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Published in Nature chemical biology (01.02.2018)
Published in Nature chemical biology (01.02.2018)
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Published in Nature chemical biology (01.04.2011)
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ERK5 kinase activity is dispensable for cellular immune response and proliferation
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Published in Proceedings of the National Academy of Sciences - PNAS (18.10.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (18.10.2016)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.2011)
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Functional Interrogation of the Kinome Using Nucleotide Acyl Phosphates
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Published in Biochemistry (Easton) (16.01.2007)
Published in Biochemistry (Easton) (16.01.2007)
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Chemoproteomic Evaluation of Target Engagement by the Cyclin-Dependent Kinase 4 and 6 Inhibitor Palbociclib Correlates with Cancer Cell Response
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Published in Biochemistry (Easton) (27.09.2016)
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Chemoproteomics Using Nucleotide Acyl Phosphates Reveals an ATP Binding Site at the Dimer Interface of Procaspase‑6
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Novel Mechanistic Class of Fatty Acid Amide Hydrolase Inhibitors with Remarkable Selectivity
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Published in Biochemistry (Easton) (13.11.2007)
Published in Biochemistry (Easton) (13.11.2007)
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Functional interrogation of kinases and other nucleotide-binding proteins
Rosenblum, Jonathan S., Nomanbhoy, Tyzoon K., Kozarich, John W.
Published in FEBS letters (27.06.2013)
Published in FEBS letters (27.06.2013)
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Discovery of PF-04457845: A Highly Potent, Orally Bioavailable, and Selective Urea FAAH Inhibitor
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Published in ACS medicinal chemistry letters (10.02.2011)
Published in ACS medicinal chemistry letters (10.02.2011)
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Pathophysiological significance and therapeutic targeting of germinal center kinase in diffuse large B-cell lymphoma
Matthews, Julie Marie, Bhatt, Shruti, Patricelli, Matthew P., Nomanbhoy, Tyzoon K., Jiang, Xiaoyu, Natkunam, Yasodha, Gentles, Andrew J., Martinez, Ezequiel, Zhu, Daxing, Chapman, Jennifer Rose, Cortizas, Elena, Shyam, Ragini, Chinichian, Shideh, Advani, Ranjana, Tan, Li, Zhang, Jianming, Choi, Hwan Geun, Tibshirani, Robert, Buhrlage, Sara J., Gratzinger, Dita, Verdun, Ramiro, Gray, Nathanael S., Lossos, Izidore S.
Published in Blood (14.07.2016)
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High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity
Zhu, Wen, Radadiya, Ashish, Bisson, Claudine, Wenzel, Sabine, Nordin, Brian E, Martínez-Márquez, Francisco, Imasaki, Tsuyoshi, Sedelnikova, Svetlana E, Coricello, Adriana, Baumann, Patrick, Berry, Alexandria H, Nomanbhoy, Tyzoon K, Kozarich, John W, Jin, Yi, Rice, David W, Takagi, Yuichiro, Richards, Nigel G J
Published in Communications biology (17.09.2019)
Published in Communications biology (17.09.2019)
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ATP Acyl Phosphate Reactivity Reveals Native Conformations of Hsp90 Paralogs and Inhibitor Target Engagement
Nordin, Brian E, Liu, Yongsheng, Aban, Arwin, Brown, Heidi E, Wu, Jiangyue, Hainley, Anna K, Rosenblum, Jonathan S, Nomanbhoy, Tyzoon K, Kozarich, John W
Published in Biochemistry (Easton) (19.05.2015)
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Identification of a Tumor Specific, Active-Site Mutation in Casein Kinase 1α by Chemical Proteomics
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Published in PloS one (31.03.2016)
Published in PloS one (31.03.2016)
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Benzothiophene piperazine and piperidine urea inhibitors of fatty acid amide hydrolase (FAAH)
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Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Correction: Identification of a Tumor Specific, Active-Site Mutation in Casein Kinase 1α by Chemical Proteomics
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Published in PloS one (2017)
Published in PloS one (2017)
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Author Correction: High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity
Zhu, Wen, Radadiya, Ashish, Bisson, Claudine, Wenzel, Sabine, Nordin, Brian E., Martínez-Márquez, Francisco, Imasaki, Tsuyoshi, Sedelnikova, Svetlana E., Coricello, Adriana, Baumann, Patrick, Berry, Alexandria H., Nomanbhoy, Tyzoon K., Kozarich, John W., Jin, Yi, Rice, David W., Takagi, Yuichiro, Richards, Nigel G. J.
Published in Communications biology (22.11.2019)
Published in Communications biology (22.11.2019)
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Published in Chemistry & biology (27.01.2012)
Published in Chemistry & biology (27.01.2012)
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In Situ Kinase Profiling Reveals Functionally Relevant Properties of Native Kinases
Patricelli, Matthew P., Nomanbhoy, Tyzoon K., Wu, Jiangyue, Brown, Heidi, Zhou, David, Zhang, Jianming, Jagannathan, Subadhra, Aban, Arwin, Okerberg, Eric, Herring, Chris, Nordin, Brian, Weissig, Helge, Yang, Qingkai, Lee, Jiing-Dwan, Gray, Nathanael S., Kozarich, John W.
Published in Chemistry & biology (24.06.2011)
Published in Chemistry & biology (24.06.2011)
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