Search Results - "Nawrozkij, Maxim B" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

by Mozhaitsev, Evgenii S, Suslov, Evgeniy V, Rastrepaeva, Daria A, Yarovaya, Olga I, Borisevich, Sophia S, Khamitov, Edward M, Kolybalov, Dmitry S, Arkhipov, Sergey G, Bormotov, Nikolai I, Shishkina, Larisa N, Serova, Olga A, Brunilin, Roman V, Vernigora, Andrey A, Nawrozkij, Maxim B, Agafonov, Alexander P, Maksyutov, Rinat A, Volcho, Konstantin P, Salakhutdinov, Nariman F
Published in Viruses (21.12.2022)

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Structural insight into the optimization of ethyl 5-hydroxybenzo[g]indol-3-carboxylates and their bioisosteric analogues as 5-LO/m-PGES-1 dual inhibitors able to suppress inflammation

Structural insight into the optimization of ethyl 5-hydroxybenzo[g]indol-3-carboxylates and their bioisosteric analogues as 5-LO/m-PGES-1 dual inhibitors able to suppress inflammation

by Bruno, Ferdinando, Errico, Suann, Pace, Simona, Nawrozkij, Maxim B., Mkrtchyan, Arthur S., Guida, Francesca, Maisto, Rosa, Olgaç, Abdurrahman, D'Amico, Michele, Maione, Sabatino, De Rosa, Mario, Banoglu, Erden, Werz, Oliver, Fiorentino, Antonio, Filosa, Rosanna
Published in European journal of medicinal chemistry (15.07.2018)

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Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity

Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity

by Fioravanti, Rossella, Proia, Eleonora, Tyurenkov, Ivan N., Kurkin, Denis V., Bakulin, Dmitry A., Kovalev, Nikolay S., Sheikin, Dmitry S., Kirillov, Ivan A., Nawrozkij, Maxim B., Vernigora, Andrey A., Brunilina, Leila L., Fiorentino, Francesco, Mladenović, Milan, Rotili, Dante, Ragno, Rino
Published in European journal of medicinal chemistry (05.01.2023)

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Effect of α‑Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3H)‑ones

Effect of α‑Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3H)‑ones

by Nawrozkij, Maxim B, Forgione, Mariantonietta, Yablokov, Alexandre S, Lucidi, Alessia, Tomaselli, Daniela, Patsilinakos, Alexandros, Panella, Cristina, Hailu, Gebremedhin S, Kirillov, Ivan A, Badia, Roger, Riveira-Muñoz, Eva, Crespan, Emmanuele, Armijos Rivera, Jorge I, Cirilli, Roberto, Ragno, Rino, Esté, José A, Maga, Giovanni, Mai, Antonello, Rotili, Dante
Published in Journal of medicinal chemistry (24.01.2019)

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Design, Synthesis, and Biological Evaluation of (+)‐Camphor‐ and (−)‐Fenchone‐Based Derivatives as Potent Orthopoxvirus Inhibitors

Design, Synthesis, and Biological Evaluation of (+)‐Camphor‐ and (−)‐Fenchone‐Based Derivatives as Potent Orthopoxvirus Inhibitors

by Sokolova, Anastasiya S., Kovaleva, Kseniya S., Kuranov, Sergey O., Bormotov, Nikolay I., Borisevich, Sophia S., Zhukovets, Anastasiya A., Yarovaya, Olga I., Serova, Olga A., Nawrozkij, Maxim B., Vernigora, Andrey A., Davidenko, Andrey V., Khamitov, Eduard M., Peshkov, Roman Y., Shishkina, Larisa N., Maksuytov, Rinat A., Salakhutdinov, Nariman F.
Published in ChemMedChem (20.06.2022)

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Diarylpyrimidine−Dihydrobenzyloxopyrimidine Hybrids: New, Wide-Spectrum Anti-HIV-1 Agents Active at (Sub)-Nanomolar Level

Diarylpyrimidine−Dihydrobenzyloxopyrimidine Hybrids: New, Wide-Spectrum Anti-HIV-1 Agents Active at (Sub)-Nanomolar Level

by Rotili, Dante, Tarantino, Domenico, Artico, Marino, Nawrozkij, Maxim B, Gonzalez-Ortega, Emmanuel, Clotet, Bonaventura, Samuele, Alberta, Esté, José A, Maga, Giovanni, Mai, Antonello
Published in Journal of medicinal chemistry (28.04.2011)

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Arbidol: a quarter-century after. Past, present and future of the original Russian antiviral

Arbidol: a quarter-century after. Past, present and future of the original Russian antiviral

by Balakin, Konstantin V., Filosa, Rosanna, Lavrenov, Sergey N., Mkrtchyan, Arthur S., Nawrozkij, Maxim B., Novakov, Ivan A.
Published in Russian chemical reviews (01.06.2018)

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Exploring the Role of 2‑Chloro-6-fluoro Substitution in 2‑Alkylthio-6-benzyl-5-alkylpyrimidin-4(3H)‑ones: Effects in HIV-1-Infected Cells and in HIV‑1 Reverse Transcriptase Enzymes

Exploring the Role of 2‑Chloro-6-fluoro Substitution in 2‑Alkylthio-6-benzyl-5-alkylpyrimidin-4(3H)‑ones: Effects in HIV-1-Infected Cells and in HIV‑1 Reverse Transcriptase Enzymes

by Rotili, Dante, Tarantino, Domenico, Nawrozkij, Maxim B, Babushkin, Alexandre S, Botta, Giorgia, Marrocco, Biagina, Cirilli, Roberto, Menta, Sergio, Badia, Roger, Crespan, Emmanuele, Ballante, Flavio, Ragno, Rino, Esté, José A, Maga, Giovanni, Mai, Antonello
Published in Journal of medicinal chemistry (26.06.2014)

