Synthesis and Evaluation of in Vivo Anti-hypothermic Effect of the N- and C-Terminus Modified Thyrotropin-Releasing Hormone Mimetic: [(4S,5S)-(5-Methyl-2-oxooxazolidine-4-yl)carbonyl]-[3-(thiazol-4-yl)-L-alanyl]-L-prolinamide
Kobayashi, Naotake, Sato, Norihito, Sugita, Katsuji, Kihara, Tsuyoshi, Koike, Katsumi, Sugawara, Tamio, Tada, Yukio, Yoshikawa, Takayoshi
Published in Chemical & pharmaceutical bulletin (01.04.2021)
Published in Chemical & pharmaceutical bulletin (01.04.2021)
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Synthesis and evaluation of in vivo anti‐hypothermic effect of all stereoisomers of the thyrotropin‐releasing hormone mimetic: Rovatirelin Hydrate
Kobayashi, Naotake, Sato, Norihito, Sugita, Katsuji, Takahashi, Kouji, Sugawara, Tamio, Tada, Yukio, Yoshikawa, Takayoshi
Published in Journal of peptide science (01.12.2019)
Published in Journal of peptide science (01.12.2019)
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Journal Article
Discovery of the Orally Effective Thyrotropin-Releasing Hormone Mimetic: 1‑{N‑[(4S,5S)‑(5-Methyl-2-oxooxazolidine-4-yl)carbonyl]-3-(thiazol-4-yl)‑l‑alanyl}-(2R)‑2-methylpyrrolidine Trihydrate (Rovatirelin Hydrate)
Kobayashi, Naotake, Sato, Norihito, Fujimura, Yuko, Kihara, Tsuyoshi, Sugita, Katsuji, Takahashi, Kouji, Koike, Katsumi, Sugawara, Tamio, Tada, Yukio, Nakai, Hiroshi, Yoshikawa, Takayoshi
Published in ACS omega (31.10.2018)
Published in ACS omega (31.10.2018)
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Journal Article
Correction to Discovery of the Orally Effective Thyrotropin-Releasing Hormone Mimetic: 1‑{N‑[(4S,5S)‑(5-Methyl-2-oxooxazolidine-4-yl)carbonyl]-3-(thiazol-4-yl)‑l‑alanyl}-(2R)‑2-methylpyrrolidine Trihydrate (Rovatirelin Hydrate)
Kobayashi, Naotake, Sato, Norihito, Fujimura, Yuko, Kihara, Tsuyoshi, Sugita, Katsuji, Takahashi, Kouji, Koike, Katsumi, Sugawara, Tamio, Tada, Yukio, Nakai, Hiroshi, Yoshikawa, Takayoshi
Published in ACS omega (30.04.2019)
Published in ACS omega (30.04.2019)
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Discovery of a novel olefin derivative as a highly potent and selective acetyl-CoA carboxylase 2 inhibitor with in vivo efficacy
Nishiura, Yuji, Matsumura, Akira, Kobayashi, Naotake, Shimazaki, Atsuyuki, Sakamoto, Shingo, Kitade, Naohisa, Tonomura, Yutaka, Ino, Akira, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
Published in Bioorganic & medicinal chemistry letters (01.08.2018)
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Pyrrolinone derivatives as a new class of P2X3 receptor antagonists. Part 1: Initial structure-activity relationship studies of a hit from a high throughput screening
Tobinaga, Hiroyuki, Kameyama, Takayuki, Oohara, Miho, Kobayashi, Naotake, Ohdan, Masahide, Ishizuka, Natsuki, Kume, Masaharu, Tomari, Maki, Tanaka, Yoshikazu, Takahashi, Fumiyo, Kinoshita, Haruki, Shimada, Shinji, Shinohara, Shunji, Kai, Hiroyuki
Published in Bioorganic & medicinal chemistry letters (15.07.2018)
Published in Bioorganic & medicinal chemistry letters (15.07.2018)
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ACC2 INHIBITORS
OHYABU, Naoki, MIYAZAKI, Keisuke, KATOU, Manabu, TOMIDA, Yutaka, OHDAN, Masahide, IWATSU, Masafumi, ASAHI, Kentarou, KURAHASHI, Kana, WADA, Toshihiro, INOUE, Takatsugu, FUMOTO, Masataka, SASAKI, Yoshikazu, URABE, Tomomi, KOBAYASHI, Naotake, NISHIURA, Yuji
Year of Publication 30.09.2020
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Year of Publication 30.09.2020
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