Search Results - "Neustadt, B. R" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoro- methyl)phenyl]ethyl]-1-piperazinyl]- piperidine N1-Oxide (Sch-350634), an Orally Bioavailable, Potent CCR5 Antagonist

Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoro- methyl)phenyl]ethyl]-1-piperazinyl]- piperidine N1-Oxide (Sch-350634), an Orally Bioavailable, Potent CCR5 Antagonist

by Tagat, Jayaram R, Steensma, Ruo W, McCombie, Stuart W, Nazareno, Dennis V, Lin, Sue-Ing, Neustadt, Bernard R, Cox, Kathleen, Xu, Serena, Wojcik, Lisa, Murray, Michael G, Vantuno, Nicole, Baroudy, Bahige M, Strizki, Julie M
Published in Journal of medicinal chemistry (11.10.2001)

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Journal Article

Synthesis and pharmacological activity of angiotensin-converting enzyme inhibitors: N-(mercaptoacyl)-4-substituted-(S)-prolines

Synthesis and pharmacological activity of angiotensin-converting enzyme inhibitors: N-(mercaptoacyl)-4-substituted-(S)-prolines

by Smith, Elizabeth M, Swiss, Gerald F, Neustadt, Bernard R, Gold, Elijah H, Sommer, Jane A, Brown, Arthur D, Chiu, Peter J. S, Moran, Rosa, Sybertz, Edmund J, Baum, Thomas
Published in Journal of medicinal chemistry (01.04.1988)

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Journal Article

Facile preparation of N-(sulfonyl)carbamates

Facile preparation of N-(sulfonyl)carbamates

by Neustadt, Bernard R.
Published in Tetrahedron letters (17.01.1994)

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Journal Article

Angiotensin converting enzyme inhibitors: spirapril and related compounds

Angiotensin converting enzyme inhibitors: spirapril and related compounds

by Smith, Elizabeth M, Swiss, Gerald F, Neustadt, Bernard R, McNamara, Paul, Gold, Elijah H, Sybertz, Edmund J, Baum, Thomas
Published in Journal of medicinal chemistry (01.07.1989)

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Journal Article

Carboxyalkyl dipeptides with atrial natriuretic factor potentiating and antihypertensive activity

Carboxyalkyl dipeptides with atrial natriuretic factor potentiating and antihypertensive activity

by Haslanger, Martin F, Sybertz, Edmund J, Neustadt, Bernard R, Smith, Elizabeth M, Nechuta, Terry L, Berger, Joel
Published in Journal of medicinal chemistry (01.04.1989)

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Journal Article

Construction of a family of biphenyl combinatorial libraries: Structure-activity studies utilizing libraries of mixtures

Construction of a family of biphenyl combinatorial libraries: Structure-activity studies utilizing libraries of mixtures

by Neustadt, Bernard R., Smith, Elizabeth M., Lindo, Neil, Nechuta, Terry, Bronnenkant, Alan, Wu, Arthur, Armstrong, Lydia, Kumar, Chandra
Published in Bioorganic & medicinal chemistry letters (08.09.1998)

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Journal Article

Chemistry of aporphines. IV. Synthesis of aporphines via Reissert alkylation, photochemical cyclization, and the Pschorr cyclization route

Chemistry of aporphines. IV. Synthesis of aporphines via Reissert alkylation, photochemical cyclization, and the Pschorr cyclization route

by Neumeyer, John L, Oh, K. H, Weinhardt, Klaus K, Neustadt, B. R
Published in Journal of organic chemistry (01.12.1969)

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Journal Article

MERCAPTOACYL AMINO-ACID INHIBITORS OF ATRIOPEPTIDASE .1. STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF METHIONINE AND S-ALKYLCYSTEINE DERIVATIVES

MERCAPTOACYL AMINO-ACID INHIBITORS OF ATRIOPEPTIDASE .1. STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF METHIONINE AND S-ALKYLCYSTEINE DERIVATIVES

by NEUSTADT, BR, SMITH, EM, NECHUTA, TL, BRONNENKANT, AA, HASLANGER, MF, WATKINS, RW, FOSTER, CJ, SYBERTZ, EJ
Published in Journal of medicinal chemistry (22.07.1994)

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Aporphines. 8. Total Synthesis and Pharmacological Evaluation of (±)-Apomorphine, (±)-Apocodeine, (±)-N-n-Propylnorapomorphine, and (±)-N-n--Propylnorapocodeine

Aporphines. 8. Total Synthesis and Pharmacological Evaluation of (±)-Apomorphine, (±)-Apocodeine, (±)-N-n-Propylnorapomorphine, and (±)-N-n--Propylnorapocodeine

by Neumeyer, John, Neustadt, Bernard, Oh, Kyung, Weinhardt, Klaus, Boyce, Charles, Rosenberg, Franklin, Teiger, David
Published in Journal of medicinal chemistry (01.11.1973)

