Stereoselective Synthesis of Baloxavir Marboxil Using Diastereoselective Cyclization and Photoredox Decarboxylation of l‑Serine
Okamoto, Kazuya, Ueno, Tatsuhiko, Hato, Yoshio, Kawaguchi, Yasunori, Hakogi, Toshikazu, Majima, Shohei, Ohara, Takafumi, Hagihara, Motoyuki, Tanimoto, Norihiko, Tsuritani, Takayuki
Published in Journal of organic chemistry (19.07.2024)
Published in Journal of organic chemistry (19.07.2024)
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Carbamoyl Pyridone HIV‑1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)
Johns, Brian A, Kawasuji, Takashi, Weatherhead, Jason G, Taishi, Teruhiko, Temelkoff, David P, Yoshida, Hiroshi, Akiyama, Toshiyuki, Taoda, Yoshiyuki, Murai, Hitoshi, Kiyama, Ryuichi, Fuji, Masahiro, Tanimoto, Norihiko, Jeffrey, Jerry, Foster, Scott A, Yoshinaga, Tomokazu, Seki, Takahiro, Kobayashi, Masanori, Sato, Akihiko, Johnson, Matthew N, Garvey, Edward P, Fujiwara, Tamio
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Discovery of Atabecestat (JNJ-54861911): A Thiazine-Based β‑Amyloid Precursor Protein Cleaving Enzyme 1 Inhibitor Advanced to the Phase 2b/3 EARLY Clinical Trial
Koriyama, Yuji, Hori, Akihiro, Ito, Hisanori, Yonezawa, Shuji, Baba, Yoshiyasu, Tanimoto, Norihiko, Ueno, Tatsuhiko, Yamamoto, Shiho, Yamamoto, Takahiko, Asada, Naoya, Morimoto, Kenji, Einaru, Shunsuke, Sakai, Katsunori, Kanazu, Takushi, Matsuda, Akihiro, Yamaguchi, Yoshitaka, Oguma, Takuya, Timmers, Maarten, Tritsmans, Luc, Kusakabe, Ken-ichi, Kato, Akira, Sakaguchi, Gaku
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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P2-049 Neuroprotective effects of 2-(2-hydroxylphenyl)benzoxazol derivatives via induction of brain-derived neurotrophic factor synthesis
Hisanori Ito, Gaku Sakaguchi, Toshinaga Tsuji, Tsuyoshi Kihara, Shoei Furukawa, Norihiko Tanimoto, Akira Kato
Published in Journal of Pharmacological Sciences (2007)
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Published in Journal of Pharmacological Sciences (2007)
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Structure of photoactive yellow protein (PYP) E46Q mutant at 1.2 Å resolution suggests how Glu46 controls the spectroscopic and kinetic characteristics of PYP
Sugishima, Masakazu, Tanimoto, Norihiko, Soda, Koji, Hamada, Norio, Tokunaga, Fumio, Fukuyama, Keiichi
Published in Acta crystallographica. Section D, Biological crystallography. (01.12.2004)
Published in Acta crystallographica. Section D, Biological crystallography. (01.12.2004)
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Carbamoyl Pyridone HIV‑1 Integrase Inhibitors. 2. Bi- and Tricyclic Derivatives Result in Superior Antiviral and Pharmacokinetic Profiles
Kawasuji, Takashi, Johns, Brian A, Yoshida, Hiroshi, Weatherhead, Jason G, Akiyama, Toshiyuki, Taishi, Teruhiko, Taoda, Yoshiyuki, Mikamiyama-Iwata, Minako, Murai, Hitoshi, Kiyama, Ryuichi, Fuji, Masahiro, Tanimoto, Norihiko, Yoshinaga, Tomokazu, Seki, Takahiro, Kobayashi, Masanori, Sato, Akihiko, Garvey, Edward P, Fujiwara, Tamio
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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2-Arylimino-5,6-dihydro-4H-1,3-thiazines as a new class of cannabinoid receptor agonists. Part 3: Synthesis and activity of isosteric analogs
