Discovery of Entrectinib: A New 3‑Aminoindazole As a Potent Anaplastic Lymphoma Kinase (ALK), c‑ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor
Menichincheri, Maria, Ardini, Elena, Magnaghi, Paola, Avanzi, Nilla, Banfi, Patrizia, Bossi, Roberto, Buffa, Laura, Canevari, Giulia, Ceriani, Lucio, Colombo, Maristella, Corti, Luca, Donati, Daniele, Fasolini, Marina, Felder, Eduard, Fiorelli, Claudio, Fiorentini, Francesco, Galvani, Arturo, Isacchi, Antonella, Borgia, Andrea Lombardi, Marchionni, Chiara, Nesi, Marcella, Orrenius, Christian, Panzeri, Achille, Pesenti, Enrico, Rusconi, Luisa, Saccardo, Maria Beatrice, Vanotti, Ermes, Perrone, Ettore, Orsini, Paolo
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
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Journal Article
Optimization of 6,6-dimethyl pyrrolo[3,4- c]pyrazoles: Identification of PHA-793887, a potent CDK inhibitor suitable for intravenous dosing
Brasca, Maria Gabriella, Albanese, Clara, Alzani, Rachele, Amici, Raffaella, Avanzi, Nilla, Ballinari, Dario, Bischoff, James, Borghi, Daniela, Casale, Elena, Croci, Valter, Fiorentini, Francesco, Isacchi, Antonella, Mercurio, Ciro, Nesi, Marcella, Orsini, Paolo, Pastori, Wilma, Pesenti, Enrico, Pevarello, Paolo, Roussel, Patrick, Varasi, Mario, Volpi, Daniele, Vulpetti, Anna, Ciomei, Marina
Published in Bioorganic & medicinal chemistry (01.03.2010)
Published in Bioorganic & medicinal chemistry (01.03.2010)
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Journal Article
3-Aminopyrazole Inhibitors of CDK2/Cyclin A as Antitumor Agents. 2. Lead Optimization
Pevarello, Paolo, Brasca, Maria Gabriella, Orsini, Paolo, Traquandi, Gabriella, Longo, Antonio, Nesi, Marcella, Orzi, Fabrizio, Piutti, Claudia, Sansonna, Pietro, Varasi, Mario, Cameron, Alexander, Vulpetti, Anna, Roletto, Fulvia, Alzani, Rachele, Ciomei, Marina, Albanese, Clara, Pastori, Wilma, Marsiglio, Aurelio, Pesenti, Enrico, Fiorentini, Francesco, Bischoff, Jim R, Mercurio, Ciro
Published in Journal of medicinal chemistry (21.04.2005)
Published in Journal of medicinal chemistry (21.04.2005)
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Journal Article
Multi-step organic synthesis using solid-supported reagents and scavengers: a new paradigm in chemical library generation
Ley, Steven V., Baxendale, Ian R., Bream, Robert N., Jackson, Philip S., Leach, Andrew G., Longbottom, Deborah A., Nesi, Marcella, Scott, James S., Storer, R. Ian, Taylor, Stephen J.
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
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Journal Article
Crystal Structures of Anaplastic Lymphoma Kinase in Complex with ATP Competitive Inhibitors
Bossi, Roberto T, Saccardo, M. Beatrice, Ardini, Elena, Menichincheri, Maria, Rusconi, Luisa, Magnaghi, Paola, Orsini, Paolo, Avanzi, Nilla, Borgia, Andrea Lombardi, Nesi, Marcella, Bandiera, Tiziano, Fogliatto, Gianpaolo, Bertrand, Jay A
Published in Biochemistry (Easton) (17.08.2010)
Published in Biochemistry (Easton) (17.08.2010)
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Journal Article
Identification of unprecedented ATP-competitive choline kinase inhibitors
Quartieri, Francesca, Nesi, Marcella, Avanzi, Nilla R., Borghi, Daniela, Casale, Elena, Corti, Emiliana, Cucchi, Ulisse, Donati, Daniele, Fasolini, Marina, Felder, Eduard R., Galvani, Arturo, Giorgini, Maria L., Lomolino, Antonio, Menichincheri, Maria, Orrenius, Christian, Perrera, Claudia, Re Depaolini, Stefania, Riccardi-Sirtori, Federico, Salsi, Enea, Isacchi, Antonella, Gnocchi, Paola
Published in Bioorganic & medicinal chemistry letters (01.11.2021)
Published in Bioorganic & medicinal chemistry letters (01.11.2021)
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Journal Article
Correction to Discovery of Entrectinib: A New 3‑Aminoindazole as a Potent Anaplastic Lymphoma Kinase (ALK), c‑ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor
Menichincheri, Maria, Ardini, Elena, Magnaghi, Paola, Avanzi, Nilla, Banfi, Patrizia, Bossi, Roberto, Buffa, Laura, Canevari, Giulia, Ceriani, Lucio, Colombo, Maristella, Corti, Luca, Donati, Daniele, Fasolini, Marina, Felder, Eduard, Fiorelli, Claudio, Fiorentini, Francesco, Galvani, Arturo, Isacchi, Antonella, Borgia, Andrea Lombardi, Marchionni, Chiara, Nesi, Marcella, Orrenius, Christian, Panzeri, Achille, Pesenti, Enrico, Rusconi, Luisa, Saccardo, Maria Beatrice, Vanotti, Ermes, Perrone, Ettore, Orsini, Paolo
Published in Journal of medicinal chemistry (12.09.2019)
Published in Journal of medicinal chemistry (12.09.2019)
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Journal Article
Abstract 4790: Identification and characterization of ATP-mimetic choline kinase inhibitors
