Basmisanil, a highly selective GABAA-α5 negative allosteric modulator: preclinical pharmacology and demonstration of functional target engagement in man
Hipp, Joerg F., Knoflach, Frederic, Comley, Robert, Ballard, Theresa M., Honer, Michael, Trube, Gerhard, Gasser, Rodolfo, Prinssen, Eric, Wallace, Tanya L., Rothfuss, Andreas, Knust, Henner, Lennon-Chrimes, Sian, Derks, Michael, Bentley, Darren, Squassante, Lisa, Nave, Stephane, Nöldeke, Jana, Wandel, Christoph, Thomas, Andrew W., Hernandez, Maria-Clemencia
Published in Scientific reports (08.04.2021)
Published in Scientific reports (08.04.2021)
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Recommendations for the use of Serious Games in people with Alzheimer's Disease, related disorders and frailty
Robert, Philippe H, König, Alexandra, Amieva, Hélene, Andrieu, Sandrine, Bremond, François, Bullock, Roger, Ceccaldi, Mathieu, Dubois, Bruno, Gauthier, Serge, Kenigsberg, Paul-Ariel, Nave, Stéphane, Orgogozo, Jean M, Piano, Julie, Benoit, Michel, Touchon, Jacques, Vellas, Bruno, Yesavage, Jerome, Manera, Valeria
Published in Frontiers in aging neuroscience (24.03.2014)
Published in Frontiers in aging neuroscience (24.03.2014)
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Sembragiline: A Novel, Selective Monoamine Oxidase Type B Inhibitor for the Treatment of Alzheimer’s Disease
Borroni, Edilio, Bohrmann, Bernd, Grueninger, Fiona, Prinssen, Eric, Nave, Stephane, Loetscher, Hansruedi, Chinta, Shankar J, Rajagopalan, Subramanian, Rane, Anand, Siddiqui, Almas, Ellenbroek, Bart, Messer, Juerg, Pähler, Axel, Andersen, Julie K, Wyler, Rene, Cesura, Andrea M
Published in The Journal of pharmacology and experimental therapeutics (01.09.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2017)
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Enhanced dopamine availability and response readiness. The influence of 3 doses of methylphenidate on contingent negative variation in the EEG of healthy volunteers
Linssen, Anke, Vuurman, Eric, Sambeth, Anke, Navé, Stephane, Riedel, Wim
Published in Neuroscience letters (01.08.2011)
Published in Neuroscience letters (01.08.2011)
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Single Ascending Dose Tolerability, Pharmacokinetic–Pharmacodynamic Study of Dihydropyrimidine Dehydrogenase Inhibitor Ro 09-4889
BELLIBAS, S. Eralp, PATEL, Indra, CHAMOREY, Emmanuel, BRIVET, Bettyna, BUSH, Ernest D, KIRCHER, Catherine, NAVE, Stephane, BANKEN, Ludger, RENEE, Nicole, MILANO, Gérard
Published in Clinical cancer research (01.04.2004)
Published in Clinical cancer research (01.04.2004)
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Haematological effects of oral administration of bitopertin, a glycine transport inhibitor, in patients with non‐transfusion‐dependent β‐thalassaemia
Taher, Ali T., Viprakasit, Vip, Cappellini, Maria Domenica, Kraus, Dominik, Cech, Patrick, Volz, Dietmar, Winter, Erica, Nave, Stephane, Dukart, Juergen, Khwaja, Omar, Koerner, Annette, Hermosilla, Ricardo, Brugnara, Carlo
Published in British journal of haematology (01.07.2021)
Published in British journal of haematology (01.07.2021)
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General Principles for the Validation of Proarrhythmia Risk Prediction Models: An Extension of the CiPA In Silico Strategy
Li, Zhihua, Mirams, Gary R., Yoshinaga, Takashi, Ridder, Bradley J., Han, Xiaomei, Chen, Janell E., Stockbridge, Norman L., Wisialowski, Todd A., Damiano, Bruce, Severi, Stefano, Morissette, Pierre, Kowey, Peter R., Holbrook, Mark, Smith, Godfrey, Rasmusson, Randall L., Liu, Michael, Song, Zhen, Qu, Zhilin, Leishman, Derek J., Steidl‐Nichols, Jill, Rodriguez, Blanca, Bueno‐Orovio, Alfonso, Zhou, Xin, Passini, Elisa, Edwards, Andrew G., Morotti, Stefano, Ni, Haibo, Grandi, Eleonora, Clancy, Colleen E., Vandenberg, Jamie, Hill, Adam, Nakamura, Mikiko, Singer, Thomas, Polonchuk, Liudmila, Greiter‐Wilke, Andrea, Wang, Ken, Nave, Stephane, Fullerton, Aaron, Sobie, Eric A., Paci, Michelangelo, Musuamba Tshinanu, Flora, Strauss, David G.
