New Generation Oxyntomodulin Peptides with Improved Pharmacokinetic Profiles Exhibit Weight Reducing and Anti-Steatotic Properties in Mice
Yang, Peng-Yu, Zou, Huafei, Amso, Zaid, Lee, Candy, Huang, David, Woods, Ashley K, Nguyen-Tran, Vân T. B, Schultz, Peter G, Shen, Weijun
Published in Bioconjugate chemistry (15.04.2020)
Published in Bioconjugate chemistry (15.04.2020)
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Discovery of CMX990: A Potent SARS-CoV‑2 3CL Protease Inhibitor Bearing a Novel Warhead
Dayan Elshan, N. G. R., Wolff, Karen C., Riva, Laura, Woods, Ashley K., Grabovyi, Gennadii, Wilson, Katy, Pedroarena, James, Ghorai, Sourav, Nazarian, Armen, Weiss, Frank, Liu, Yuyin, Mazumdar, Wrickban, Song, Lirui, Okwor, Neechi, Malvin, Jacqueline, Bakowski, Malina A., Beutler, Nathan, Kirkpatrick, Melanie G., Gebara-Lamb, Amal, Huang, Edward, Nguyen-Tran, Vân T. B., Chi, Victor, Li, Shuangwei, Rogers, Thomas F., McNamara, Case W., Gupta, Anil Kumar, Rahimi, Alireza, Chen, Jian Jeffrey, Joseph, Sean B., Schultz, Peter G., Chatterjee, Arnab K.
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Design of Potent and Proteolytically Stable Biaryl-Stapled GLP-1R/GIPR Peptide Dual Agonists
Yang, Yifang, Lee, Candy, Reddy, Reddy Rajasekhar, Huang, David J., Zhong, Weixia, Nguyen-Tran, Vân T. B., Shen, Weijun, Lin, Qing
Published in ACS chemical biology (20.05.2022)
Published in ACS chemical biology (20.05.2022)
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Rational design of a Kv1.3 channel-blocking antibody as a selective immunosuppressant
Wang, Rongsheng E., Wang, Ying, Zhang, Yuhan, Gabrelow, Chase, Zhang, Yong, Chi, Victor, Fu, Qiangwei, Luo, Xiaozhou, Wang, Danling, Joseph, Sean, Johnson, Kristen, Chatterjee, Arnab K., Wright, Timothy M., Nguyen-Tran, Vân T. B., Teijaro, John, Theofilopoulos, Argyrios N., Schultz, Peter G., Wang, Feng
Published in Proceedings of the National Academy of Sciences - PNAS (11.10.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (11.10.2016)
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Selective DYRK1A Inhibitor for the Treatment of Type 1 Diabetes: Discovery of 6‑Azaindole Derivative GNF2133
Liu, Yahu A, Jin, Qihui, Zou, Yefen, Ding, Qiang, Yan, Shanshan, Wang, Zhicheng, Hao, Xueshi, Nguyen, Bao, Zhang, Xiaoyue, Pan, Jianfeng, Mo, Tingting, Jacobsen, Kate, Lam, Thanh, Wu, Tom Y.-H, Petrassi, H. Michael, Bursulaya, Badry, DiDonato, Michael, Gordon, W. Perry, Liu, Bo, Baaten, Janine, Hill, Robert, Nguyen-Tran, Vân, Qiu, Minhua, Zhang, You-Qing, Kamireddy, Anwesh, Espinola, Sheryll, Deaton, Lisa, Ha, Sukwon, Harb, George, Jia, Yong, Li, Jing, Shen, Weijun, Schumacher, Andrew M, Colman, Karyn, Glynne, Richard, Pan, Shifeng, McNamara, Peter, Laffitte, Bryan, Meeusen, Shelly, Molteni, Valentina, Loren, Jon
Published in Journal of medicinal chemistry (26.03.2020)
Published in Journal of medicinal chemistry (26.03.2020)
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Recombinant Expression and Stapling of a Novel Long-Acting GLP-1R Peptide Agonist
