Discovery of MDV6058 (PF-06952229), a selective and potent TGFβR1 inhibitor: Design, synthesis and optimization
Pujala, Brahmam, Ramachandran, Sreekanth A., Sonawane, Mukesh, Kamble, Maruti M., Panpatil, Dayanand, Adhikari, Swati, Soni, Sanjeev, Subbareddy, Venkata, Shinde, Bharat U., Nayak, Anjan K., Bansal, Chandni, Gupta, Ashu, Mukherjee, Kakoli, Agarwal, Anil K., Guerrero, Javier, Herrera, Francisco J., Bernales, Sebastian, Guha, Mausumee, Chakravarty, Sarvajit, Pham, Son M., Rai, Roopa
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Targeting prostate cancer with compounds possessing dual activity as androgen receptor antagonists and HDAC6 inhibitors
Jadhavar, Pradeep S., Ramachandran, Sreekanth A., Riquelme, Eduardo, Gupta, Ashu, Quinn, Kevin P., Shivakumar, Devleena, Ray, Soumya, Zende, Dnyaneshwar, Nayak, Anjan K., Miglani, Sandeep K., Sathe, Balaji D., Raja, Mohd, Farias, Olivia, Alfaro, Ivan, Belmar, Sebastián, Guerrero, Javier, Bernales, Sebastián, Chakravarty, Sarvajit, Hung, David T., Lindquist, Jeffrey N., Rai, Roopa
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
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Journal Article
Dual Inhibition of Bruton's Tyrosine Kinase and Phosphoinositide-3-Kinase p110 δ as a Therapeutic Approach to Treat Non-Hodgkin's B Cell Malignancies
Alfaro, Jennifer, Pérez de Arce, Felipe, Belmar, Sebastián, Fuentealba, Glenda, Avila, Patricio, Ureta, Gonzalo, Flores, Camila, Acuña, Claudia, Delgado, Luz, Gaete, Diana, Pujala, Brahmam, Barde, Anup, Nayak, Anjan K, Upendra, T V R, Patel, Dhananjay, Chauhan, Shailender, Sharma, Vijay K, Kanno, Stacy, Almirez, Ramona G, Hung, David T, Chakravarty, Sarvajit, Rai, Roopa, Bernales, Sebastián, Quinn, Kevin P, Pham, Son M, McCullagh, Emma
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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Discovery of Pyrazolopyrimidine Derivatives as Novel Dual Inhibitors of BTK and PI3Kδ
Pujala, Brahmam, Agarwal, Anil K, Middya, Sandip, Banerjee, Monali, Surya, Arjun, Nayak, Anjan K, Gupta, Ashu, Khare, Sweta, Guguloth, Rambabu, Randive, Nitin A, Shinde, Bharat U, Thakur, Anamika, Patel, Dhananjay I, Raja, Mohd, Green, Michael J, Alfaro, Jennifer, Avila, Patricio, Pérez de Arce, Felipe, Almirez, Ramona G, Kanno, Stacy, Bernales, Sebastián, Hung, David T, Chakravarty, Sarvajit, McCullagh, Emma, Quinn, Kevin P, Rai, Roopa, Pham, Son M
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
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Journal Article
Discovery of MDV6058 (PF-06952229), a selective and potent TGF?R1 inhibitor: Design, synthesis and optimization
Pujala, Brahmam, Ramachandran, Sreekanth A., Sonawane, Mukesh, Kamble, Maruti M., Panpatil, Dayanand, Adhikari, Swati, Soni, Sanjeev, Subbareddy, Venkata, Shinde, Bharat U., Nayak, Anjan K., Bansal, Chandni, Gupta, Ashu, Mukherjee, Kakoli, Agarwal, Anil K., Guerrero, Javier, Herrera, Francisco J., Bernales, Sebastian, Guha, Mausumee, Chakravarty, Sarvajit, Pham, Son M., Rai, Roopa
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Journal Article