A Phase I, First‐in‐Human Study of GSK2849330, an Anti‐HER3 Monoclonal Antibody, in HER3‐Expressing Solid Tumors
Gan, Hui K., Millward, Michael, Jalving, Mathilde, Garrido‐Laguna, Ignacio, Lickliter, Jason D., Schellens, Jan H.M., Lolkema, Martijn P., Van Herpen, Carla L.M., Hug, Bruce, Tang, Lihua, O'Connor‐Semmes, Robin, Gagnon, Robert, Ellis, Catherine, Ganji, Gopinath, Matheny, Christopher, Drilon, Alexander
Published in The oncologist (Dayton, Ohio) (01.10.2021)
Published in The oncologist (Dayton, Ohio) (01.10.2021)
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Pharmacokinetics and ADME Characterization of Intravenous and Oral [ 14 C]-Linerixibat in Healthy Male Volunteers
Zamek-Gliszczynski, Maciej J, Kenworthy, David, Bershas, David A, Sanghvi, Mitesh, Pereira, Adrian I, Mudunuru, Jennypher, Crossman, Lee, Pirhalla, Jill L, Thorpe, Karl M, Dennison, Jeremy M T J, McLaughlin, Megan M, Allinder, Matthew, Swift, Brandon, O'Connor-Semmes, Robin L, Young, Graeme C
Published in Drug metabolism and disposition (01.12.2021)
Published in Drug metabolism and disposition (01.12.2021)
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Total body skeletal muscle mass: estimation by creatine (methyl-d3) dilution in humans
Clark, Richard V, Walker, Ann C, O'Connor-Semmes, Robin L, Leonard, Michael S, Miller, Ram R, Stimpson, Stephen A, Turner, Scott M, Ravussin, Eric, Cefalu, William T, Hellerstein, Marc K, Evans, William J
Published in Journal of applied physiology (1985) (15.06.2014)
Published in Journal of applied physiology (1985) (15.06.2014)
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Remogliflozin Etabonate, a Selective Inhibitor of the Sodium-Glucose Transporter 2, Improves Serum Glucose Profiles in Type 1 Diabetes
MUDALIAR, Sunder, ARMSTRONG, Debra A, MAVIAN, Annie A, O'CONNOR-SEMMES, Robin, MYDLOW, Patricia K, YE, June, HUSSEY, Elizabeth K, NUNEZ, Derek J, HENRY, Robert R, DOBBINS, Robert L
Published in Diabetes care (01.11.2012)
Published in Diabetes care (01.11.2012)
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Single-dose pharmacokinetics and pharmacodynamics of sergliflozin etabonate, a novel inhibitor of glucose reabsorption, in healthy volunteers and patients with type 2 diabetes mellitus
Hussey, Elizabeth K, Clark, Richard V, Amin, Dipti M, Kipnes, Mark S, O'Connor-Semmes, Robin L, O'Driscoll, Eilis C, Leong, Jenny, Murray, Sharon C, Dobbins, Robert L, Layko, Debbi, Nunez, Derek J R
Published in Journal of clinical pharmacology (01.06.2010)
Published in Journal of clinical pharmacology (01.06.2010)
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Multiple-dose pharmacokinetics and pharmacodynamics of sergliflozin etabonate, a novel inhibitor of glucose reabsorption, in healthy overweight and obese subjects: a randomized double-blind study
Hussey, Elizabeth K, Dobbins, Robert L, Stoltz, Randall R, Stockman, Nancy L, O'Connor-Semmes, Robin L, Kapur, Anita, Murray, Sharon C, Layko, Debbi, Nunez, Derek J R
Published in Journal of clinical pharmacology (01.06.2010)
Published in Journal of clinical pharmacology (01.06.2010)
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Journal Article
First‐in‐Human Studies for a Selective RET Tyrosine Kinase Inhibitor, GSK3179106, to Investigate the Safety, Tolerability, and Pharmacokinetics in Healthy Volunteers
Cooper, Melisa, O'Connor‐Semmes, Robin, Reedy, Beth Ann, Hacquoil, Kimberley, Gorycki, Peter, Pannullo, Kristen, Verticelli, Adeline, Shakib, Sepehr
Published in Clinical pharmacology in drug development (01.02.2019)
Published in Clinical pharmacology in drug development (01.02.2019)
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Assessment of the drug interaction risk for remogliflozin etabonate, a sodium-dependent glucose cotransporter-2 inhibitor: evidence from in vitro, human mass balance, and ketoconazole interaction studies
Sigafoos, James F, Bowers, Gary D, Castellino, Stephen, Culp, Amanda G, Wagner, David S, Reese, Melinda J, Humphreys, Joan E, Hussey, Elizabeth K, O'Connor Semmes, Robin L, Kapur, Anita, Tao, Wenli, Dobbins, Robert L, Polli, Joseph W
Published in Drug metabolism and disposition (01.11.2012)
Published in Drug metabolism and disposition (01.11.2012)
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Journal Article
