Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H3PO4
Reeves, Jonathan T, Fandrick, Daniel R, Tan, Zhulin, Song, Jinhua J, Rodriguez, Sonia, Qu, Bo, Kim, Soojin, Niemeier, Oliver, Li, Zhibin, Byrne, Denis, Campbell, Scot, Chitroda, Ashish, DeCroos, Phil, Fachinger, Thomas, Fuchs, Victor, Gonnella, Nina C, Grinberg, Nelu, Haddad, Nizar, Jäger, Burkhard, Lee, Heewon, Lorenz, Jon C, Ma, Shengli, Narayanan, Bikshandarkoil A, Nummy, Larry J, Premasiri, Ajith, Roschangar, Frank, Sarvestani, Max, Shen, Sherry, Spinelli, Earl, Sun, Xiufeng, Varsolona, Richard J, Yee, Nathan, Brenner, Michael, Senanayake, Chris H
Published in Journal of organic chemistry (19.04.2013)
Published in Journal of organic chemistry (19.04.2013)
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Journal Article
A Scalable and Regioselective Synthesis of 2‑Difluoromethyl Pyridines from Commodity Chemicals
Desrosiers, Jean-Nicolas, Kelly, Christopher B, Fandrick, Daniel R, Nummy, Larry, Campbell, Scot J, Wei, Xudong, Sarvestani, Max, Lee, Heewon, Sienkiewicz, Alexander, Sanyal, Sanjit, Zeng, Xingzhong, Grinberg, Nelu, Ma, Shengli, Song, Jinhua J, Senanayake, Chris H
Published in Organic letters (21.03.2014)
Published in Organic letters (21.03.2014)
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Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT-2, Utilizing an AlCl3-Promoted Si lane Reduction of a beta-Glycopyranoside
Wang, Xiao-jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H.
Published in Organic letters (15.08.2014)
Published in Organic letters (15.08.2014)
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Journal Article
Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT-2, Utilizing an AlCl3‑Promoted Silane Reduction of a β‑Glycopyranoside
Wang, Xiao-jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H
Published in Organic letters (15.08.2014)
Published in Organic letters (15.08.2014)
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Journal Article
Process Development of the BACE Inhibitors BI 1147560 BS and BI 1181181 MZ
Li, Guisheng, Tan, Zhulin, Xu, Yibo, Sidhu, Kanwar P. S., Qu, Bo, Herbage, Melissa A., Eriksson, Magnus C., Zeng, Xingzhong, Busacca, Carl A., Desrosiers, Jean-Nicolas, Hampel, Thomas, Niemeier, Oliver, Reichel, Carsten, Quynh Dang, Mai Thi, Schoerer, Marvin, Kemmer, Dirk, Eick, Melanie, Werle, Holger, Kim, Soojin, Li, Zhibin, Venkatraman, Shankar, Jia, Lanqi, Claremon, David A., Fuchs, Klaus, Heine, Niklas, Byrne, Denis, Narayanan, Bikshandarkoil, Sarvestani, Max, Johnson, Joe, Premasiri, Ajith, Nummy, Larry J., Lorenz, Jon C., Haddad, Nizar, Gonnella, Nina C., Pennino, Scott, Krawiec, Mariusz, Senanayake, Chris H., Buono, Frederic, Lee, Heewon, Hossain, Azad, Song, Jinhua J., Reeves, Jonathan T.
Published in Organic process research & development (16.12.2022)
Published in Organic process research & development (16.12.2022)
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Journal Article
Development of a Large-Scale Asymmetric Process for tert-Butanesulfinamide
DeCroos, Philomen, Han, Zhengxu S, Sidhu, Kanwar, Lorenz, Jon, Nummy, Larry, Byrne, Denis, Qu, Bo, Xu, Yibo, Wu, Ling, Lee, Heewon, Roschangar, Frank, Song, Jinhua J, Senanayake, Chris H
Published in Organic process research & development (15.02.2019)
Published in Organic process research & development (15.02.2019)
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Journal Article
Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT-2, Utilizing an AlCl 3 -Promoted Silane Reduction of a β-Glycopyranoside
Wang, Xiao-jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H.
Published in Organic letters (15.08.2014)
Published in Organic letters (15.08.2014)
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Journal Article
The P‑Chiral Phosphane Ligand (MeO-BIBOP) for Efficient and Practical Large-Scale Rh-Catalyzed Asymmetric Hydrogenation of N‑Acetyl Enamides with High TONs
Li, Wenjie, Rodriguez, Sonia, Duran, Adil, Sun, Xiufeng, Tang, Wenjun, Premasiri, Ajith, Wang, Jun, Sidhu, Kanwar, Patel, Nitinchandra D, Savoie, Jolaine, Qu, Bo, Lee, Heewon, Haddad, Nizar, Lorenz, Jon C, Nummy, Larry, Hossain, Azad, Yee, Nathan, Lu, Bruce, Senanayake, Chris H
Published in Organic process research & development (16.08.2013)
Published in Organic process research & development (16.08.2013)
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Journal Article
Synthesis of potent lymphocyte function-associated antigen-1 inhibitors labeled with carbon-14 and deuterium, part 1
Latli, Bachir, Byrne, Denis, Nummy, Larry, Krishnamurthy, Dhileepkumar, Senanayake, Chris H.
Published in Journal of labelled compounds & radiopharmaceuticals (01.10.2011)
Published in Journal of labelled compounds & radiopharmaceuticals (01.10.2011)
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Journal Article
Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H 3 PO 4
Reeves, Jonathan T., Fandrick, Daniel R., Tan, Zhulin, Song, Jinhua J., Rodriguez, Sonia, Qu, Bo, Kim, Soojin, Niemeier, Oliver, Li, Zhibin, Byrne, Denis, Campbell, Scot, Chitroda, Ashish, DeCroos, Phil, Fachinger, Thomas, Fuchs, Victor, Gonnella, Nina C., Grinberg, Nelu, Haddad, Nizar, Jäger, Burkhard, Lee, Heewon, Lorenz, Jon C., Ma, Shengli, Narayanan, Bikshandarkoil A., Nummy, Larry J., Premasiri, Ajith, Roschangar, Frank, Sarvestani, Max, Shen, Sherry, Spinelli, Earl, Sun, Xiufeng, Varsolona, Richard J., Yee, Nathan, Brenner, Michael, Senanayake, Chris H.
Published in Journal of organic chemistry (19.04.2013)
Published in Journal of organic chemistry (19.04.2013)
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ChemInform Abstract: Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT‐2, Utilizing an AlCl 3 ‐Promoted Silane Reduction of a β‐Glycopyranoside
Wang, Xiao‐jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H.
Published in ChemInform (01.02.2015)
Published in ChemInform (01.02.2015)
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Journal Article
ChemInform Abstract: Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT-2, Utilizing an AlCl3-Promoted Silane Reduction of a [beta]-Glycopyranoside
Wang, Xiao-jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H
Published in ChemInform (01.02.2015)
Published in ChemInform (01.02.2015)
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Journal Article
ChemInform Abstract: Efficient Synthesis of Empagliflozin, an Inhibitor of SGLT-2, Utilizing an AlCl3-Promoted Silane Reduction of a β-Glycopyranoside
Wang, Xiao-jun, Zhang, Li, Byrne, Denis, Nummy, Larry, Weber, Dirk, Krishnamurthy, Dhileep, Yee, Nathan, Senanayake, Chris H.
Published in ChemInform (01.02.2015)
Published in ChemInform (01.02.2015)
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