Design, synthesis and evaluation of N-aryl-glyoxamide derivatives as structurally novel bacterial quorum sensing inhibitors
Nizalapur, Shashidhar, Kimyon, Oender, Biswas, Nripendra Nath, Gardner, Christopher R., Griffith, Renate, Rice, Scott A., Manefield, Mike, Willcox, Mark, Black, David StC, Kumar, Naresh
Published in Organic & biomolecular chemistry (01.01.2016)
Published in Organic & biomolecular chemistry (01.01.2016)
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Journal Article
Synthesis and biological evaluation of N-naphthoyl-phenylglyoxamide-based small molecular antimicrobial peptide mimics as novel antimicrobial agents and biofilm inhibitors
Nizalapur, Shashidhar, Ho, Kitty K. K., Kimyon, Oender, Yee, Eugene, Berry, Thomas, Manefield, Mike, Cranfield, Charles G., Willcox, Mark, Black, David StC, Kumar, Naresh
Published in Organic & biomolecular chemistry (14.04.2016)
Published in Organic & biomolecular chemistry (14.04.2016)
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Journal Article
Design and Synthesis of Lactams Derived from Mucochloric and Mucobromic Acids as Pseudomonas aeruginosa Quorum Sensing Inhibitors
Almohaywi, Basmah, Taunk, Aditi, Wenholz, Daniel S, Nizalapur, Shashidhar, Biswas, Nripendra N, Ho, Kitty K K, Rice, Scott A, Iskander, George, Black, David StC, Griffith, Renate, Kumar, Naresh
Published in Molecules (Basel, Switzerland) (07.05.2018)
Published in Molecules (Basel, Switzerland) (07.05.2018)
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Journal Article
N-Acetylglucosamine Inhibits LuxR, LasR and CviR Based Quorum Sensing Regulated Gene Expression Levels
Kimyon, Önder, Ulutürk, Zehra I, Nizalapur, Shashidhar, Lee, Matthew, Kutty, Samuel K, Beckmann, Sabrina, Kumar, Naresh, Manefield, Mike
Published in Frontiers in microbiology (23.08.2016)
Published in Frontiers in microbiology (23.08.2016)
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Journal Article
Inhibitors of pantothenate synthetase of Mycobacterium tuberculosis - a medicinal chemist perspective
Suresh, Amaroju, Srinivasarao, Singireddi, Khetmalis, Yogesh Mahadu, Nizalapur, Shashidhar, Sankaranarayanan, Murugesan, Gowri Chandra Sekhar, Kondapalli Venkata
Published in RSC advances (07.10.2020)
Published in RSC advances (07.10.2020)
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Journal Article
Design, synthesis and biological evaluation of 1,2,3-triazole based 2-aminobenzimidazoles as novel inhibitors of LasR dependent quorum sensing in Pseudomonas aeruginosa
Srinivasarao, Singireddi, Nandikolla, Adinarayana, Nizalapur, Shashidhar, Yu, Tsz Tin, Pulya, Sravani, Ghosh, Balaram, Murugesan, Sankaranarayanan, Kumar, Naresh, Chandra Sekhar, Kondapalli Venkata Gowri
Published in RSC advances (17.09.2019)
Published in RSC advances (17.09.2019)
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Journal Article
Synthesis and biological evaluation of novel acyclic and cyclic glyoxamide based derivatives as bacterial quorum sensing and biofilm inhibitors
Nizalapur, Shashidhar, Kimyon, Onder, Yee, Eugene, Bhadbhade, Mohan M., Manefield, Mike, Willcox, Mark, Black, David StC, Kumar, Naresh
Published in Organic & biomolecular chemistry (21.07.2017)
Published in Organic & biomolecular chemistry (21.07.2017)
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Journal Article
Design and synthesis of short amphiphilic cationic peptidomimetics based on biphenyl backbone as antibacterial agents
Kuppusamy, Rajesh, Yasir, Muhammad, Berry, Thomas, Cranfield, Charles G., Nizalapur, Shashidhar, Yee, Eugene, Kimyon, Onder, Taunk, Aditi, Ho, Kitty K.K., Cornell, Bruce, Manefield, Mike, Willcox, Mark, Black, David StC, Kumar, Naresh
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
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Journal Article
Amphipathic guanidine-embedded glyoxamide-based peptidomimetics as novel antibacterial agents and biofilm disruptors
Nizalapur, Shashidhar, Kimyon, Onder, Yee, Eugene, Ho, Kitty, Berry, Thomas, Manefield, Mike, Cranfield, Charles G., Willcox, Mark, Black, David StC, Kumar, Naresh
Published in Organic & biomolecular chemistry (01.03.2017)
Published in Organic & biomolecular chemistry (01.03.2017)
