In Vivo Evaluation and Dosimetry Estimate for a High Affinity Affibody PET Tracer Targeting PD-L1
Rubins, Daniel J, Meng, Xiangjun, McQuade, Paul, Klimas, Michael, Getty, Krista, Lin, Shu-An, Connolly, Brett M., O’Malley, Stacey S., Haley, Hyking, Purcell, Mona, Gantert, Liza, Holahan, Marie, Lindgren, Joel, Eklund, Pär, Ekblad, Caroline, Frejd, Fredrik Y., Hostetler, Eric D., González Trotter, Dinko E., Evelhoch, Jeffrey L.
Published in Molecular imaging and biology (01.04.2021)
Published in Molecular imaging and biology (01.04.2021)
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Synthesis and Evaluation of 5-Fluoro-2-aryloxazolo[5,4-b]pyridines as β-Amyloid PET Ligands and Identification of MK-3328
Harrison, Scott T, Mulhearn, James, Wolkenberg, Scott E, Miller, Patricia J, O’Malley, Stacey S, Zeng, Zhizhen, Williams, David L, Hostetler, Eric D, Sanabria-Bohórquez, Sandra, Gammage, Linda, Fan, Hong, Sur, Cyrille, Culberson, J. Christopher, Hargreaves, Richard J, Cook, Jacquelynn J, Hartman, George D, Barrow, James C
Published in ACS medicinal chemistry letters (14.07.2011)
Published in ACS medicinal chemistry letters (14.07.2011)
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A novel radioligand for glycine transporter 1: characterization and use in autoradiographic and in vivo brain occupancy studies
Zeng, Zhizhen, O'Brien, Julie A, Lemaire, Wei, O'Malley, Stacey S, Miller, Patricia J, Zhao, Zhijian, Wallace, Michael A, Raab, Conrad, Lindsley, Craig W, Sur, Cyrille, Williams, David L
Published in Nuclear medicine and biology (01.04.2008)
Published in Nuclear medicine and biology (01.04.2008)
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In Vivo Imaging of the Programmed Death Ligand 1 by 18 F PET
González Trotter, Dinko E, Meng, Xiangjun, McQuade, Paul, Rubins, Daniel, Klimas, Michael, Zeng, Zhizhen, Connolly, Brett M, Miller, Patricia J, O'Malley, Stacey S, Lin, Shu-An, Getty, Krista L, Fayadat-Dilman, Laurence, Liang, Linda, Wahlberg, Elisabet, Widmark, Olof, Ekblad, Caroline, Frejd, Fredrik Y, Hostetler, Eric D, Evelhoch, Jeffrey L
Published in Journal of Nuclear Medicine (01.11.2017)
Published in Journal of Nuclear Medicine (01.11.2017)
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IN VITRO BINDING STUDIES TO EVALUATE THE NFT-SPECIFICITY OF [3H]MK-6240 AND [3H]AV-1451 BINDING IN SUBCORTICAL REGIONS OF HUMAN AD BRAIN
Zeng, Zhizhen, Miller, Partricia J., Connolly, Brett M., O’Malley, Stacey S., Lohith, Talakad, Mulhearn, James, Bennacef, Idriss, Walji, Abbas, Schenk, David J., Hesk, David, Sur, Cyrille, Li, Wenping, Hostetler, Eric D., Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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IN VITRO BINDING STUDIES TO EVALUATE THE NFT-SPECIFICITY OF [3H]MK-6240 AND [3H]AV-1451 BINDING IN SUBCORTICAL REGIONS OF THE HUMAN AD BRAIN
Zeng, Zhizhen, Miller, Patricia J., Connolly, Brett M., O’Malley, Stacey S., Lohith, Talakad, Bennacef, Idriss, Mulhearn, James, Schenk, David J., Hesk, David, Walji, Abbas, Sur, Cyrille, Li, Wenping, Hostetler, Eric D., Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2017)
Published in Alzheimer's & dementia (01.07.2017)
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In Vivo Imaging of the Programmed Death Ligand 1 by 18F PET
González Trotter, Dinko E, Meng, Xiangjun, McQuade, Paul, Rubins, Daniel, Klimas, Michael, Zeng, Zhizhen, Connolly, Brett M, Miller, Patricia J, O'Malley, Stacey S, Lin, Shu-An, Getty, Krista L, Fayadat-Dilman, Laurence, Liang, Linda, Wahlberg, Elisabet, Widmark, Olof, Ekblad, Caroline, Frejd, Fredrik Y, Hostetler, Eric D, Evelhoch, Jeffrey L
Published in The Journal of nuclear medicine (1978) (01.11.2017)
Published in The Journal of nuclear medicine (1978) (01.11.2017)
