Racemisation in Chemistry and Biology
Ballard, Andrew, Narduolo, Stefania, Ahmed, Hiwa O., Keymer, Nathaniel I., Asaad, Nabil, Cosgrove, David A., Buurma, Niklaas J., Leach, Andrew G.
Published in Chemistry : a European journal (23.03.2020)
Published in Chemistry : a European journal (23.03.2020)
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Frontispiece: Racemisation in Chemistry and Biology
Ballard, Andrew, Narduolo, Stefania, Ahmed, Hiwa O., Keymer, Nathaniel I., Asaad, Nabil, Cosgrove, David A., Buurma, Niklaas J., Leach, Andrew G.
Published in Chemistry : a European journal (23.03.2020)
Published in Chemistry : a European journal (23.03.2020)
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Quantitative Prediction of Rate Constants for Aqueous Racemization To Avoid Pointless Stereoselective Syntheses
Ballard, Andrew, Ahmad, Hiwa O., Narduolo, Stefania, Rosa, Lucy, Chand, Nikki, Cosgrove, David A., Varkonyi, Peter, Asaad, Nabil, Tomasi, Simone, Buurma, Niklaas J., Leach, Andrew G.
Published in Angewandte Chemie International Edition (22.01.2018)
Published in Angewandte Chemie International Edition (22.01.2018)
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The problem of racemization in drug discovery and tools to predict it
Ballard, Andrew, Narduolo, Stefania, Ahmad, Hiwa O, Cosgrove, David A, Leach, Andrew G, Buurma, Niklaas J
Published in Expert opinion on drug discovery (03.06.2019)
Published in Expert opinion on drug discovery (03.06.2019)
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Enantiomeric pairs reveal that key medicinal chemistry parameters vary more than simple physical property based models can explain
Leach, Andrew G., Pilling, Elizabeth A., Rabow, Alfred A., Tomasi, Simone, Asaad, Nabil, Buurma, Niklaas J., Ballard, Andrew, Narduolo, Stefania
Published in MedChemComm (01.05.2012)
Published in MedChemComm (01.05.2012)
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Abstracts of the 28th International Isotope Society (UK group) Symposium: The synthesis and applications of labelled compounds 2019
Nelson, Adam, Phipps, Robert J., Crane, Georgie J., Venanzi, Niccolo A.E., Lockley, William J.S., Tredwell, Matthew, Buurma, Niklaas J., Ballard, Andrew, Ahmad, Hiwa O., Narduolo, Stefania, Rosa, Lucy, Chand, Nikki, Cosgrove, David A., Varkonyi, Peter, Asaad, Nabil, Tomasi, Simone, Leach, Andrew G., Summerhill, Nick, Bloom, Jon, Newby, Mark, Madden, Stephen, Roman, Daniela, Exner, Ruediger M., Cortezon‐Tamarit, Fernando, Ge, Haobo, Paisey, Stephen, Pascu, Sofia I., Rosales, Rafael T.M., Hailes, Helen C., Wang, Yu, Zhao, Jianxiong, Méndez‐Sánchez, Daniel, Rodan, Rebecca, Subrizi, Fabiana, Lichman, Benjamin R., Keep, Nicholas H., Ward, John M., Harris, Mark, Lamb, Martin, Wilson, Vernon, Iafrate, Peter, Bulat, Flaviu, Néves, Andre A., Hesse, Friederike, Hu, De‐En, Aigbirhio, Franklin, Leeper, Finian J., Brindle, Kevin M., Rowbotham, Jack S., Urata, Koji, Reeve, Holly A., Vincent, Kylie A., Hueting, Rebekka
Published in Journal of labelled compounds & radiopharmaceuticals (01.12.2020)
Published in Journal of labelled compounds & radiopharmaceuticals (01.12.2020)
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Journal Article
Quantitative Prediction of Rate Constants for Aqueous Racemization To Avoid Pointless Stereoselective Syntheses
Ballard, Andrew, Ahmad, Hiwa O., Narduolo, Stefania, Rosa, Lucy, Chand, Nikki, Cosgrove, David A., Varkonyi, Peter, Asaad, Nabil, Tomasi, Simone, Buurma, Niklaas J., Leach, Andrew G.
Published in Angewandte Chemie (22.01.2018)
Published in Angewandte Chemie (22.01.2018)
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Journal Article
Abstracts of the 28 th International Isotope Society (UK group) Symposium: The Synthesis & Applications of Labelled Compounds 2019
Nelson, Adam, Phipps, Robert J, Crane, Georgie J, Venanzi, Niccolo A E, Lockley, William J S, Tredwell, Matthew, Buurma, Niklaas J, Ballard, Andrew, Ahmad, Hiwa O, Narduolo, Stefania, Rosa, Lucy, Chand, Nikki, Cosgrove, David A, Varkonyi, Peter, Asaad, Nabil, Tomasi, Simone, Leach, Andrew G, Summerhill, Nick, Bloom, Jon, Newby, Mark, Madden, Stephen, Roman, Daniela, Exner, Ruediger M, Cortezon-Tamarit, Fernando, Ge, Haobo, Paisey, Stephen, Pascu, Sofia I, de Rosales, Rafael T M, Hailes, Helen C, Wang, Yu, Zhao, Jianxiong, Méndez-Sánchez, Daniel, Rodan, Rebecca, Subrizi, Fabiana, Lichman, Benjamin R, Keep, Nicholas H, Ward, John M, Harris, Mark, Lamb, Martin, Wilson, Vernon, Iafrate, Peter, Bulat, Flaviu, Néves, Andre A, Hesse, Friederike, Hu, De-En, Aigbirhio, Franklin, Leeper, Finian J, Brindle, Kevin M, Rowbotham, Jack S, Urata, Koji, Reeve, Holly A, Vincent, Kylie A, Hueting, Rebekka
Published in Journal of labelled compounds & radiopharmaceuticals (17.07.2020)
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Published in Journal of labelled compounds & radiopharmaceuticals (17.07.2020)
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Enantiomeric pairs reveal that key medicinal chemistry parameters vary more than simple physical property based models can explainElectronic supplementary information (ESI) available: Description of the data sources mined in this work. See DOI: 10.1039/c2md20010d
Leach, Andrew G, Pilling, Elizabeth A, Rabow, Alfred A, Tomasi, Simone, Asaad, Nabil, Buurma, Niklaas J, Ballard, Andrew, Narduolo, Stefania
Year of Publication 02.05.2012
Year of Publication 02.05.2012
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