Multi-Target Directed Ligands (MTDLs) Binding the σ1 Receptor as Promising Therapeutics: State of the Art and Perspectives
Abatematteo, Francesca Serena, Niso, Mauro, Contino, Marialessandra, Leopoldo, Marcello, Abate, Carmen
Published in International journal of molecular sciences (14.06.2021)
Published in International journal of molecular sciences (14.06.2021)
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Journal Article
PB28, the Sigma-1 and Sigma-2 Receptors Modulator With Potent Anti-SARS-CoV-2 Activity: A Review About Its Pharmacological Properties and Structure Affinity Relationships
Abate, Carmen, Niso, Mauro, Abatematteo, Francesca Serena, Contino, Marialessandra, Colabufo, Nicola Antonio, Berardi, Francesco
Published in Frontiers in pharmacology (07.12.2020)
Published in Frontiers in pharmacology (07.12.2020)
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Journal Article
Multifunctional thiosemicarbazones targeting sigma receptors: in vitro and in vivo antitumor activities in pancreatic cancer models
Niso, Mauro, Kopecka, Joanna, Abatematteo, Francesca Serena, Berardi, Francesco, Riganti, Chiara, Abate, Carmen
Published in Cellular oncology (Dordrecht) (01.12.2021)
Published in Cellular oncology (Dordrecht) (01.12.2021)
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Journal Article
Design and Synthesis of Arylpiperazine Serotonergic/Dopaminergic Ligands with Neuroprotective Properties
Mastromarino, Margherita, Niso, Mauro, Abate, Carmen, Proschak, Ewgenij, Dubiel, Mariam, Stark, Holger, Castro, Marián, Lacivita, Enza, Leopoldo, Marcello
Published in Molecules (Basel, Switzerland) (15.02.2022)
Published in Molecules (Basel, Switzerland) (15.02.2022)
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Journal Article
New Pharmacological Strategies against Pancreatic Adenocarcinoma: The Multifunctional Thiosemicarbazone FA4
Anobile, Dario P, Niso, Mauro, Puerta, Adrian, Fraga Rodrigues, Stephanie M, Abatematteo, Francesca S, Avan, Amir, Abate, Carmen, Riganti, Chiara, Giovannetti, Elisa
Published in Molecules (Basel, Switzerland) (04.03.2022)
Published in Molecules (Basel, Switzerland) (04.03.2022)
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Journal Article
Perspectives of P-Glycoprotein Modulating Agents in Oncology and Neurodegenerative Diseases: Pharmaceutical, Biological, and Diagnostic Potentials
Colabufo, Nicola Antonio, Berardi, Francesco, Cantore, Mariangela, Contino, Marialessandra, Inglese, Carmela, Niso, Mauro, Perrone, Roberto
Published in Journal of medicinal chemistry (11.03.2010)
Published in Journal of medicinal chemistry (11.03.2010)
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Journal Article
Sigma-2 Receptor Ligand Binding Modulates Association between TSPO and TMEM97
Thejer, Bashar M, Infantino, Vittoria, Santarsiero, Anna, Pappalardo, Ilaria, Abatematteo, Francesca S, Teakel, Sarah, Van Oosterum, Ashleigh, Mach, Robert H, Denora, Nunzio, Lee, Byung Chul, Resta, Nicoletta, Bagnulo, Rosanna, Niso, Mauro, Contino, Marialessandra, Montsch, Bianca, Heffeter, Petra, Abate, Carmen, Cahill, Michael A
Published in International journal of molecular sciences (28.03.2023)
Published in International journal of molecular sciences (28.03.2023)
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Journal Article
Mitochondrial Membranes of Human SH-SY5Y Neuroblastoma Cells Express Serotonin 5-HT7 Receptor
Tempio, Alessandra, Niso, Mauro, Laera, Luna, Trisolini, Lucia, Favia, Maria, Ciranna, Lucia, Marzulli, Domenico, Petrosillo, Giuseppe, Pierri, Ciro Leonardo, Lacivita, Enza, Leopoldo, Marcello
Published in International journal of molecular sciences (17.12.2020)
Published in International journal of molecular sciences (17.12.2020)
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Journal Article
Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity
Niso, Mauro, Abate, Carmen, Contino, Marialessandra, Ferorelli, Savina, Azzariti, Amalia, Perrone, Roberto, Colabufo, Nicola Antonio, Berardi, Francesco
Published in ChemMedChem (01.12.2013)
Published in ChemMedChem (01.12.2013)
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Journal Article
Nature-Inspired 1-Phenylpyrrolo[2,1- a ]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance
