Novel gut-based pharmacology of metformin in patients with type 2 diabetes mellitus
Napolitano, Antonella, Miller, Sam, Nicholls, Andrew W, Baker, David, Van Horn, Stephanie, Thomas, Elizabeth, Rajpal, Deepak, Spivak, Aaron, Brown, James R, Nunez, Derek J
Published in PloS one (02.07.2014)
Published in PloS one (02.07.2014)
Get full text
Journal Article
A Systematic Review of Biomarkers and Risk of Incident Type 2 Diabetes: An Overview of Epidemiological, Prediction and Aetiological Research Literature
Abbasi, Ali, Sahlqvist, Anna-Stina, Lotta, Luca, Brosnan, Julia M, Vollenweider, Peter, Giabbanelli, Philippe, Nunez, Derek J, Waterworth, Dawn, Scott, Robert A, Langenberg, Claudia, Wareham, Nicholas J
Published in PloS one (27.10.2016)
Published in PloS one (27.10.2016)
Get full text
Journal Article
Gut hormone pharmacology of a novel GPR119 agonist (GSK1292263), metformin, and sitagliptin in type 2 diabetes mellitus: results from two randomized studies
Nunez, Derek J, Bush, Mark A, Collins, David A, McMullen, Susan L, Gillmor, Dawn, Apseloff, Glen, Atiee, George, Corsino, Leonor, Morrow, Linda, Feldman, Paul L
Published in PloS one (03.04.2014)
Published in PloS one (03.04.2014)
Get full text
Journal Article
Remogliflozin Etabonate, a Selective Inhibitor of the Sodium-Glucose Transporter 2, Improves Serum Glucose Profiles in Type 1 Diabetes
MUDALIAR, Sunder, ARMSTRONG, Debra A, MAVIAN, Annie A, O'CONNOR-SEMMES, Robin, MYDLOW, Patricia K, YE, June, HUSSEY, Elizabeth K, NUNEZ, Derek J, HENRY, Robert R, DOBBINS, Robert L
Published in Diabetes care (01.11.2012)
Published in Diabetes care (01.11.2012)
Get full text
Journal Article
Assessment of plasma acylcarnitines before and after weight loss in obese subjects
Schooneman, Marieke G., Napolitano, Antonella, Houten, Sander M., Ambler, Graeme K., Murgatroyd, Peter R., Miller, Sam R., Hollak, Carla E.M., Tan, Chong Y., Virtue, Samuel, Vidal-Puig, Antonio, Nunez, Derek J., Soeters, Maarten R.
Published in Archives of biochemistry and biophysics (15.09.2016)
Published in Archives of biochemistry and biophysics (15.09.2016)
Get full text
Journal Article
Weight and Glucose Reduction Observed with a Combination of Nutritional Agents in Rodent Models Does Not Translate to Humans in a Randomized Clinical Trial with Healthy Volunteers and Subjects with Type 2 Diabetes
Hodge, Rebecca J, Paulik, Mark A, Walker, Ann, Boucheron, Joyce A, McMullen, Susan L, Gillmor, Dawn S, Nunez, Derek J
Published in PloS one (19.04.2016)
Published in PloS one (19.04.2016)
Get full text
Journal Article
Multiple-dose pharmacokinetics and pharmacodynamics of sergliflozin etabonate, a novel inhibitor of glucose reabsorption, in healthy overweight and obese subjects: a randomized double-blind study
Hussey, Elizabeth K, Dobbins, Robert L, Stoltz, Randall R, Stockman, Nancy L, O'Connor-Semmes, Robin L, Kapur, Anita, Murray, Sharon C, Layko, Debbi, Nunez, Derek J R
Published in Journal of clinical pharmacology (01.06.2010)
Published in Journal of clinical pharmacology (01.06.2010)
Get more information
Journal Article
Validation of a Quantitative Magnetic Resonance Method for Measuring Human Body Composition
Napolitano, Antonella, Miller, Sam R, Murgatroyd, Peter R, Coward, W. Andrew, Wright, Antony, Finer, Nick, De Bruin, Tjerk W, Bullmore, Edward T, Nunez, Derek, J
Published in Obesity (Silver Spring, Md.) (01.01.2008)
Published in Obesity (Silver Spring, Md.) (01.01.2008)
Get full text
Journal Article
Single-dose pharmacokinetics and pharmacodynamics of sergliflozin etabonate, a novel inhibitor of glucose reabsorption, in healthy volunteers and patients with type 2 diabetes mellitus
Hussey, Elizabeth K, Clark, Richard V, Amin, Dipti M, Kipnes, Mark S, O'Connor-Semmes, Robin L, O'Driscoll, Eilis C, Leong, Jenny, Murray, Sharon C, Dobbins, Robert L, Layko, Debbi, Nunez, Derek J R
Published in Journal of clinical pharmacology (01.06.2010)
Published in Journal of clinical pharmacology (01.06.2010)
Get more information
