Hinge Binder Scaffold Hopping Identifies Potent Calcium/Calmodulin-Dependent Protein Kinase Kinase 2 (CAMKK2) Inhibitor Chemotypes
Eduful, Benjamin J, O’Byrne, Sean N, Temme, Louisa, Asquith, Christopher R. M, Liang, Yi, Picado, Alfredo, Pilotte, Joseph R, Hossain, Mohammad Anwar, Wells, Carrow I, Zuercher, William J, Catta-Preta, Carolina M. C, Zonzini Ramos, Priscila, Santiago, André de S, Couñago, Rafael M, Langendorf, Christopher G, Nay, Kévin, Oakhill, Jonathan S, Pulliam, Thomas L, Lin, Chenchu, Awad, Dominik, Willson, Timothy M, Frigo, Daniel E, Scott, John W, Drewry, David H
Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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In Depth Analysis of Kinase Cross Screening Data to Identify CAMKK2 Inhibitory Scaffolds
O'Byrne, Sean N, Scott, John W, Pilotte, Joseph R, Santiago, André da S, Langendorf, Christopher G, Oakhill, Jonathan S, Eduful, Benjamin J, Couñago, Rafael M, Wells, Carrow I, Zuercher, William J, Willson, Timothy M, Drewry, David H
Published in Molecules (Basel, Switzerland) (13.01.2020)
Published in Molecules (Basel, Switzerland) (13.01.2020)
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