Nevskaya, Alisa A, Purgatorio, Rosa, Borisova, Tatiana N, Varlamov, Alexey V, Anikina, Lada V, Obydennik, Arina Yu, Nevskaya, Elena Yu, Niso, Mauro, Colabufo, Nicola A, Carrieri, Antonio, Catto, Marco, de Candia, Modesto, Voskressensky, Leonid G, Altomare, Cosimo D
Published in Pharmaceuticals (Basel, Switzerland) (01.04.2024)
Published in Pharmaceuticals (Basel, Switzerland) (01.04.2024)
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Journal Article
Structural Determinants in the Binding of BB2 Receptor Ligands: In Silico, X-Ray and NMR Studies in PD176252 Analogues
Carrieri, Antonio, Lacivita, Enza, Belviso, Benny Danilo, Caliandro, Rocco, Mastrorilli, Piero, Gallo, Vito, Niso, Mauro, Leopoldo, Marcello
Published in Current topics in medicinal chemistry (01.05.2017)
Published in Current topics in medicinal chemistry (01.05.2017)
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Journal Article
Phenylsulfonylfuroxans as Modulators of Multidrug-Resistance-Associated Protein-1 and P-Glycoprotein
Fruttero, Roberta, Crosetti, Marco, Chegaev, Konstantin, Guglielmo, Stefano, Gasco, Alberto, Berardi, Francesco, Niso, Mauro, Perrone, Roberto, Panaro, Maria Antonietta, Colabufo, Nicola Antonio
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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Journal Article
ABC pumps and their role in active drug transport
Colabufo, Nicola A, Berardi, Francesco, Contino, Marialessandra, Niso, Mauro, Perrone, Roberto
Published in Current topics in medicinal chemistry (01.02.2009)
Published in Current topics in medicinal chemistry (01.02.2009)
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Journal Article
Cyclohexylpiperazine derivative PB28, a σ2 agonist and σ1 antagonist receptor, inhibits cell growth, modulates P-glycoprotein, and synergizes with anthracyclines in breast cancer
Azzariti, Amalia, Colabufo, Nicola A., Berardi, Francesco, Porcelli, Letizia, Niso, Mauro, Simone, Grazia M., Perrone, Roberto, Paradiso, Angelo
Published in Molecular cancer therapeutics (01.07.2006)
Published in Molecular cancer therapeutics (01.07.2006)
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Journal Article
F281, synthetic agonist of the sigma-2 receptor, induces Ca2+ efflux from the endoplasmic reticulum and mitochondria in SK-N-SH cells
Cassano, Giuseppe, Gasparre, Giuseppe, Niso, Mauro, Contino, Marialessandra, Scalera, Vito, Colabufo, Nicola Antonio
Published in Cell calcium (Edinburgh) (01.04.2009)
Published in Cell calcium (Edinburgh) (01.04.2009)
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Journal Article
Is the σ2 Receptor a Histone Binding Protein?
Colabufo, Nicola Antonio, Berardi, Francesco, Abate, Carmen, Contino, Marialessandra, Niso, Mauro, Perrone, Roberto
Published in Journal of medicinal chemistry (13.07.2006)
Published in Journal of medicinal chemistry (13.07.2006)
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Journal Article
Bicalutamide failure in prostate cancer treatment: Involvement of Multi Drug Resistance proteins
Colabufo, Nicola Antonio, Pagliarulo, Vincenzo, Berardi, Francesco, Contino, Marialessandra, Inglese, Carmela, Niso, Mauro, Ancona, Patrizia, Albo, Giancarlo, Pagliarulo, Arcangelo, Perrone, Roberto
Published in European journal of pharmacology (28.12.2008)
Published in European journal of pharmacology (28.12.2008)
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Journal Article
Design, Synthesis, and Binding Affinities of Potential Positron Emission Tomography (PET) Ligands for Visualization of Brain Dopamine D3 Receptors
Leopoldo, Marcello, Lacivita, Enza, De Giorgio, Paola, Colabufo, Nicola A, Niso, Mauro, Berardi, Francesco, Perrone, Roberto
Published in Journal of medicinal chemistry (12.01.2006)
Published in Journal of medicinal chemistry (12.01.2006)
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Journal Article
PB183, a sigma receptor ligand, as a potential PET probe for the imaging of prostate adenocarcinoma
Colabufo, Nicola Antonio, Abate, Carmen, Contino, Marialessandra, Inglese, Carmela, Niso, Mauro, Berardi, Francesco, Perrone, Roberto
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
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