Lear, Sam, Seo, Hyosuk, Lee, Candy, Lei, Lei, Amso, Zaid, Huang, David, Zou, Huafei, Zhou, Zhihong, Nguyen-Tran, Vân T B, Shen, Weijun
Published in Molecules (Basel, Switzerland) (28.05.2020)
Published in Molecules (Basel, Switzerland) (28.05.2020)
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Engineering a Potent, Long-Acting, and Periphery-Restricted Oxytocin Receptor Agonist with Anorexigenic and Body Weight Reducing Effects
Pflimlin, Elsa, Zhou, Zhihong, Amso, Zaid, Fu, Qiangwei, Lee, Candy, Muppiddi, Avinash, Joseph, Sean B, Nguyen-Tran, Vân, Shen, Weijun
Published in Journal of medicinal chemistry (09.01.2020)
Published in Journal of medicinal chemistry (09.01.2020)
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Journal Article
Correction to “Discovery of CMX990: A Potent SARS-CoV‑2 3CL Protease Inhibitor Bearing a Novel Warhead”
Elshan, N. G. R. Dayan, Wolff, Karen C., Riva, Laura, Woods, Ashley K., Grabovyi, Gennadii, Wilson, Katy, Pedroarena, James, Ghorai, Sourav, Nazarian, Armen, Weiss, Frank, Liu, Yuyin, Mazumdar, Wrickban, Song, Lirui, Okwor, Neechi, Malvin, Jacqueline, Liu, Dongdong, Bakowski, Malina A., Beutler, Nathan, Kirkpatrick, Melanie G., Gebara-Lamb, Amal, Huang, Edward, Nguyen-Tran, Vân T. B., Chi, Victor, Li, Shuangwei, Rogers, Thomas F., McNamara, Case W., Gupta, Anil Kumar, Rahimi, Alireza, Chen, Jian Jeffrey, Joseph, Sean B., Schultz, Peter G., Chatterjee, Arnab K.
Published in Journal of medicinal chemistry (27.06.2024)
Published in Journal of medicinal chemistry (27.06.2024)
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The activity of sulfono-γ-AApeptide helical foldamers that mimic GLP-1
Sang, Peng, Zhou, Zhihong, Shi, Yan, Lee, Candy, Amso, Zaid, Huang, David, Odom, Timothy, Nguyen-Tran, Vân T B, Shen, Weijun, Cai, Jianfeng
Published in Science advances (01.05.2020)
Published in Science advances (01.05.2020)
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α/Sulfono-γ-AA peptide hybrids agonist of GLP-1R with prolonged action both in vitro and in vivo
Shi, Yan, Lee, Candy, Sang, Peng, Amso, Zaid, Huang, David, Zhong, Weixia, Gu, Meng, Wei, Lulu, Nguyen-Tran, Vân T.B., Zhang, Jingyao, Shen, Weijun, Cai, Jianfeng
Published in Acta pharmaceutica Sinica. B (01.04.2023)
Published in Acta pharmaceutica Sinica. B (01.04.2023)
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Novel Bisaryl Substituted Thiazoles and Oxazoles as Highly Potent and Selective Peroxisome Proliferator-Activated Receptor δ Agonists
Epple, Robert, Cow, Christopher, Xie, Yongping, Azimioara, Mihai, Russo, Ross, Wang, Xing, Wityak, John, Karanewsky, Donald S, Tuntland, Tove, Nguyêñ-Trân, Vân T. B, Cuc Ngo, Cara, Huang, David, Saez, Enrique, Spalding, Tracy, Gerken, Andrea, Iskandar, Maya, Seidel, H. Martin, Tian, Shin-Shay
Published in Journal of medicinal chemistry (14.01.2010)
Published in Journal of medicinal chemistry (14.01.2010)
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Identification of Potent and Selective RIPK2 Inhibitors for the Treatment of Inflammatory Diseases
