Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors
Chino, Ayaka, Seo, Ryushi, Amano, Yasushi, Namatame, Ichiji, Hamaguchi, Wataru, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki, Masuda, Naoyuki
Published in Chemical & pharmaceutical bulletin (2018)
Published in Chemical & pharmaceutical bulletin (2018)
Get full text
Journal Article
Stepwise Construction of Head-to-Tail-Type Oligothiophenes via Iterative Palladium-Catalyzed CH Arylation and Halogen Exchange
Masuda, Naoyuki, Tanba, Shunsuke, Sugie, Atsushi, Monguchi, Daiki, Koumura, Nagatoshi, Hara, Kohjiro, Mori, Atsunori
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
Get full text
Journal Article
Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436
Hamaguchi, Wataru, Masuda, Naoyuki, Miyamoto, Satoshi, Kikuchi, Shigetoshi, Narazaki, Fumie, Shiina, Yasuhiro, Seo, Ryushi, Amano, Yasushi, Mihara, Takuma, Moriguchi, Hiroyuki, Hattori, Kouji
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
Get full text
Journal Article
Dinuclear Copper(II) 3,4,5-Tri-O-benzylgallate
Mikuriya, Masahiro, Yamakawa, Chihiro, Masuda, Naoyuki, Yoshioka, Daisuke, Yamaguchi, Sayuri, Yamada, Hidetoshi, Mizuta, Tsutomu, Kawata, Naomi, Tanaka, Hidekazu, Handa, Makoto
Published in Open Chemistry Journal (22.03.2019)
Published in Open Chemistry Journal (22.03.2019)
Get full text
Journal Article
Potent and orally bioavailable CCR4 antagonists: Synthesis and structure–activity relationship study of 2-aminoquinazolines
Yokoyama, Kazuhiro, Ishikawa, Noriko, Igarashi, Susumu, Kawano, Noriyuki, Masuda, Naoyuki, Hamaguchi, Wataru, Yamasaki, Shingo, Koganemaru, Yohei, Hattori, Kazuyuki, Miyazaki, Takahiro, Ogino, Shin-ichi, Matsumoto, Yuzo, Takeuchi, Makoto, Ohta, Mitsuaki
Published in Bioorganic & medicinal chemistry (2009)
Published in Bioorganic & medicinal chemistry (2009)
Get full text
Journal Article
ITERATIVE EXTENSION OF THIOPHENE RING LEADING TO HEAD-TO-TAIL-TYPE OLIGOTHIOPHENES VIA STEPWISE CH ARYLATION AND HALOGEN EXCHANGE SEQUENCE
Tanba, Shunsuke, Sugie, Atsushi, Masuda, Naoyuki, Monguchi, Daiki, Koumura, Nagatoshi, Hara, Kohjiro, Mori, Atsunori
Published in Heterocycles (31.12.2010)
Published in Heterocycles (31.12.2010)
Get more information
Journal Article
KDR-5169, a new gastrointestinal prokinetic agent, enhances gastric contractile and emptying activities in dogs and rats
Tazawa, Shigeki, Masuda, Naoyuki, Koizumi, Takashi, Kitazawa, Makio, Nakane, Tokio, Miyata, Hiroshi
Published in European journal of pharmacology (11.01.2002)
Published in European journal of pharmacology (11.01.2002)
Get full text
Journal Article
Binding Modes of Two Novel Non-Nucleoside Reverse Transcriptase Inhibitors, YM-215389 and YM-228855, to HIV Type-1 Reverse Transcriptase
Kodama, Eiichi, Orita, Masaya, Masuda, Naoyuki, Yamamoto, Osamu, Fujii, Masahiro, Ohgami, Tetsuro, Kageyama, Shunji, Ohta, Mitsuaki, Hatta, Toshifumi, Inoue, Hiroshi, Suzuki, Hiroshi, Sudo, Kenji, Shimizu, Yasuaki, Matsuoka, Masao
Published in Antiviral chemistry & chemotherapy (01.06.2008)
Published in Antiviral chemistry & chemotherapy (01.06.2008)
Get full text
Journal Article
Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability
Chino, Ayaka, Masuda, Naoyuki, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Yamazaki, Mayako, Tomishima, Masaki
Published in Bioorganic & medicinal chemistry (01.07.2014)
Published in Bioorganic & medicinal chemistry (01.07.2014)
Get full text
Journal Article
Synthesis, SAR study, and biological evaluation of novel 2,3-dihydro-1H-imidazo[1,2-a]benzimidazole derivatives as phosphodiesterase 10A inhibitors
Chino, Ayaka, Honda, Shugo, Morita, Masataka, Yonezawa, Koichi, Hamaguchi, Wataru, Amano, Yasushi, Moriguchi, Hiroyuki, Yamazaki, Mayako, Aota, Masaki, Tomishima, Masaki, Masuda, Naoyuki
Published in Bioorganic & medicinal chemistry (15.08.2019)
Published in Bioorganic & medicinal chemistry (15.08.2019)
Get full text
Journal Article
Design and synthesis of novel benzimidazole derivatives as phosphodiesterase 10A inhibitors with reduced CYP1A2 inhibition
Hamaguchi, Wataru, Masuda, Naoyuki, Isomura, Mai, Miyamoto, Satoshi, Kikuchi, Shigetoshi, Amano, Yasushi, Honbou, Kazuya, Mihara, Takuma, Watanabe, Toshihiro
Published in Bioorganic & medicinal chemistry (15.12.2013)
Published in Bioorganic & medicinal chemistry (15.12.2013)
Get full text
Journal Article
Synthesis, SAR study, and biological evaluation of novel quinoline derivatives as phosphodiesterase 10A inhibitors with reduced CYP3A4 inhibition
Hamaguchi, Wataru, Masuda, Naoyuki, Miyamoto, Satoshi, Shiina, Yasuhiro, Kikuchi, Shigetoshi, Mihara, Takuma, Moriguchi, Hiroyuki, Fushiki, Hiroshi, Murakami, Yoshihiro, Amano, Yasushi, Honbou, Kazuya, Hattori, Kouji
Published in Bioorganic & medicinal chemistry (15.01.2015)
Published in Bioorganic & medicinal chemistry (15.01.2015)
Get full text
Journal Article
Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors
Ayaka Chino, Ryushi Seo, Yasushi Amano, Ichiji Namatame, Wataru Hamaguchi, Kazuya Honbou, Takuma Mihara, Mayako Yamazaki, Masaki Tomishima, Naoyuki Masuda
Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
Get full text
Published in Chemical and Pharmaceutical Bulletin (01.03.2018)
Journal Article
Mononuclear cobalt (III) complexes with N-salicylidene-2-hydroxy-5-bromobenzylamine and N-salicylidene-2-hydroxy-5-chlorobenzylamine
Mikuriya, Masahiro, Masuda, Naoyuki, Kakuta, Yoshihisa, Minato, Shinya, Inui, Takaya, Yoshioka, Daisuke
Published in Chemical papers (2016)
Published in Chemical papers (2016)
Get full text
Journal Article