Published in Clinical pharmacology and therapeutics (01.01.2020)
Published in Clinical pharmacology and therapeutics (01.01.2020)
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Sembragiline in Moderate Alzheimer's Disease: Results of a Randomized, Double-Blind, Placebo-Controlled Phase II Trial (MAyflOwer RoAD)
Nave, Stephane, Doody, Rachelle S, Boada, Mercè, Grimmer, Timo, Savola, Juha-Matti, Delmar, Paul, Pauly-Evers, Meike, Nikolcheva, Tania, Czech, Christian, Borroni, Edilio, Ricci, Benedicte, Dukart, Juergen, Mannino, Marie, Carey, Tracie, Moran, Emma, Gilaberte, Inma, Muelhardt, Nicoletta Milani, Gerlach, Irene, Santarelli, Luca, Ostrowitzki, Susanne, Fontoura, Paulo
Published in Journal of Alzheimer's disease (01.01.2017)
Published in Journal of Alzheimer's disease (01.01.2017)
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Phase 2 Clinical Trial Results for Bitopertin, an Oral Glycine Transporter 1 Inhibitor, in Patients with Non-Transfusion Dependent Beta-Thalassemia
Taher, Ali, Viprakasit, Vip, Cappellini, Maria Domenica, Kraus, Dominik, Cech, Patrick, Dietmar, Volz, Winter, Erica, Mazer, Norman Alan, Nave, Stephane, Dukart, Juergen, Schaedeli Stark, Franziska, Koerner, Annette, Khwaja, Omar, Hermosilla, Ricardo
Published in Blood (29.11.2018)
Published in Blood (29.11.2018)
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Positron emission tomography measurement of brain MAO-B inhibition in patients with Alzheimer’s disease and elderly controls after oral administration of sembragiline
Sturm, Stefan, Forsberg, Anton, Nave, Stephane, Stenkrona, Per, Seneca, Nicholas, Varrone, Andrea, Comley, Robert A., Fazio, Patrik, Jamois, Candice, Nakao, Ryuji, Ejduk, Zbigniew, Al-Tawil, Nabil, Akenine, Ulrika, Halldin, Christer, Andreasen, Niels, Ricci, Benedicte
Published in European journal of nuclear medicine and molecular imaging (01.03.2017)
Published in European journal of nuclear medicine and molecular imaging (01.03.2017)
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Contingent negative variation as a dopaminergic biomarker: evidence from dose-related effects of methylphenidate
Linssen, Anke M. W., Vuurman, Eric F. P. M., Sambeth, Anke, Nave, Stephane, Spooren, Will, Vargas, Gabriel, Santarelli, Luca, Riedel, Wim J.
Published in Psychopharmacologia (01.12.2011)
Published in Psychopharmacologia (01.12.2011)
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Risdiplam treatment has not led to retinal toxicity in patients with spinal muscular atrophy
Sergott, Robert C., Amorelli, Giulia M., Baranello, Giovanni, Barreau, Emmanuel, Beres, Shannon, Kane, Steven, Mercuri, Eugenio, Orazi, Lorenzo, SantaMaria, Melissa, Tremolada, Gemma, Santarsiero, Diletta, Waskowska, Agnieszka, Yashiro, Shigeko, Denk, Nora, Fürst‐Recktenwald, Sabine, Gerber, Marianne, Gorni, Ksenija, Jaber, Birgit, Jacobsen, Bjoern, Mueller, Lutz, Nave, Stephane, Scalco, Renata S., Marzoli, Stefania B.
