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Discovery of (pyridin-4-yl)-2H-tetrazole as a novel scaffold to identify highly selective matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis
SCHNUTE, Mark E, O'BRIEN, Patrick M, CARROLL, Jeffery N, PATT, William C, SHIEH, Huey S, COLLINS, Brandon, PAVLOVSKY, Alexander G, PALMQUIST, Katherine E, ASTON, Karl W, HITCHCOCK, Jeffrey, ROGERS, Michael D, MCDONALD, Joseph, NAHRA, Joe, JOHNSON, Adam R, MUNIE, Grace E, WITTWER, Arthur J, MAN, Chiu-Fai, SETTLE, Steven L, NEMIROVSKIY, Olga, VICKERY, Lillian E, AGAWAL, Arun, DYER, Richard D, SUNYER, Teresa, MORRIS, Mark, HOWARD ROARK, W, HANAU, Cathleen E, RUMINSKI, Peter G, SCHOLTEN, Jeffrey A, FLETCHER, Theresa R, HAMPER, Bruce C
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Structure−Activity Relationships and Pharmacokinetic Analysis for a Series of Potent, Systemically Available Biphenylsulfonamide Matrix Metalloproteinase Inhibitors
O'Brien, Patrick M, Ortwine, Daniel F, Pavlovsky, Alexander G, Picard, Joseph A, Sliskovic, Drago R, Roth, Bruce D, Dyer, Richard D, Johnson, Linda L, Man, Chiu Fai, Hallak, Hussein
Published in Journal of medicinal chemistry (27.01.2000)
Published in Journal of medicinal chemistry (27.01.2000)
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Subscapularis Function After Total Shoulder Arthroplasty Using Lesser Tuberosity Osteotomy or Tenotomy
OʼBrien, Patrick M, Kazanjian, Jack E, Kelly, 2nd, James D, Hobgood, E Rhett
Published in Journal of the American Academy of Orthopaedic Surgeons. Global research & reviews (01.05.2020)
Published in Journal of the American Academy of Orthopaedic Surgeons. Global research & reviews (01.05.2020)
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Emergency medicine and public health: New steps in old directions
Pollock, Daniel A., Lowery, Douglas W., O'Brien, Patrick M.
Published in Annals of emergency medicine (01.12.2001)
Published in Annals of emergency medicine (01.12.2001)
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Stereoselective binding of an enantiomeric pair of stromelysin-1 inhibitors caused by conformational entropy factors
Parker, Matthew H, Ortwine, Daniel F, O'Brien, Patrick M, Lunney, Elizabeth A, Banotai, Craig A, Mueller, William T, McConnell, Patrick, Brouillette, Christie G
Published in Bioorganic & medicinal chemistry letters (06.11.2000)
Published in Bioorganic & medicinal chemistry letters (06.11.2000)
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Antiatherosclerotic activity of inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase in cholesterol-fed rabbits: a biochemical and morphological evaluation
Bocan, Thomas M.A., Mazur, Michelle J., Bak Mueller, Sandra, Brown, Edie Quenby, Sliskovic, D.Robert, O'Brien, Patrick M., Creswell, Mark W., Lee, Helen, Uhlendorf, Paul D., Roth, Bruce D., Newton, Roger S.
Published in Atherosclerosis (01.11.1994)
Published in Atherosclerosis (01.11.1994)
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Inhibitors of Acyl-CoA:Cholesterol O-Acyltransferase. 17. Structure−Activity Relationships of Several Series of Compounds Derived from N-Chlorosulfonyl Isocyanate
Picard, Joseph A, O'Brien, Patrick M, Sliskovic, Drago R, Anderson, Maureen K, Bousley, Richard F, Hamelehle, Katherine L, Krause, Brian R, Stanfield, Richard L
Published in Journal of medicinal chemistry (15.03.1996)
Published in Journal of medicinal chemistry (15.03.1996)
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Inhibitors of Acyl-CoA:Cholesterol O-Acyl Transferase (ACAT) as Hypocholesterolemic Agents. 8. Incorporation of Amide or Amine Functionalities into a Series of Disubstituted Ureas and Carbamates. Effects on ACAT Inhibition in vitro and Efficacy in vivo
O'Brien, Patrick M, Sliskovic, Drago R, Blankley, C. John, Roth, Bruce. D, Wilson, Michael W, Hamelehle, Katherine L, Krause, Brian R, Stanfield, Richard L
Published in Journal of medicinal chemistry (01.06.1994)
Published in Journal of medicinal chemistry (01.06.1994)
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Inhibitors of Acyl-CoA:Cholesterol O-Acyltransferase. Synthesis and Pharmacological Activity of (±)-2-Dodecyl-α-phenyl-N-(2,4,6-trimethoxyphenyl)-2H-tetrazole-5-acetamide and Structurally Related Tetrazole Amide Derivatives
O'Brien, Patrick M, Sliskovic, Drago R, Picard, Joseph A, Lee, Helen T, Purchase, Claude F, Roth, Bruce D, White, Andrew D, Anderson, Maureen, Mueller, Sandra Bak, Bocan, Thomas, Bousley, Richard, Hamelehle, Katherine L, Homan, Reynold, Lee, Peter, Krause, Brian R, Reindel, J. F, Turluck, Daniel
Published in Journal of medicinal chemistry (07.06.1996)
Published in Journal of medicinal chemistry (07.06.1996)
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α-Substituted Malonester Amides: Tools To Define the Relationship between ACAT Inhibition and Adrenal Toxicity
Sliskovic, Drago R, Picard, Joseph A, O'Brien, Patrick M, Liao, Peggy, Roark, W. Howard, Roth, Bruce D, Anderson, Maureen A, Mueller, Sandra Bak, Bocan, Thomas M. A, Bousley, Richard F, Hamelehle, Katherine L, Homan, Reynold, Reindel, James F, Stanfield, Richard L, Turluck, Daniel, Krause, Brian R
Published in Journal of medicinal chemistry (26.02.1998)
Published in Journal of medicinal chemistry (26.02.1998)
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Transparency as a means to rebuild trust within the Church: a case study in how Catholic dioceses and eparchies in the United States have responded to the clergy sex abuse crisis
O'Brien, Patrick M.
Published in Church, Communication and Culture: Special issue: Trust in Institutions (01.09.2020)
Published in Church, Communication and Culture: Special issue: Trust in Institutions (01.09.2020)
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Risk Factors for Early Failure of Surgical Amputations: An Analysis of 8,878 Isolated Lower Extremity Amputation Procedures
O'Brien, Patrick J., MD, Cox, Mitchell W., MD, FACS, Shortell, Cynthia K., MD, FACS, Scarborough, John E., MD, FACS
Published in Journal of the American College of Surgeons (01.04.2013)
Published in Journal of the American College of Surgeons (01.04.2013)
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Analysis of Infection Risk following Covered Stent Exclusion of Pseudoaneurysms in Prosthetic Arteriovenous Hemodialysis Access Grafts
Kim, Charles Y., MD, Guevara, Carlos J., MD, Engstrom, Bjorn I., MD, Gage, Shawn M., PA, O'Brien, Patrick J., MD, Miller, Michael J., MD, Suhocki, Paul V., MD, Lawson, Jeffrey H., MD, Smith, Tony P., MD
Published in Journal of vascular and interventional radiology (2012)
Published in Journal of vascular and interventional radiology (2012)
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