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Journal Article

Piperazine-based CCR5 antagonists as HIV-1 inhibitors. III: synthesis, antiviral and pharmacokinetic profiles of symmetrical heteroaryl carboxamides

Piperazine-based CCR5 antagonists as HIV-1 inhibitors. III: synthesis, antiviral and pharmacokinetic profiles of symmetrical heteroaryl carboxamides

by McCombie, Stuart W., Tagat, Jayaram R., Vice, Susan F., Lin, Sue-Ing, Steensma, Ruo, Palani, Anandan, Neustadt, Bernard R., Baroudy, Bahige M., Strizki, Julie M., Endres, Michael, Cox, Kathleen, Dan, Niya, Chou, Chuan-Chu
Published in Bioorganic & medicinal chemistry letters (10.02.2003)

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Journal Article

Construction of a family of biphenyl combinatorial libraries : Structure-activity studies utilizing libraries of mixtures: Combinatorial chemistry

Construction of a family of biphenyl combinatorial libraries : Structure-activity studies utilizing libraries of mixtures: Combinatorial chemistry

by NEUSTADT, B. R, SMITH, E. M, LINDO, N, NECHUTA, T, BRONNENKANT, A, WU, A, ARMSTRONG, L, KUMAR, C
Published in Bioorganic & medicinal chemistry letters (1998)

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Journal Article

Mercaptoacyl amino acid inhibitors of atriopeptidase. I: Structure-activity relationship studies of methionine and S-alkylcysteine derivatives

Mercaptoacyl amino acid inhibitors of atriopeptidase. I: Structure-activity relationship studies of methionine and S-alkylcysteine derivatives

by NEUSTADT, B. R, SMITH, E. M, NECHUTA, T. L, BRONNENKANT, A. A, HASLANGER, M. F, WATKINS, R. W, FOSTER, C. J, SYBERTZ, E
Published in Journal of medicinal chemistry (1994)

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Journal Article

Combinatorial libraries based on a novel and readily accessible “centroid” scaffold

Combinatorial libraries based on a novel and readily accessible “centroid” scaffold

by Neustadt, Bernard R., Smith, Elizabeth M., Nechuta, Terry, Zhang, Yongzheng
Published in Tetrahedron letters (23.07.1998)

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Journal Article

ANALOGIFORFARANDE FOR FRAMSTELLNING AV NYA TERAPEUTISKT AKTIVA FENYLUREAFORENINGAR

ANALOGIFORFARANDE FOR FRAMSTELLNING AV NYA TERAPEUTISKT AKTIVA FENYLUREAFORENINGAR

by B R NEUSTADT
Year of Publication 11.06.1980

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Patent

SUBSTITUEREDE UREIDOFORBINDELSER

SUBSTITUEREDE UREIDOFORBINDELSER

by NEUSTADT B R
Year of Publication 03.06.1976

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Patent

NO753984L

NO753984L

by NEUSTADT B R
Year of Publication 03.06.1976

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Patent

SUBSTITUERADE UREIDOFORENINGAR

SUBSTITUERADE UREIDOFORENINGAR

by NEUSTADT B R
Year of Publication 03.06.1976

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Patent

5-(2-ANILINOALKYLAMINO-1-HYDROXYALKYL) SALICYLAMIDER FREMGANGSMAADE TIL DERES FREMSTILLING SAMT FARMACEUTISKE KOMPOSITIONER INDEHOLDENDE DISSE

5-(2-ANILINOALKYLAMINO-1-HYDROXYALKYL) SALICYLAMIDER FREMGANGSMAADE TIL DERES FREMSTILLING SAMT FARMACEUTISKE KOMPOSITIONER INDEHOLDENDE DISSE

by NEUSTADT B R, GOLD E H
Year of Publication 28.06.1979

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Patent

Aporphines. V. Total synthesis of (plus or minus)-apomorphine

Aporphines. V. Total synthesis of (plus or minus)-apomorphine

by Neumeyer, J L, Neustadt, B R, Weinhardt, K K
Published in Journal of pharmaceutical sciences (01.12.1970)

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Journal Article

ANALOGIFORFARANDE FOR FRAMSTELLNING AV NYA TERAPEUTISKT AKTIVA FENYLUREAFORENINGAR

ANALOGIFORFARANDE FOR FRAMSTELLNING AV NYA TERAPEUTISKT AKTIVA FENYLUREAFORENINGAR

by B R NEUSTADT
Year of Publication 11.06.1980

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Patent