Gnocchi, Paola, Quartieri, Francesca, Badari, Alessandra, Bosotti, Roberta, Casale, Elena, Corti, Emiliana, Cristiani, Cinzia G., Cucchi, Ulisse, Gasparri, Fabio, Gianellini, Laura M., Giorgini, Laura M., Montemartini, Marisa, Mion, Giuliana, Nesi, Marcella, Orrenius, Christian, Re, Claudia E., Donati, Daniele, Felder, Eduard R., Galvani, Arturo, Isacchi, Antonella
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Novel pyrrole carboxamide inhibitors of JAK2 as potential treatment of myeloproliferative disorders
Brasca, Maria Gabriella, Gnocchi, Paola, Nesi, Marcella, Amboldi, Nadia, Avanzi, Nilla, Bertrand, Jay, Bindi, Simona, Canevari, Giulia, Casero, Daniele, Ciomei, Marina, Colombo, Nicoletta, Cribioli, Sabrina, Fachin, Gabriele, Felder, Eduard R., Galvani, Arturo, Isacchi, Antonella, Motto, Ilaria, Panzeri, Achille, Donati, Daniele
Published in Bioorganic & medicinal chemistry (15.05.2015)
Published in Bioorganic & medicinal chemistry (15.05.2015)
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Journal Article
Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors
Brasca, Maria Gabriella, Nesi, Marcella, Avanzi, Nilla, Ballinari, Dario, Bandiera, Tiziano, Bertrand, Jay, Bindi, Simona, Canevari, Giulia, Carenzi, Davide, Casero, Daniele, Ceriani, Lucio, Ciomei, Marina, Cirla, Alessandra, Colombo, Maristella, Cribioli, Sabrina, Cristiani, Cinzia, Della Vedova, Franco, Fachin, Gabriele, Fasolini, Marina, Felder, Eduard R., Galvani, Arturo, Isacchi, Antonella, Mirizzi, Danilo, Motto, Ilaria, Panzeri, Achille, Pesenti, Enrico, Vianello, Paola, Gnocchi, Paola, Donati, Daniele
Published in Bioorganic & medicinal chemistry (01.09.2014)
Published in Bioorganic & medicinal chemistry (01.09.2014)
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Journal Article
Abstract A179: NMS-P113, a novel orally available JAK2 selective inhibitor
Gnocchi, Paola, Brasca, Maria Gabriella, Amboldi, Nadia, Avanzi, Nilla, Bindi, Simona, Canevari, Giulia, Casero, Daniele, Ceruti, Roberta, Ciomei, Marina, Cribioli, Sabrina, Cristiani, Cinzia, Nesi, Marcella, Pastori, Wilma, Patton, Veronica, Pellizzoni, Cinzia, Texido, Gemma, Ardini, Elena, Felder, Eduard R., Isacchi, Antonella, Donati, Daniele, Galvani, Arturo
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Journal Article
Regioselective halogenation of aminopyrimidinyl-pyrrole carboxylic acid derivatives
Vanotti, Ermes, Caldarelli, Marina, Disingrini, Teresa, Nesi, Marcella, Tatò, Marco, Vianello, Paola, Menichincheri, Maria
Published in Tetrahedron (12.12.2009)
Published in Tetrahedron (12.12.2009)
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Journal Article
Abstract B230: NMS-P948, a potent dual FLT3/KIT inhibitor, also active on secondary resistance mutations
Ciomei, Marina, Fraietta, Ivan, Cribioli, Sabrina, Marsiglio, Aurelio, Casero, Daniele, Nesi, Marcella, Donati, Daniele, Isacchi, Antonella, Pesenti, Enrico, Galvani, Arturo, Borgia, Andrea Lombardi
Published in Molecular cancer therapeutics (12.11.2011)
Published in Molecular cancer therapeutics (12.11.2011)
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Journal Article
SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS
MARCHIONNI CHIARA, NESI MARCELLA, LOMBARDI BORGIA ANDREA, MENICHINCHERI MARIA, PANZERI ACHILLE, VANOTTI ERMES, ORSINI PAOLO, PERRONE ETTORE
Year of Publication 28.05.2015
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Year of Publication 28.05.2015
Patent
A practical synthesis of the major 3-hydroxy-2-pyrrolidinone metabolite of a potent CDK2/cyclin A inhibitor
Nesi, Marcella, Borghi, Daniela, Brasca, Maria Gabriella, Fiorentini, Francesco, Pevarello, Paolo
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
Published in Bioorganic & medicinal chemistry letters (15.06.2006)
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Journal Article
6-Substituted Pyrrolo[3,4-c]pyrazoles: An Improved Class of CDK2 Inhibitors
Brasca, Maria Gabriella, Albanese, Clara, Amici, Raffaella, Ballinari, Dario, Corti, Luca, Croci, Valter, Fancelli, Daniele, Fiorentini, Francesco, Nesi, Marcella, Orsini, Paolo, Orzi, Fabrizio, Pastori, Wilma, Perrone, Ettore, Pesenti, Enrico, Pevarello, Paolo, Riccardi-Sirtori, Federico, Roletto, Fulvia, Roussel, Patrick, Varasi, Mario, Vulpetti, Anna, Mercurio, Ciro
Published in ChemMedChem (11.06.2007)
Published in ChemMedChem (11.06.2007)
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Journal Article
SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS
PEVARELLO PAOLO, ORZI FABRIZIO, ROUSSEL PATRICK, NESI MARCELLA, AMICI RAFFAELLA, FANCELLI DANIELE, VULPETTI ANNA, BRASCA MARIA GABRIELLA, ORSINI PAOLO
Year of Publication 23.04.2012
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Year of Publication 23.04.2012
Patent