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2-(Alkyl/Aryl)Amino-6-Benzylpyrimidin-4(3H)-ones as Inhibitors of Wild-Type and Mutant HIV-1: Enantioselectivity Studies

2-(Alkyl/Aryl)Amino-6-Benzylpyrimidin-4(3H)-ones as Inhibitors of Wild-Type and Mutant HIV-1: Enantioselectivity Studies

by Rotili, Dante, Samuele, Alberta, Tarantino, Domenico, Ragno, Rino, Musmuca, Ira, Ballante, Flavio, Botta, Giorgia, Morera, Ludovica, Pierini, Marco, Cirilli, Roberto, Nawrozkij, Maxim B, Gonzalez, Emmanuel, Clotet, Bonaventura, Artico, Marino, Esté, José A, Maga, Giovanni, Mai, Antonello
Published in Journal of medicinal chemistry (12.04.2012)

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Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains

Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains

by Mai, Antonello, Artico, Marino, Rotili, Dante, Tarantino, Domenico, Clotet-Codina, Imma, Armand-Ugón, Mercedes, Ragno, Rino, Simeoni, Silvia, Sbardella, Gianluca, Nawrozkij, Maxim B, Samuele, Alberta, Maga, Giovanni, Esté, José A
Published in Journal of medicinal chemistry (01.11.2007)

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5-Alkyl-6-benzyl-2-(2-oxo-2-phenylethylsulfanyl)pyrimidin-4(3H)-ones, a Series of Anti-HIV-1 Agents of the Dihydro-alkoxy-benzyl-oxopyrimidine Family with Peculiar Structure−Activity Relationship Profile

by Nawrozkij, Maxim B, Rotili, Dante, Tarantino, Domenico, Botta, Giorgia, Eremiychuk, Alexandre S, Musmuca, Ira, Ragno, Rino, Samuele, Alberta, Zanoli, Samantha, Armand-Ugón, Mercedes, Clotet-Codina, Imma, Novakov, Ivan A, Orlinson, Boris S, Maga, Giovanni, Esté, José A, Artico, Marino, Mai, Antonello
Published in Journal of medicinal chemistry (14.08.2008)

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The synthesis of new acyclic analogs of 3-phenacyluridine and comparative evaluation of their in vivo biological activity

The synthesis of new acyclic analogs of 3-phenacyluridine and comparative evaluation of their in vivo biological activity

by Novakov, Ivan А., Brunilina, Leila L., Kirillov, Ivan А., Nawrozkij, Maxim B., Robinovich, Mariya D., Titova, Evgeniya S., Sheikin, Dmitry S., Ruchko, Evsey А., Pavlova, Alla V., Kotlyarova, Anastasiya А., Tolstikova, Tatyana G.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.06.2020)

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Structural insight into the optimization of ethyl 5-hydroxybenzo[g] indol-3-carboxylates and their bioisosteric analogues as 5-LO/mPGES-1 dual inhibitors able to suppress inflammation

Structural insight into the optimization of ethyl 5-hydroxybenzo[g] indol-3-carboxylates and their bioisosteric analogues as 5-LO/mPGES-1 dual inhibitors able to suppress inflammation

by Bruno, Ferdinando, Errico, Suann, Pace, Simona, Nawrozkij, Maxim B., Mkrtchyan, Arthur S., Guida, Francesca, Maisto, Rosa, Olgac, Abdurrahman, D'Amico, Michele, Maione, Sabatino, De Rosa, Mario, Banoglu, Erden, Werz, Oliver, Fiorentino, Antonio, Filosa, Rosanna
Published in European journal of medicinal chemistry (15.07.2018)

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A Practical Synthesis of 4’-Fluorospiro[cyclopropane-1,3’-indol]-2’(1’H)-one: a Valuable Terminal Building-Block for Biologically Active Podands

A Practical Synthesis of 4’-Fluorospiro[cyclopropane-1,3’-indol]-2’(1’H)-one: a Valuable Terminal Building-Block for Biologically Active Podands

by Babushkin, Alexandre S., Nawrozkij, Maxim B., Novakov, Ivan A., Yablokov, Alexandre S.
Published in Macroheterocycles (2016)

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Convenient Synthesis of Building-Blocks for Pyridine/Piperidine-Decorated Crown Ethers

Convenient Synthesis of Building-Blocks for Pyridine/Piperidine-Decorated Crown Ethers

by Nawrozkij, Maxim B., Gorbunov, Evgeniy B., Babushkin, Alexandre S., Ruchko, Evsey A., Rusinov, Gennadiy L., Charushin, Valeriy N., Novakov, Ivan A.
Published in Macroheterocycles (2014)

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5-Alkyl-6-benzyl-2-(2-oxo-2-phenylethylsulfanyl)pyrimidin-4(3H)-ones, a Series of Anti-HIV-1 Agents of the Dihydro-alkoxy-benzyl-oxopyrimidine Family with Peculiar Structure-Activity Relationship Profile

by NAWROZKIJ, Maxim B, ROTILI, Dante, CLOTET-CODINA, Imma, NOVAKOV, Ivan A, ORLINSON, Boris S, MAGA, Giovanni, ESTE, José A, ARTICO, Marino, MAI, Antonello, TARANTINO, Domenico, BOTTA, Giorgia, EREMIYCHUK, Alexandre S, MUSMUCA, Ira, RAGNO, Rino, SAMUELE, Alberta, ZANOLI, Samantha, ARMAND-UGON, Mercedes
Published in Journal of medicinal chemistry (2008)

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