Creatine ( methyl-d 3 ) dilution in urine for estimation of total body skeletal muscle mass: accuracy and variability vs. MRI and DXA
Clark, Richard V, Walker, Ann C, Miller, Ram R, O'Connor-Semmes, Robin L, Ravussin, Eric, Cefalu, William T
Published in Journal of applied physiology (1985) (01.01.2018)
Published in Journal of applied physiology (1985) (01.01.2018)
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Journal Article
Assessment of safety and tolerability of remogliflozin etabonate (GSK189075) when administered with total daily dose of 2000 mg of metformin
Dobbins, Robert, Hussey, Elizabeth K, O'Connor-Semmes, Robin, Andrews, Susan, Tao, Wenli, Wilkison, William O, Cheatham, Bentley, Sagar, Katare, Hanmant, Barkate
Published in BMC pharmacology & toxicology (13.06.2021)
Published in BMC pharmacology & toxicology (13.06.2021)
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Journal Article
Effect of ranitidine on the pharmacokinetics of triazolam and alpha-hydroxytriazolam in both young (19-60 years) and older (61-78 years) people
O'Connor-Semmes, R L, Kersey, K, Williams, D H, Lam, R, Koch, K M
Published in Clinical pharmacology and therapeutics (01.08.2001)
Published in Clinical pharmacology and therapeutics (01.08.2001)
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First human dose-escalation study with remogliflozin etabonate, a selective inhibitor of the sodium-glucose transporter 2 (SGLT2), in healthy subjects and in subjects with type 2 diabetes mellitus
Kapur, Anita, O'Connor-Semmes, Robin, Hussey, Elizabeth K, Dobbins, Robert L, Tao, Wenli, Hompesch, Marcus, Smith, Glenn A, Polli, Joseph W, James, Jr, Charles D, Mikoshiba, Imao, Nunez, Derek J
Published in BMC pharmacology & toxicology (13.05.2013)
Published in BMC pharmacology & toxicology (13.05.2013)
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Journal Article
Stereoselective Pharmacokinetics of Chlorpheniramine and the Effect of Ranitidine
Koch, Kevin M., O’Connor-Semmes, Robin L., Davis, Ian M., Yin, Yin
Published in Journal of pharmaceutical sciences (01.09.1998)
Published in Journal of pharmaceutical sciences (01.09.1998)
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Journal Article
Pharmacokinetics and Pharmacodynamics of the SGLT2 Inhibitor Remogliflozin Etabonate in Subjects with Mild and Moderate Renal Impairment
O'Connor-Semmes, Robin, Walker, Susan, Kapur, Anita, Hussey, Elizabeth K, Ye, June, Wang-Smith, Laurene, Tao, Wenli, Dobbins, Robert L, Cheatham, Bentley, Wilkison, William O
Published in Drug metabolism and disposition (01.07.2015)
Published in Drug metabolism and disposition (01.07.2015)
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Journal Article
Safety, pharmacokinetics and pharmacodynamics of remogliflozin etabonate, a novel SGLT2 inhibitor, and metformin when co-administered in subjects with type 2 diabetes mellitus
Hussey, Elizabeth K, Kapur, Anita, O'Connor-Semmes, Robin, Tao, Wenli, Rafferty, Bryan, Polli, Joseph W, James, Jr, Charles D, Dobbins, Robert L
Published in BMC pharmacology & toxicology (30.04.2013)
Published in BMC pharmacology & toxicology (30.04.2013)
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Journal Article
Effect of oral CCK-1 agonist GI181771X on fasting and postprandial gastric functions in healthy volunteers
Castillo, Emma Janet, Delgado-Aros, Silvia, Camilleri, Michael, Burton, Duane, Stephens, Debra, O'Connor-Semmes, Robin, Walker, Ann, Shachoy-Clark, Anne, Zinsmeister, Alan R
Published in American journal of physiology: Gastrointestinal and liver physiology (01.08.2004)
Published in American journal of physiology: Gastrointestinal and liver physiology (01.08.2004)
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Journal Article
Effect of oral CCK-1 agonist GI181771X on fasting and postprandial gastric functions in healthy volunteers
CASTILLO, Emma Janet, DELGADO-AROS, Silvia, CAMILLERI, Michael, BURTON, Duane, STEPHENS, Debra, O'CONNOR-SEMMES, Robin, WALKER, Ann, SHACHOY-CLARK, Anne, ZINSMEISTER, Alan R
Published in American journal of physiology: Gastrointestinal and liver physiology (01.08.2004)
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Published in American journal of physiology: Gastrointestinal and liver physiology (01.08.2004)
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