Journal Article
Reduced T2 values in soleus muscle of patients with type 2 diabetes mellitus
Zuo, Chun S, Sung, Young-Hoon, Simonson, Donald C, Habecker, Erin, Wang, Jian, Haws, Charlotte, Villafuerte, Rosemond A, Henry, Michael E, Dobbins, Robert L, Hodge, Rebecca J, Nunez, Derek J R, Renshaw, Perry F
Published in PloS one (26.11.2012)
Published in PloS one (26.11.2012)
Get full text
Journal Article
Factors influencing longitudinal changes of circulating liver enzyme concentrations in subjects randomized to placebo in four clinical trials
Nunez, Derek J, Alexander, Myriam, Yerges-Armstrong, Laura, Singh, Gurparkash, Byttebier, Geert, Fabbrini, Elisa, Waterworth, Dawn, Meininger, Gary, Galwey, Nicholas, Wallentin, Lars, White, Harvey D, Vannieuwenhuyse, Bart, Alazawi, William, Kendrick, Stuart, Sattar, Naveed, Ferrannini, Ele
Published in American journal of physiology: Gastrointestinal and liver physiology (01.03.2019)
Published in American journal of physiology: Gastrointestinal and liver physiology (01.03.2019)
Get full text
Journal Article
Assessment of Acute and Chronic Pharmacological Effects on Energy Expenditure and Macronutrient Oxidation in Humans: Responses to Ephedrine
Murgatroyd, Peter R., Hussey, Elizabeth K., Napolitano, Antonella, Nunez, Derek J. R., O'Rahilly, Steve, Dobbins, Robert, Finer, Nick
Published in Journal of Obesity (01.01.2011)
Published in Journal of Obesity (01.01.2011)
Get full text
Journal Article
Evaluation of drug interactions of GSK1292263 (a GPR119 agonist) with statins: from in vitro data to clinical study design
Polli, Joseph W., Hussey, Elizabeth, Bush, Mark, Generaux, Grant, Smith, Glenn, Collins, David, McMullen, Susan, Turner, Nancy, Nunez, Derek J.
Published in Xenobiotica (01.06.2013)
Published in Xenobiotica (01.06.2013)
Get full text
Journal Article
Safety, Pharmacokinetics, and Pharmacodynamic Effects of a Selective TGR5 Agonist, SB-756050, in Type 2 Diabetes
Hodge, Rebecca J, Lin, Jiang, Vasist Johnson, Lakshmi S, Gould, Elizabeth P, Bowers, Gary D, Nunez, Derek J
Published in Clinical pharmacology in drug development (01.07.2013)
Published in Clinical pharmacology in drug development (01.07.2013)
Get more information
Journal Article
Quantitative Magnetic Resonance (QMR) for Longitudinal Evaluation of Body Composition Changes With Two Dietary Regimens
Myint, Khin Swe, Napolitano, Antonella, Miller, Sam R, Murgatroyd, Peter R, Elkhawad, Maysoon, Nunez, Derek J.R, Finer, Nick
Published in Obesity (Silver Spring, Md.) (01.02.2010)
Published in Obesity (Silver Spring, Md.) (01.02.2010)
Get full text
Journal Article
Pharmacokinetics and Tolerability of Exenatide Delivered by 7-Day Continuous Subcutaneous Infusion in Healthy Volunteers
Vlasakakis, Georgios, Johnson, Susan L., Lin, Jiang, Yao, Xiaozhou, Gruenloh, Christopher J., Chism, John P., Nunez, Derek J.
Published in Advances in therapy (01.07.2015)
Published in Advances in therapy (01.07.2015)
Get full text
Journal Article
Exploring glycosuria as a mechanism for weight and fat mass reduction. A pilot study with remogliflozin etabonate and sergliflozin etabonate in healthy obese subjects
Napolitano, Antonella, Miller, Sam, Murgatroyd, Peter R, Hussey, Elizabeth, Dobbins, Robert L, Bullmore, Edward T, Nunez, Derek J.R
Published in Journal of clinical & translational endocrinology (01.03.2014)
Published in Journal of clinical & translational endocrinology (01.03.2014)
Get full text
Journal Article
First human dose-escalation study with remogliflozin etabonate, a selective inhibitor of the sodium-glucose transporter 2 (SGLT2), in healthy subjects and in subjects with type 2 diabetes mellitus
Kapur, Anita, O'Connor-Semmes, Robin, Hussey, Elizabeth K, Dobbins, Robert L, Tao, Wenli, Hompesch, Marcus, Smith, Glenn A, Polli, Joseph W, James, Jr, Charles D, Mikoshiba, Imao, Nunez, Derek J
Published in BMC pharmacology & toxicology (13.05.2013)
Published in BMC pharmacology & toxicology (13.05.2013)
Get full text
Journal Article