KAI, Hiroyuki, MORIOKA, Yasuhide, TAKAHASHI, Kohji, TANIMOTO, Norihiko, KORIYAMA, Yuji, OKAMOTO, Kazuya, HASEGAWA, Yasushi, HATTORI, Maki, KOIKE, Katsumi, CHIBA, Hiroki, SHINOHARA, Shunji, IWAMOTO, Yuka
Published in Bioorganic & medicinal chemistry (15.12.2008)
Published in Bioorganic & medicinal chemistry (15.12.2008)
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STRUCTURE-ACTIVITY RELATIONSHIP OF GLYCINOECLEPIN-A
MURAI, A, OHKITA, M, HONMA, T, HOSHI, K, TANIMOTO, N, ARAKI, S, FUKUZAWA, A
Published in Chemistry letters (01.11.1992)
Published in Chemistry letters (01.11.1992)
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A novel series of parenteral cephalosporins exhibiting potent activities against both Pseudomonas aeruginosa and other Gram-negative pathogens. Part 2: Synthesis and structure–activity relationships
Yamawaki, Kenji, Nomura, Takashi, Yasukata, Tatsuro, Tanimoto, Norihiko, Uotani, Koichi, Miwa, Hideaki, Yamano, Yoshinori, Takeda, Kei, Nishitani, Yasuhiro
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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2-Arylimino-5,6-dihydro-4 H-1,3-thiazines as a new class of cannabinoid receptor agonists. Part 3: Synthesis and activity of isosteric analogs
Kai, Hiroyuki, Morioka, Yasuhide, Koriyama, Yuji, Okamoto, Kazuya, Hasegawa, Yasushi, Hattori, Maki, Koike, Katsumi, Chiba, Hiroki, Shinohara, Shunji, Iwamoto, Yuka, Takahashi, Kohji, Tanimoto, Norihiko
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Glycinoeclepins, Natural Hatching Stimuli for the Soybean Cyst Nematode, Heterodera Glycines. II. Structural Elucidation
Masamune, Tadashi, Fukuzawa, Akio, Furusaki, Akio, Ikura, Mitsuhiko, Matsue, Hideki, Kaneko, Tatsuya, Abiko, Atsushi, Sakamoto, Noriyasu, Tanimoto, Norihiko, Murai, Akio
Published in Bulletin of the Chemical Society of Japan (1987)
Published in Bulletin of the Chemical Society of Japan (1987)
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The Effects of Diesel Exhaust Particles (DEPs) on a Murine Testis (Proceedings of the 22nd Symposium on Toxicology and Environmental Health)
YOSHIDA, Seiichi, TANIMOTO, Norihiko, NAGAO, Kenji, SUGIMOTO, Natuki, KUWABARA, Yuko, TABATA, Masako, TAKEDA, Ken, OSHIO, Shigeru, UMEDA, Takashi, MIYABARA, Yuichi, ICHINOSE, Takamichi, SAGAI, Masaru, SUGAWARA, Isamu
Published in Eisei kagaku (1997)
Published in Eisei kagaku (1997)
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Total synthesis of glycinoeclepin A
Murai, Akio, Tanimoto, Norihiko, Sakamoto, Noriyasu, Masamune, Tadashi
Published in Journal of the American Chemical Society (01.03.1988)
Published in Journal of the American Chemical Society (01.03.1988)
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Glycosidase antibodies induced to a half-chair transition-state analog
Suga, Hiroaki, Tanimoto, Norihiko, Sinskey, Anthony J, Masamune, Satoru
Published in Journal of the American Chemical Society (01.11.1994)
Published in Journal of the American Chemical Society (01.11.1994)
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Compounds exhibiting PGD 2 receptor antagonism
INAGAKI, MASANAO, MITSUMORI, SUSUMU, HIRAMATSU, YOSHIHARU, TANIMOTO, NORIHIKO
Year of Publication 29.02.2012
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Year of Publication 29.02.2012
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