He, Xiaohui, Da Ros, Sara, Nelson, John, Zhu, Xuefeng, Jiang, Tao, Okram, Barun, Jiang, Songchun, Michellys, Pierre-Yves, Iskandar, Maya, Espinola, Sheryll, Jia, Yong, Bursulaya, Badry, Kreusch, Andreas, Gao, Mu-Yun, Spraggon, Glen, Baaten, Janine, Clemmer, Leah, Meeusen, Shelly, Huang, David, Hill, Robert, Nguyen-Tran, Vân, Fathman, John, Liu, Bo, Tuntland, Tove, Gordon, Perry, Hollenbeck, Thomas, Ng, Kenneth, Shi, Jian, Bordone, Laura, Liu, Hong
Published in ACS medicinal chemistry letters (12.10.2017)
Published in ACS medicinal chemistry letters (12.10.2017)
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Biofilm reactors filled with Stick-bed Biofix and Swim-bed Biofringe biomass carriers in treating chitin production wastewater containing high salinity
Nguyen, Tan Phong, Vo, Thi Kim Quyen, Tran, Nguyen Van Nhu, Tran, Nguyen Van Nhi
Published in Environmental technology (01.10.2024)
Published in Environmental technology (01.10.2024)
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Co-precipitation polymerization of dual functional monomers and polystyrene- co -divinylbenzene for ciprofloxacin imprinted polymer preparation
Nguyen, Huy Truong, Vuong Bui, Nhat Thao, Kanhounnon, Wilfried G, Vu Huynh, Kim Long, Nguyen, Tran-Van-Anh, Nguyen, Hien Minh, Do, Minh Huy, Badawi, Michael, Thach, Ut Dong
Published in RSC advances (18.10.2021)
Published in RSC advances (18.10.2021)
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Multifunctional Antibody Agonists Targeting Glucagon-like Peptide-1, Glucagon, and Glucose-Dependent Insulinotropic Polypeptide Receptors
Wang, Ying, Du, Jintang, Zou, Huafei, Liu, Yan, Zhang, Yuhan, Gonzalez, Jose, Chao, Elizabeth, Lu, Lucy, Yang, Pengyu, Parker, Holly, Nguyen-Tran, Van, Shen, Weijun, Wang, Danling, Schultz, Peter G., Wang, Feng
Published in Angewandte Chemie (International ed.) (26.09.2016)
Published in Angewandte Chemie (International ed.) (26.09.2016)
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A New Carvotacetone Derivative from the Aerial Part of Sphaeranthus africanus
Thuy Le, Huong, Vu, Thien‐Y, Nguyen, Tran‐Van‐Anh, Dinh Tri, Mai, Pham, Nguyen‐Kim‐Tuyen, Truong Nguyen, Huy, Nguyen, Ngoc‐Hong, Nguyen, Huu‐Hung, Duong, Thuc‐Huy
Published in Chemistry & biodiversity (01.06.2023)
Published in Chemistry & biodiversity (01.06.2023)
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α‐Glucosidase Inhibition by Usnic Acid Derivatives
Nguyen, Huy Truong, Devi, Asshaima Paramita, Nguyen, Tran‐Van‐Anh, Chavasiri, Warinthorn, Pham, Duc‐Dung, Sichaem, Jirapast, Nguyen, Ngoc‐Hong, Huynh, Bui‐Linh‐Chi, Nguyen, Van‐Kieu, Duong, Thuc Huy
Published in Chemistry & biodiversity (01.04.2021)
Published in Chemistry & biodiversity (01.04.2021)
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α-Glucosidase inhibitory derivatives of protocetraric acid
Nguyen, Huu-Hung, Duong, Thuc-Huy, Nguyen, Tran-Van-Anh, Do, Thanh-Hung, Pham, Duc-Dung, Nguyen, Ngoc-Hong, Nguyen, Huy Truong
Published in Natural product research (18.06.2023)
Published in Natural product research (18.06.2023)
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