Search Results - "Nagasree Chakka" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

Discovery of Novel, Induced-Pocket Binding Oxazolidinones as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

by Bregman, Howard, Chakka, Nagasree, Guzman-Perez, Angel, Gunaydin, Hakan, Gu, Yan, Huang, Xin, Berry, Virginia, Liu, Jingzhou, Teffera, Yohannes, Huang, Liyue, Egge, Bryan, Mullady, Erin L, Schneider, Steve, Andrews, Paul S, Mishra, Ankita, Newcomb, John, Serafino, Randy, Strathdee, Craig A, Turci, Susan M, Wilson, Cindy, DiMauro, Erin F
Published in Journal of medicinal chemistry (13.06.2013)

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Journal Article

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors

by DiMauro, Erin F, Altmann, Stephen, Berry, Loren M, Bregman, Howard, Chakka, Nagasree, Chu-Moyer, Margaret, Bojic, Elma Feric, Foti, Robert S, Fremeau, Robert, Gao, Hua, Gunaydin, Hakan, Guzman-Perez, Angel, Hall, Brian E, Huang, Hongbing, Jarosh, Michael, Kornecook, Thomas, Lee, Josie, Ligutti, Joseph, Liu, Dong, Moyer, Bryan D, Ortuno, Daniel, Rose, Paul E, Schenkel, Laurie B, Taborn, Kristin, Wang, Jean, Wang, Yan, Yu, Violeta, Weiss, Matthew M
Published in Journal of medicinal chemistry (08.09.2016)

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Journal Article

Discovery of a biarylamide series of potent, state-dependent NaV1.7 inhibitors

Discovery of a biarylamide series of potent, state-dependent NaV1.7 inhibitors

by Schenkel, Laurie B., DiMauro, Erin F., Nguyen, Hanh N., Chakka, Nagasree, Du, Bingfan, Foti, Robert S., Guzman-Perez, Angel, Jarosh, Michael, La, Daniel S., Ligutti, Joseph, Milgram, Benjamin C., Moyer, Bryan D., Peterson, Emily A., Roberts, John, Yu, Violeta L., Weiss, Matthew M.
Published in Bioorganic & medicinal chemistry letters (15.08.2017)

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Journal Article

Discovery of benzylisothioureas as potent divalent metal transporter 1 (DMT1) inhibitors

Discovery of benzylisothioureas as potent divalent metal transporter 1 (DMT1) inhibitors

by Zhang, Zaihui, Kodumuru, Vishnumurthy, Sviridov, Serguei, Liu, Shifeng, Chafeev, Mikhail, Chowdhury, Sultan, Chakka, Nagasree, Sun, Jianyu, Gauthier, Simon J., Mattice, Maryanne, Ratkay, Laszlo G., Kwan, Rainbow, Thompson, Jay, Cutts, Alison Brownlie, Fu, Jianmin, Kamboj, Rajender, Goldberg, Y. Paul, Cadieux, Jay A.
Published in Bioorganic & medicinal chemistry letters (01.08.2012)

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Journal Article

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na(V)1.7 Inhibitors

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na(V)1.7 Inhibitors

by DiMauro, Erin F., Altmann, Stephen, Berry, Loren M., Bregman, Howard, Chakka, Nagasree, Chu-Moyer, Margaret, Bojic, Elma Feric, Foti, Robert S., Fremeau, Robert, Gao, Hua, Gunaydin, Hakan, Guzman-Perez, Angel, Hall, Brian E., Huang, Hongbing, Jarosh, Michael, Korneook, Thomas, Lee, Josie, Ligutti, Joseph, Liu, Dong, Moyer, Bryan D., Ortuno, Daniel, Rose, Paul E., Schenkel, Laurie B., Taborn, Kristin, Wang, Jean, Wang, Yan, Yu, Violeta, Weiss, Matthew M.
Published in Journal of medicinal chemistry (08.09.2016)

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Journal Article

Applications of parallel synthetic lead hopping and pharmacophore-based virtual screening in the discovery of efficient glycine receptor potentiators