Published in Annals of clinical and translational neurology (01.01.2021)
Published in Annals of clinical and translational neurology (01.01.2021)
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Preclinical characterization of RO4602522, a novel, selective and orally active monoamine oxidase type B inhibitor for the treatment of Alzheimer's disease
Borroni, Edilio, Wyler, Rene, Messer, Juergen, Nave, Stephane, Cesura, Andrea
Published in Alzheimer's & dementia (01.07.2013)
Published in Alzheimer's & dementia (01.07.2013)
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P4–312: Preclinical characterization of RO4602522, a novel, selective and orally active monoamine oxidase type B inhibitor for the treatment of Alzheimer's disease
Borroni, Edilio, Wyler, Rene, Messer, Juergen, Nave, Stephane, Cesura, Andrea
Published in Alzheimer's & dementia (01.07.2013)
Published in Alzheimer's & dementia (01.07.2013)
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Basmisanil, a highly selective GABA A -α5 negative allosteric modulator: preclinical pharmacology and demonstration of functional target engagement in man
Hipp, Joerg F, Knoflach, Frederic, Comley, Robert, Ballard, Theresa M, Honer, Michael, Trube, Gerhard, Gasser, Rodolfo, Prinssen, Eric, Wallace, Tanya L, Rothfuss, Andreas, Knust, Henner, Lennon-Chrimes, Sian, Derks, Michael, Bentley, Darren, Squassante, Lisa, Nave, Stephane, Nöldeke, Jana, Wandel, Christoph, Thomas, Andrew W, Hernandez, Maria-Clemencia
Published in Scientific reports (08.04.2021)
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Published in Scientific reports (08.04.2021)
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Sembragiline: A Novel, Selective Monoamine Oxidase Type B Inhibitor for the Treatment of Alzheimer's Disease
Borroni, Edilio, Bohrmann, Bernd, Grueninger, Fiona, Prinssen, Eric, Nave, Stephane, Loetscher, Hansruedi, Chinta, Shankar J, Rajagopalan, Subramanian, Rane, Anand, Siddiqui, Almas, Ellenbroek, Bart, Messer, Juerg, Pähler, Axel, Andersen, Julie K, Wyler, Rene, Cesura, Andrea M
Published in The Journal of pharmacology and experimental therapeutics (01.09.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2017)
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Brain MAO-B inhibition in healthy elderly and people with Alzheimer's disease after oral administration of RO4602522
Ricci, Benedicte, Sturm, Stefan, Seneca, Nicholas, Jamois, Candice, Nave, Stephane, Ejduk, Zbigniew, Skenkrona, Per, Varonne, Andrea, Forsberg, Anton, Fazio, Patrik, Halldin, Christer, Al-Tawil, Nabil, Akenine, Ulrika, Andreasen, Niels
Published in Alzheimer's & dementia (01.07.2013)
Published in Alzheimer's & dementia (01.07.2013)
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P3–300: Brain MAO‐B inhibition in healthy elderly and people with Alzheimer's disease after oral administration of RO4602522
Ricci, Benedicte, Sturm, Stefan, Seneca, Nicholas, Jamois, Candice, Nave, Stephane, Ejduk, Zbigniew, Skenkrona, Per, Varonne, Andrea, Forsberg, Anton, Fazio, Patrik, Halldin, Christer, Al‐Tawil, Nabil, Akenine, Ulrika, Andreasen, Niels
Published in Alzheimer's & dementia (01.07.2013)
Published in Alzheimer's & dementia (01.07.2013)
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Intravenous dolasetron mesilate in the prevention of postoperative nausea and vomiting in females undergoing gynecological surgery
Diemunsch, Pierre, D'Hollander, Alain, Paxton, Lionel, Schoeffler, Pierre, Wessel, Pierrette, Navé, Stephane, Brown, Robert A., Hahne, William F.
Published in Journal of clinical anesthesia (01.08.1997)
Published in Journal of clinical anesthesia (01.08.1997)
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