A functional genomics predictive network model identifies regulators of inflammatory bowel disease
Peters, Lauren A, Perrigoue, Jacqueline, Mortha, Arthur, Iuga, Alina, Song, Won-min, Neiman, Eric M, Llewellyn, Sean R, Di Narzo, Antonio, Kidd, Brian A, Telesco, Shannon E, Zhao, Yongzhong, Stojmirovic, Aleksandar, Sendecki, Jocelyn, Shameer, Khader, Miotto, Riccardo, Losic, Bojan, Shah, Hardik, Lee, Eunjee, Wang, Minghui, Faith, Jeremiah J, Kasarskis, Andrew, Brodmerkel, Carrie, Curran, Mark, Das, Anuk, Friedman, Joshua R, Fukui, Yoshinori, Humphrey, Mary Beth, Iritani, Brian M, Sibinga, Nicholas, Tarrant, Teresa K, Argmann, Carmen, Hao, Ke, Roussos, Panos, Zhu, Jun, Zhang, Bin, Dobrin, Radu, Mayer, Lloyd F, Schadt, Eric E
Published in Nature genetics (01.10.2017)
Published in Nature genetics (01.10.2017)
Get full text
Journal Article
The Novel SMAC Mimetic Birinapant Exhibits Potent Activity against Human Melanoma Cells
KREPLER, Clemens, CHUNDURU, Srinivas K, NATHANSON, Katherine L, AMARAVADI, Ravi K, PEHAMBERGER, Hubert, MCKINLAY, Mark, HERLYN, Meenhard, HALLORAN, Molly B, XU HE, MIN XIAO, VULTUR, Adina, VILLANUEVA, Jessie, MITSUUCHI, Yasuhiro, NEIMAN, Eric M, BENETATOS, Christopher
Published in Clinical cancer research (01.04.2013)
Published in Clinical cancer research (01.04.2013)
Get full text
Journal Article
Gene coexpression networks reveal a broad role for lncRNAs in inflammatory bowel disease
Johnson, John L, Sargsyan, Davit, Neiman, Eric M, Hart, Amy, Stojmirovic, Aleksandar, Kosoy, Roman, Irizar, Haritz, Suárez-Fariñas, Mayte, Song, Won-Min, Argmann, Carmen, Avey, Stefan, Shmuel-Galia, Liraz, Vierbuchen, Tim, Bongers, Gerold, Sun, Yu, Edelstein, Leonard, Perrigoue, Jacqueline, Towne, Jennifer E, Hall, Aisling O'Hara, Fitzgerald, Katherine A, Hoebe, Kasper
Published in JCI insight (08.02.2024)
Published in JCI insight (08.02.2024)
Get full text
Journal Article
Su1858 Integrative Networks Identify Novel Regulators of Susceptibility and Pathogenesis of Inflammatory Bowel Disease
Peters, Lauren, Perrigoue, Jacqueline, Mortha, Arthur, Stojmirovic, Aleksandar, Neiman, Eric M, Iuga, Alina, Song, Won-min, Kidd, Brian A, Losic, Bojan, Llewellyn, Sean, Miotto, Riccardo, Shameer, Khader, Zhao, Yongzhong, Di Narzo, Antonio, Shah, Hardik, Cohain, Ariella, Dudley, Joel T, Faith, Jeremiah, Merad, Miriam, Fukui, Fumiyuki, Iritani, Brian, Sibinga, Nicholas, Tarrant, Teresa, Argmann, Carmen, Kasarskis, Andrew, Curran, Mark, Das, Anuk, Dobrin, Radu, Hao, Ke, Roussos, Panos, Zhang, Bin, Zhu, Jun, Mayer, Lloyd F, Friedman, Joshua, Schadt, Eric E
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
Get full text
Journal Article
Birinapant (TL32711), a bivalent SMAC mimetic, targets TRAF2-associated cIAPs, abrogates TNF-induced NF-κB activation, and is active in patient-derived xenograft models
Benetatos, Christopher A, Mitsuuchi, Yasuhiro, Burns, Jennifer M, Neiman, Eric M, Condon, Stephen M, Yu, Guangyao, Seipel, Martin E, Kapoor, Gurpreet S, Laporte, Matthew G, Rippin, Susan R, Deng, Yijun, Hendi, Mukta S, Tirunahari, Pavan K, Lee, Yu-Hua, Haimowitz, Thomas, Alexander, Matthew D, Graham, Martin A, Weng, David, Shi, Yigong, McKinlay, Mark A, Chunduru, Srinivas K
Published in Molecular cancer therapeutics (01.04.2014)
Published in Molecular cancer therapeutics (01.04.2014)
Get full text
Journal Article
Abstract 2278: The SMAC-mimetic birinapant regulates autocrine TNF production by caspase-8:RIPK1 complex via p38MAPK pathway
Kapoor, Gurpreet Singh, Benetatos, Christopher A., Mitsuuchi, Yasuhiro, Neiman, Eric M., Yu, Guangyao, Mckinlay, Mark A., Burns, Jennifer, Silke, John, Condon, Stephen M., Chunduru, Srinivas K.
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Get full text
Journal Article
Abstract 599: Potential biomarkers of Smac mimetic tumor sensitivity: inhibitor of apoptosis protein DNA copy number
Kapoor, Gurpreet S., Geier, Brian, Neiman, Eric M., Mitsuuchi, Yasuhiro, Benetatos, Christopher A., Condon, Stephen M., Chunduru, Srinivas, Begley, C. Glenn
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article
Abstract 5302: Characterization of tumor cell lines resistant to birinapant, a novel bivalent smac mimetic
Neiman, Eric M., Benetatos, Christopher A., Kapoor, Gurpreet S., Mitsuuchi, Yasuhiro, McKinlay, Mark A., Seipel, Martin E., Yu, Guangyao, Condon, Stephen M., Chunduru, Srinivas K.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article
Abstract 3336: The Smac Mimetic Birinapant Synergistically Induces Apoptosis in Combination with Type I Interferons and GM-CSF
Benetatos, Christopher A., Burns, Jennifer M., Borden, Ernest C., Lindner, Daniel, Mitsuuchi, Yasuhiro, Mckinlay, Mark A., Kapoor, Gurpreet Singh, Neiman, Eric M., Seipel, Martin E., Yu, Guangyao, Graham, Martin, Weng, David, Condon, Stephen M., Begley, C. Glenn, Chunduru, Srinivas
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article
Abstract 3333: Birinapant, a novel bivalent Smac mimetic drug, is superior to monovalent Smac mimetics in inhibition of NF-kB by targeting TRAF2-bound cIAP1 and cIAP2
Mitsuuchi, Yasuhiro, Condon, Stephen M., Neiman, Eric M., Benetatos, Christopher A., Seipel, Martin E., Kapoor, Gurpreet Singh, Mufalli, Angeline C., Yu, Guangyao, Maguire, Orla, Minderman, Hans, Mckinlay, Mark A., Graham, Martin, Weng, David, Chunduru, Srinivas
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article