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Journal Article
A highly regio- and stereoselective Pd-catalyzed tandem allylic rearrangement/intramolecular decarboxylative coupling of aryl propiolates derived from Baylis–Hillman adducts
Satyanarayana, Tummanapalli, Vangapandu, Dhanunjaya Naidu, Muthuraman, Parthasarathy, Nizalapur, Shashidhar
Published in Tetrahedron letters (08.04.2015)
Published in Tetrahedron letters (08.04.2015)
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Journal Article
Synthesis and biological evaluation of novel acyclic and cyclic glyoxamide based derivatives as bacterial quorum sensing and biofilm inhibitorsElectronic supplementary information (ESI) available. CCDC 1541725 and 1541726. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c7ob01011g
Nizalapur, Shashidhar, Kimyon, Onder, Yee, Eugene, Bhadbhade, Mohan M, Manefield, Mike, Willcox, Mark, Black, David StC, Kumar, Naresh
Year of Publication 12.07.2017
Year of Publication 12.07.2017
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Journal Article
Synthesis of antimicrobial glucosamides as bacterial quorum sensing mechanism inhibitors
Biswas, Nripendra N., Yu, Tsz Tin, Kimyon, Önder, Nizalapur, Shashidhar, Gardner, Christopher R., Manefield, Mike, Griffith, Renate, Black, David StC, Kumar, Naresh
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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Journal Article
Design, synthesis, and characterisation of glyoxylamide-based short peptides as self-assembled gels
Aldilla, Vina R., Nizalapur, Shashidhar, Martin, Adam, Marjo, Chris E., Rich, Anne, Yee, Eugene, Suwannakot, Panthipa, Black, David StC, Thordarson, Pall, Kumar, Naresh
Published in New journal of chemistry (2017)
Published in New journal of chemistry (2017)
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Journal Article
Synthesis, quorum sensing inhibition and docking studies of 1,5-dihydropyrrol-2-ones
Goh, Wai-Kean, Gardner, Christopher R., Chandra Sekhar, Kondapalli V.G., Biswas, Nripendra N., Nizalapur, Shashidhar, Rice, Scott A., Willcox, Mark, Black, David StC, Kumar, Naresh
Published in Bioorganic & medicinal chemistry (01.12.2015)
Published in Bioorganic & medicinal chemistry (01.12.2015)
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Journal Article
Inhibitors of pantothenate synthetase of - a medicinal chemist perspective
Suresh, Amaroju, Srinivasarao, Singireddi, Khetmalis, Yogesh Mahadu, Nizalapur, Shashidhar, Sankaranarayanan, Murugesan, Gowri Chandra Sekhar, Kondapalli Venkata
Published in RSC advances (07.10.2020)
Published in RSC advances (07.10.2020)
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Journal Article
Design, synthesis, and characterisation of glyoxylamide-based short peptides as self-assembled gelsElectronic supplementary information (ESI) available. See DOI: 10.1039/c7nj02248d
Aldilla, Vina R, Nizalapur, Shashidhar, Martin, Adam, Marjo, Chris E, Rich, Anne, Yee, Eugene, Suwannakot, Panthipa, Black, David StC, Thordarson, Pall, Kumar, Naresh
Year of Publication 06.11.2017
Year of Publication 06.11.2017
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Journal Article
Amphipathic guanidine-embedded glyoxamide-based peptidomimetics as novel antibacterial agents and biofilm disruptorsElectronic supplementary information (ESI) available. See DOI: 10.1039/c7ob00053g
Nizalapur, Shashidhar, Kimyon, Onder, Yee, Eugene, Ho, Kitty, Berry, Thomas, Manefield, Mike, Cranfield, Charles G, Willcox, Mark, Black, David StC, Kumar, Naresh
Year of Publication 01.03.2017
Year of Publication 01.03.2017
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Journal Article
Glyoxylamide-based self-assembly hydrogels for sustained ciprofloxacin delivery
Aldilla, Vina R, Martin, Adam D, Nizalapur, Shashidhar, Marjo, Christopher E, Rich, Anne M, Ho, Kitty K K, Ittner, Lars M, Black, David StC, Thordarson, Pall, Kumar, Naresh
Published in Journal of materials chemistry. B, Materials for biology and medicine (14.10.2018)
Published in Journal of materials chemistry. B, Materials for biology and medicine (14.10.2018)
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Journal Article