Determining target engagement in living systems
Simon, Gabriel M, Niphakis, Micah J, Cravatt, Benjamin F
Published in Nature chemical biology (01.04.2013)
Published in Nature chemical biology (01.04.2013)
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Journal Article
A Global Map of Lipid-Binding Proteins and Their Ligandability in Cells
Niphakis, Micah J., Lum, Kenneth M., Cognetta, Armand B., Correia, Bruno E., Ichu, Taka-Aki, Olucha, Jose, Brown, Steven J., Kundu, Soumajit, Piscitelli, Fabiana, Rosen, Hugh, Cravatt, Benjamin F.
Published in Cell (18.06.2015)
Published in Cell (18.06.2015)
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Journal Article
Proteome-wide mapping of cholesterol-interacting proteins in mammalian cells
Hulce, Jonathan J, Cognetta, Armand B, Niphakis, Micah J, Tully, Sarah E, Cravatt, Benjamin F
Published in Nature methods (01.03.2013)
Published in Nature methods (01.03.2013)
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Journal Article
ABHD17 regulation of plasma membrane palmitoylation and N-Ras-dependent cancer growth
Remsberg, Jarrett R, Suciu, Radu M, Zambetti, Noemi A, Hanigan, Thomas W, Firestone, Ari J, Inguva, Anagha, Long, Amanda, Ngo, Nhi, Lum, Kenneth M, Henry, Cassandra L, Richardson, Stewart K, Predovic, Marina, Huang, Ben, Dix, Melissa M, Howell, Amy R, Niphakis, Micah J, Shannon, Kevin, Cravatt, Benjamin F
Published in Nature chemical biology (01.08.2021)
Published in Nature chemical biology (01.08.2021)
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Journal Article
Palladium(II)-Catalyzed Direct Arylation of Enaminones Using Organotrifluoroborates
Ge, Haibo, Niphakis, Micah J, Georg, Gunda I
Published in Journal of the American Chemical Society (26.03.2008)
Published in Journal of the American Chemical Society (26.03.2008)
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Journal Article
Monoacylglycerol Lipase Inhibitors Reverse Paclitaxel-Induced Nociceptive Behavior and Proinflammatory Markers in a Mouse Model of Chemotherapy-Induced Neuropathy
Curry, Zachary A, Wilkerson, Jenny L, Bagdas, Deniz, Kyte, S Lauren, Patel, Nipa, Donvito, Giulia, Mustafa, Mohammed A, Poklis, Justin L, Niphakis, Micah J, Hsu, Ku-Lung, Cravatt, Benjamin F, Gewirtz, David A, Damaj, M Imad, Lichtman, Aron H
Published in The Journal of pharmacology and experimental therapeutics (01.07.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2018)
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The endocannabinoid hydrolysis inhibitor SA-57: Intrinsic antinociceptive effects, augmented morphine-induced antinociception, and attenuated heroin seeking behavior in mice
Wilkerson, Jenny L., Ghosh, Sudeshna, Mustafa, Mohammed, Abdullah, Rehab A., Niphakis, Micah J., Cabrera, Roberto, Maldonado, Rafael L., Cravatt, Benjamin F., Lichtman, Aron H.
Published in Neuropharmacology (01.03.2017)
Published in Neuropharmacology (01.03.2017)
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Journal Article
Inflammation causes insulin resistance in mice via interferon regulatory factor 3 (IRF3)-mediated reduction in FAHFA levels
Yan, Shuai, Santoro, Anna, Niphakis, Micah J, Pinto, Antonio M, Jacobs, Christopher L, Ahmad, Rasheed, Suciu, Radu M, Fonslow, Bryan R, Herbst-Graham, Rachel A, Ngo, Nhi, Henry, Cassandra L, Herbst, Dylan M, Saghatelian, Alan, Kahn, Barbara B, Rosen, Evan D
Published in Nature communications (30.05.2024)
Published in Nature communications (30.05.2024)
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Journal Article
Single-Cell Profiling and SCOPE-Seq Reveal Lineage Dynamics of Adult Ventricular-Subventricular Zone Neurogenesis and NOTUM as a Key Regulator
Mizrak, Dogukan, Bayin, N. Sumru, Yuan, Jinzhou, Liu, Zhouzerui, Suciu, Radu M., Niphakis, Micah J., Ngo, Nhi, Lum, Kenneth M., Cravatt, Benjamin F., Joyner, Alexandra L., Sims, Peter A.
Published in Cell reports (Cambridge) (23.06.2020)
Published in Cell reports (Cambridge) (23.06.2020)
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Journal Article
Neuroprotective effects of fatty acid amide hydrolase catabolic enzyme inhibition in a HIV-1 Tat model of neuroAIDS
Hermes, Douglas J., Xu, Changqing, Poklis, Justin L., Niphakis, Micah J., Cravatt, Benjamin F., Mackie, Ken, Lichtman, Aron H., Ignatowska-Jankowska, Bogna M., Fitting, Sylvia
Published in Neuropharmacology (01.10.2018)
Published in Neuropharmacology (01.10.2018)
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Journal Article
Chemoproteomic identification of a DPP4 homolog in Bacteroides thetaiotaomicron
Keller, Laura J, Nguyen, Taylor H, Liu, Lawrence J, Hurysz, Brianna M, Lakemeyer, Markus, Guerra, Matteo, Gelsinger, Danielle J, Chanin, Rachael, Ngo, Nhi, Lum, Kenneth M, Faucher, Franco, Ipock, Phillip, Niphakis, Micah J, Bhatt, Ami S, O'Donoghue, Anthony J, Huang, Kerwyn Casey, Bogyo, Matthew
Published in Nature chemical biology (01.12.2023)
Published in Nature chemical biology (01.12.2023)
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Journal Article
Selective monoacylglycerol lipase inhibitors: antinociceptive versus cannabimimetic effects in mice
Ignatowska-Jankowska, Bogna, Wilkerson, Jenny L, Mustafa, Mohammed, Abdullah, Rehab, Niphakis, Micah, Wiley, Jenny L, Cravatt, Benjamin F, Lichtman, Aron H
Published in The Journal of pharmacology and experimental therapeutics (01.05.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2015)
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