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Synthesis, characterization, and first successful monkey imaging studies of metabotropic glutamate receptor subtype 5 (mGluR5) PET radiotracers
Hamill, Terence G., Krause, Stephen, Ryan, Christine, Bonnefous, Celine, Govek, Steve, Seiders, T. Jon, Cosford, Nicholas D.P., Roppe, Jeffrey, Kamenecka, Ted, Patel, Shil, Gibson, Raymond E., Sanabria, Sandra, Riffel, Kerry, Eng, Waisi, King, Christopher, Yang, Xiaoqing, Green, Mitchell D., O'malley, Stacey S., Hargreaves, Richard, Burns, H. Donald
Published in Synapse (New York, N.Y.) (15.06.2005)
Published in Synapse (New York, N.Y.) (15.06.2005)
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Potent and orally active angiotensin II receptor antagonists with equal affinity for human AT1 and AT2 subtypes
Chang, Linda L, Ashton, Wallace T, Flanagan, Kelly L, Chen, Tsing-Bau, O'Malley, Stacey S, Zingaro, Gloria J, Kivlighn, Salah D, Siegl, Peter K. S, Lotti, Victor J
Published in Journal of medicinal chemistry (01.09.1995)
Published in Journal of medicinal chemistry (01.09.1995)
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In Vivo Imaging of the Programmed Death Ligand 1 by F-18 PET
Trotter, Dinko E. Gonzalez, Meng, Xiangjun, McQuade, Paul, Rubins, Daniel, Klimas, Michael, Zeng, Zhizhen, Connolly, Brett M., Miller, Patricia J., O'Malley, Stacey S., Lin, Shu-An, Getty, Krista L., Fayadat-Dilman, Laurence, Liang, Linda, Wahlberg, Elisabet, Widmark, Olof, Ekblad, Caroline, Frejd, Fredrik Y., Hostetler, Eric D., Evelhoch, Jeffrey L.
Published in The Journal of nuclear medicine (1978) (01.11.2017)
Published in The Journal of nuclear medicine (1978) (01.11.2017)
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Benzodiazepines as Potent and Selective Bradykinin B1 Antagonists
Wood, Michael R, Kim, June J, Han, Wei, Dorsey, Bruce D, Homnick, Carl F, DiPardo, Robert M, Kuduk, Scott D, MacNeil, Tanya, Murphy, Kathy L, Lis, Edward V, Ransom, Richard W, Stump, Gary L, Lynch, Joseph J, O'Malley, Stacey S, Miller, Patricia J, Chen, Tsing-Bau, Harrell, Charles M, Chang, Raymond S. L, Sandhu, Punam, Ellis, Joan D, Bondiskey, Peter J, Pettibone, Douglas J, Freidinger, Roger M, Bock, Mark G
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Pharmacological characterization and radioligand binding properties of a high-affinity, nonpeptide, bradykinin B1 receptor antagonist
RANSOM, Richard W, HARRELL, Charles M, SU, Dai-Shi, MARKOWITZ, M. Kristine, WALLACE, Michael A, RAAB, Conrad E, JONES, Allen N, DEAN, Dennis C, PETTIBONE, Douglas J, FREIDINGER, Roger M, BOCK, Mark G, REISS, Duane R, MURPHY, Kathryn L, CHANG, Raymond S. L, HESS, J. Fred, MILLER, Patricia J, O'MALLEY, Stacey S, HEY, Pat J, KUNAPULI, Priya
Published in European journal of pharmacology (19.09.2004)
Published in European journal of pharmacology (19.09.2004)
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COMPARING [3 H]MK-6240 AND [3 H]AV-1451(T-807) IN IN VITRO BINDING STUDIES IN BRAIN TISSUES
Zeng, Zhizhen, Miller, Patricia J, Connolly, Brett M, O’Malley, Stacey S, Bennacef, Idriss, Mulhearn, James, Schenk, David J, Hesk, David, Soriano, Aileen, Abbas, Walji, Hostetler, Eric D
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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Journal Article
COMPARING [3 H]MK-6240 AND [3 H]AV-1451(T-807) IN IN VITRO BINDING STUDIES IN BRAIN TISSUES
Zeng, Zhizhen, Miller, Patricia J, Connolly, Brett M, O’Malley, Stacey S, Bennacef, Idriss, Mulhearn, James, David, Schenk J, Hesk, David, Soriano, Aileen, Abbas, Walji, Eric, Hostetler D
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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DISCOVERY AND FIRST-IN-HUMAN EVALUATION OF THE TAU-IMAGING PET RADIOTRACER [18 F]MK-6240
