Journal Article
Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues
Jarvest, Richard L, Armstrong, Sula A, Berge, John M, Brown, Pamela, Elder, John S, Brown, Murray J, Copley, Royston C.B, Forrest, Andrew K, Hamprecht, Dieter W, O'Hanlon, Peter J, Mitchell, Darren J, Rittenhouse, Stephen, Witty, David R
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Get full text
Journal Article
Discovery of potent and stable conformationally constrained analogues of the MCH R1 antagonist SB-568849
Witty, David R., Bateson, John, Hervieu, Guillaume J., Al-Barazanji, Kamal, Jeffrey, Phillip, Hamprecht, Dieter, Haynes, Andrea, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin, Winborn, Kim Y.
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Get full text
Journal Article
Rational Design of Femtomolar Inhibitors of Isoleucyl tRNA Synthetase from a Binding Model for Pseudomonic Acid-A
Brown, Murray J. B, Mensah, Lucy M, Doyle, Michael L, Broom, Nigel J. P, Osbourne, Neal, Forrest, Andrew K, Richardson, Christine M, O'Hanlon, Peter J, Pope, Andrew J
Published in Biochemistry (Easton) (23.05.2000)
Published in Biochemistry (Easton) (23.05.2000)
Get full text
Journal Article
Analogues of SB-203207 as inhibitors of tRNA synthetases
Banwell, Martin G, Crasto, Curtis F, Easton, Christopher J, Forrest, Andrew K, Karoli, Tomislav, March, Darren R, Mensah, Lucy, Nairn, Michael R, O'Hanlon, Peter J, Oldham, Mark D, Yue, Weimin
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
Published in Bioorganic & medicinal chemistry letters (16.10.2000)
Get full text
Journal Article
The Chemistry of Pseudomonic Acid. † 18. Heterocyclic Replacement of the α,β-Unsaturated Ester: Synthesis, Molecular Modeling, and Antibacterial Activity
Brown, Pamela, Best, Desmond J, Broom, Nigel J. P, Cassels, Robert, O'Hanlon, Peter J, Mitchell, Timothy J, Osborne, Neal F, Wilson, Jennifer M
Published in Journal of medicinal chemistry (01.08.1997)
Published in Journal of medicinal chemistry (01.08.1997)
Get full text
Journal Article
Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity
Jarvest, Richard L, Berge, John M, Brown, Murray J, Brown, Pamela, Elder, John S, Forrest, Andrew K, Houge-Frydrych, C.S.V, O'Hanlon, Peter J, McNair, David J, Rittenhouse, Stephen, Sheppard, Robert J
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
Get full text
Journal Article
Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity
Jarvest, Richard L., Berge, John M., Brown, Pamela, Houge-Frydrych, Catherine S.V., O'Hanlon, Peter J., McNair, David J., Pope, Andrew J., Rittenhouse, Stephen
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
Get full text
Journal Article
Discovery and optimisation of potent, selective, ethanolamine inhibitors of bacterial phenylalanyl tRNA synthetase
Jarvest, Richard L., Erskine, Symon G., Forrest, Andrew K., Fosberry, Andrew P., Hibbs, Martin J., Jones, Joanna J., O’Hanlon, Peter J., Sheppard, Robert J., Worby, Angela
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Get full text
Journal Article
Synthesis and activity of analogues of the isoleucyl tRNA synthetase inhibitor SB-203207
CRASTO, Curtis F, FORREST, Andrew K, EASTON, Christopher J, KAROLI, Tomislav, MARCH, Darren R, MENSAH, Lucy, O'HANLON, Peter J, NAIRN, Michael R, OLDHAM, Mark D, WEIMIN YUE, BANWELL, Martin G
Published in Bioorganic & medicinal chemistry (03.07.2003)
Published in Bioorganic & medicinal chemistry (03.07.2003)
Get full text
Journal Article
Chemistry of Pseudomonic Acid. Part 16: Aryl and Heteroaryl Ketone Derivatives of Monic Acid
ABSON, ANGELA, BROOM, NIGEL J. P., COATES, PHILIPPA A., ELDER, JOHN S., FORREST, ANDREW K., HANNAN, PETER C. T., HICKS, AMANDA J., O'HANLON, PETER J., MASSON, NICKY D., PEARSON, NEIL D., PONS, JEAN E., WILSON, JENNIFER M.
Published in Journal of antibiotics (1996)
Published in Journal of antibiotics (1996)
Get full text
Journal Article
Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase
Brown, Pamela, Eggleston, Drake S., Haltiwanger, R.Curtis, Jarvest, Richard L., Mensah, Lucy, O'Hanlon, Peter J., Pope, Andrew J.
Published in Bioorganic & medicinal chemistry letters (12.03.2001)
Published in Bioorganic & medicinal chemistry letters (12.03.2001)
Get full text
Journal Article