Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials
Albrecht, Brian K, Gehling, Victor S, Hewitt, Michael C, Vaswani, Rishi G, Côté, Alexandre, Leblanc, Yves, Nasveschuk, Christopher G, Bellon, Steve, Bergeron, Louise, Campbell, Robert, Cantone, Nico, Cooper, Michael R, Cummings, Richard T, Jayaram, Hariharan, Joshi, Shivangi, Mertz, Jennifer A, Neiss, Adrianne, Normant, Emmanuel, O’Meara, Michael, Pardo, Eneida, Poy, Florence, Sandy, Peter, Supko, Jeffrey, Sims, Robert J, Harmange, Jean-Christophe, Taylor, Alexander M, Audia, James E
Published in Journal of medicinal chemistry (25.02.2016)
Published in Journal of medicinal chemistry (25.02.2016)
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Bromodomain inhibition of the transcriptional coactivators CBP/EP300 as a therapeutic strategy to target the IRF4 network in multiple myeloma
Conery, Andrew R, Centore, Richard C, Neiss, Adrianne, Keller, Patricia J, Joshi, Shivangi, Spillane, Kerry L, Sandy, Peter, Hatton, Charlie, Pardo, Eneida, Zawadzke, Laura, Bommi-Reddy, Archana, Gascoigne, Karen E, Bryant, Barbara M, Mertz, Jennifer A, Sims, Robert J
Published in eLife (05.01.2016)
Published in eLife (05.01.2016)
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miR-34a confers chemosensitivity through modulation of MAGE-A and p53 in medulloblastoma
Weeraratne, Shyamal D., Amani, Vladimir, Neiss, Adrianne, Teider, Natalia, Scott, Deborah K., Pomeroy, Scott L., Cho, Yoon-Jae
Published in Neuro-oncology (Charlottesville, Va.) (01.02.2011)
Published in Neuro-oncology (Charlottesville, Va.) (01.02.2011)
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Correction: Bromodomain inhibition of the transcriptional coactivators CBP/EP300 as a therapeutic strategy to target the IRF4 network in multiple myeloma
Conery, Andrew R, Centore, Richard C, Neiss, Adrianne, Keller, Patricia J, Joshi, Shivangi, Spillane, Kerry L, Sandy, Peter, Hatton, Charlie, Pardo, Eneida, Zawadzke, Laura, Bommi-Reddy, Archana, Gascoigne, Karen E, Bryant, Barbara M, Mertz, Jennifer A, Sims, Robert J
Published in eLife (14.07.2016)
Published in eLife (14.07.2016)
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Discovery of Benzotriazolo[4,3‑d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains
Taylor, Alexander M, Vaswani, Rishi G, Gehling, Victor S, Hewitt, Michael C, Leblanc, Yves, Audia, James E, Bellon, Steve, Cummings, Richard T, Côté, Alexandre, Harmange, Jean-Christophe, Jayaram, Hari, Joshi, Shivangi, Lora, Jose M, Mertz, Jennifer A, Neiss, Adrianne, Pardo, Eneida, Nasveschuk, Christopher G, Poy, Florence, Sandy, Peter, Setser, Jeremy W, Sims, Robert J, Tang, Yong, Albrecht, Brian K
Published in ACS medicinal chemistry letters (11.02.2016)
Published in ACS medicinal chemistry letters (11.02.2016)
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Neuralized1 causes apoptosis and downregulates Notch target genes in medulloblastoma
Teider, Natalia, Scott, Deborah K., Neiss, Adrianne, Weeraratne, S. Dilhan, Amani, Vladimir M., Wang, Yifei, Marquez, Victor E., Cho, Yoon-Jae, Pomeroy, Scott L.
Published in Neuro-oncology (Charlottesville, Va.) (01.12.2010)
Published in Neuro-oncology (Charlottesville, Va.) (01.12.2010)
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GNE-064: A Potent, Selective, and Orally Bioavailable Chemical Probe for the Bromodomains of SMARCA2 and SMARCA4 and the Fifth Bromodomain of PBRM1
Taylor, Alexander M., Bailey, Chris, Belmont, Lisa D., Campbell, Robert, Cantone, Nico, Côté, Alexandre, Crawford, Terry D., Cummings, Richard, DeMent, Kevin, Duplessis, Martin, Flynn, Megan, Good, Andrew C., Huang, Hon-Ren, Joshi, Shivangi, Leblanc, Yves, Murray, Jeremy, Nasveschuk, Christopher G., Neiss, Adrianne, Poy, Florence, Romero, F. Anthony, Sandy, Peter, Tang, Yong, Tsui, Vickie, Zawadzke, Laura, Sims, Robert J., Audia, James E., Bellon, Steven F., Magnuson, Steven R., Albrecht, Brian K., Cochran, Andrea G.
Published in Journal of medicinal chemistry (25.08.2022)
Published in Journal of medicinal chemistry (25.08.2022)
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Abstract A20: A leukemic model of acquired resistance to BET inhibition reveals a role for CBP/EP300 bromodomains in the regulation of c-MYC expression
Conery, Andrew R., Centore, Richard C., Hatton, Charlie, Neiss, Adrianne, Huang, Hon-Ren, Keller, Patricia J., Taylor, Alexander M., Cote, Alexandre, Hewitt, Michael C., Nasveschuk, Christopher G., Leblanc, Yves, Yao, Shihua, Pardo, Eneida, Zawadzke, Laura, Poy, Florence, Jayaram, Hari, Joshi, Shivangi, Sandy, Peter, Romero, Anthony, Crawford, Terry, Pastor, Richard, Lai, Tommy, Chen, Kevin, Wang, Jian, Magnuson, Steven, Albrecht, Brian K., Bellon, Steve, Bryant, Barbara M., Sims, Robert J.
Published in Molecular cancer research (01.10.2015)
Published in Molecular cancer research (01.10.2015)
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