Bennacef, Idriss, Zeng, Zhizhen, Lohith, Talakad, Miller, Patricia J, Salinas, Cristian A, Connolly, Brett M, Gantert, Liza T, Haley, Hyking D, Marie, Holahan A, O’Malley, Stacey S, Purcell, Mona L, Riffel, Kerry, Coleman, Paul J, Li, Jing, Balsells-Padros, Jaume, Soriano, Aileen, Ogawa, Aimie M, Xu, Serena, Xiaoping, Zhang, Della Rocca, Joseph, Schachter, Joel B, Hesk, David, David, Schenk J, Telan-Choing, Florestina, Struyk, Arie, Sur, Cyrille, Celen, Sofie, Serdons, Kim, Bormans, Guy, Vandenbulcke, Mathieu, Vandenberghe, Rik, De Hoon, Jan, Koole, Michel, Van Laere, Koen, Declercq, Ruben, Tom, Reynders, Abbas, Walji, Eric, Hostetler D, Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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Journal Article
DISCOVERY AND FIRST-IN-HUMAN EVALUATION OF THE TAU-IMAGING PET RADIOTRACER [18 F]MK-6240
Bennacef, Idriss, Zeng, Zhizhen, Lohith, Talakad, Miller, Patricia J, Salinas, Cristian A, Connolly, Brett M, Gantert, Liza T, Hyking, Haley D, Holahan, Marie A, O’Malley, Stacey S, Purcell, Mona L, Riffel, Kerry, Coleman, Paul J, Li, Jing, Balsells-Padros, Jaume, Soriano, Aileen, Ogawa, Aimie M, Xu, Serena, Xiaoping, Zhang, Della Rocca, Joseph, Schachter, Joel B, Hesk, David, Telan-Choing, Florestina, Struyk, Arie, Sur, Cyrille, Celen, Sofie, Serdons, Kim, Bormans, Guy, Vandenbulcke, Mathieu, Vandenberghe, Rik, De Hoon, Jan, Koole, Michel, Van Laere, Koen, Declercq, Ruben, Reynders, Tom, Abbas, Walji, Hostetler, Eric D, Evelhoch, Jeffrey
Published in Alzheimer's & dementia (01.07.2016)
Published in Alzheimer's & dementia (01.07.2016)
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Triazolinone Biphenylsulfonamides as Angiotensin II Receptor Antagonists with High Affinity for Both the AT1 and AT2 Subtypes
Chang, Linda L, Ashton, Wallace T, Flanagan, Kelly L, Chen, Tsing-Bau, O'Malley, Stacey S, Zingaro, Gloria J, Siegl, Peter K. S, Kivlighn, Salah D, Lotti, Victor J
Published in Journal of medicinal chemistry (01.12.1994)
Published in Journal of medicinal chemistry (01.12.1994)
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De Novo Design of a Novel Oxazolidinone Analogue as a Potent and Selective α1A Adrenergic Receptor Antagonist with High Oral Bioavailability
Lagu, Bharat, Tian, Dake, Jeon, Yoon, Li, Chao, Wetzel, John M, Nagarathnam, Dhanapalan, Shen, Quanrong, Forray, Carlos, Chang, Raymond S. L, Broten, Theodore P, Ransom, Richard W, Chan, Tsing-Bao, O'Malley, Stacey S, Schorn, Terry W, Rodrigues, A. David, Kassahun, Kelem, Pettibone, Douglas J, Freidinger, Roger, Gluchowski, Charles
Published in Journal of medicinal chemistry (27.07.2000)
Published in Journal of medicinal chemistry (27.07.2000)
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In Vitro and in Vivo Evaluation of Dihydropyrimidinone C-5 Amides as Potent and Selective α1A Receptor Antagonists for the Treatment of Benign Prostatic Hyperplasia
Barrow, James C, Nantermet, Philippe G, Selnick, Harold G, Glass, Kristen L, Rittle, Kenneth E, Gilbert, Kevin F, Steele, Thomas G, Homnick, Carl F, Freidinger, Roger M, Ransom, Rick W, Kling, Paul, Reiss, Duane, Broten, Theodore P, Schorn, Terry W, Chang, Raymond S. L, O'Malley, Stacey S, Olah, Timothy V, Ellis, Joan D, Barrish, Andrea, Kassahun, Kelem, Leppert, Paula, Nagarathnam, Dhanapalan, Forray, Carlos
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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Characterization of specific binding of [formula omitted]L-762,459, a selective α1A-adrenoceptor radioligand to rat and human tissues
O'Malley, Stacey S, Chen, Tsing B, Francis, Barbara E, Gibson, Raymond E, Burns, H.Donald, DiSalvo, Jerry, Bayne, Marvin L, Wetzel, John M, Nagarathnam, Dhanapalan, Marzabadi, Mohammad, Gluchowski, Charles, Chang, Raymond S.L
Published in European journal of pharmacology (01.05.1998)
Published in European journal of pharmacology (01.05.1998)
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