Applications of parallel synthetic lead hopping and pharmacophore-based virtual screening in the discovery of efficient glycine receptor potentiators

by Chakka, Nagasree, Andrews, Kristin L., Berry, Loren M., Bregman, Howard, Gunaydin, Hakan, Huang, Liyue, Guzman-Perez, Angel, Plant, Matthew H., Simard, Jeffrey R., Gingras, Jacinthe, DiMauro, Erin F.
Published in European journal of medicinal chemistry (08.09.2017)

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Journal Article

Discovery of a biarylamide series of potent, state-dependent Na(V)1.7 inhibitors

Discovery of a biarylamide series of potent, state-dependent Na(V)1.7 inhibitors

by Schenkel, Laurie B., DiMauro, Erin F., Nguyen, Hanh N., Chakka, Nagasree, Du, Bingfan, Foti, Robert S., Guzman-Perez, Angel, Jarosh, Michael, La, Daniel S., Ligutti, Joseph, Milgram, Benjamin C., Moyer, Bryan D., Peterson, Emily A., Roberts, John, Yu, Violeta L., Weiss, Matthew M.
Published in Bioorganic & medicinal chemistry letters (15.08.2017)

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Journal Article

Discovery of Piperazin-1-ylpyridazine-Based Potent and Selective Stearoyl-CoA Desaturase‑1 Inhibitors for the Treatment of Obesity and Metabolic Syndrome

Discovery of Piperazin-1-ylpyridazine-Based Potent and Selective Stearoyl-CoA Desaturase‑1 Inhibitors for the Treatment of Obesity and Metabolic Syndrome

by Zhang, Zaihui, Sun, Shaoyi, Kodumuru, Vishnumurthy, Hou, Duanjie, Liu, Shifeng, Chakka, Nagasree, Sviridov, Serguei, Chowdhury, Sultan, McLaren, David G, Ratkay, Leslie G, Khakh, Kuldip, Cheng, Xing, Gschwend, Heinz W, Kamboj, Rajender, Fu, Jianmin, Winther, Michael D
Published in Journal of medicinal chemistry (24.01.2013)

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Journal Article

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na V 1.7 Inhibitors

Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective Na V 1.7 Inhibitors

by DiMauro, Erin F., Altmann, Stephen, Berry, Loren M., Bregman, Howard, Chakka, Nagasree, Chu-Moyer, Margaret, Bojic, Elma Feric, Foti, Robert S., Fremeau, Robert, Gao, Hua, Gunaydin, Hakan, Guzman-Perez, Angel, Hall, Brian E., Huang, Hongbing, Jarosh, Michael, Kornecook, Thomas, Lee, Josie, Ligutti, Joseph, Liu, Dong, Moyer, Bryan D., Ortuno, Daniel, Rose, Paul E., Schenkel, Laurie B., Taborn, Kristin, Wang, Jean, Wang, Yan, Yu, Violeta, Weiss, Matthew M.
Published in Journal of medicinal chemistry (08.09.2016)

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Journal Article

Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Na(v)1.7 antagonists

Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Na(v)1.7 antagonists

by Chakka, Nagasree, Bregman, Howie, Du, Bingfan, Nguyen, Hanh Nho, Buchanan, John L, Feric, Elma, Ligutti, Joseph, Liu, Dong, McDermott, Jeff S, Zou, Anruo, McDonough, Stefan I, Dimauro, Erin F
Published in Bioorganic & medicinal chemistry letters (01.03.2012)

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Journal Article

Abstract 1621: Discovery of pyridyl pyrrolopyridinones as potent and selective CK1γ inhibitors

Abstract 1621: Discovery of pyridyl pyrrolopyridinones as potent and selective CK1γ inhibitors

by Huang, Hongbing, Acquaviva, Lisa, Bregman, Howard, Buchanan, John, Chakka, Nagasree, DiMauro, Erin F., Dovey, Jennifer, Gunaydin, Hakan, Hua, Zihao, Huang, Xin, Huang, Liyue, Patel, Vinod F., Martin, Matthew W., Serafino, Randy, Wilson, Cindy
Published in Cancer research (Chicago, Ill.) (01.10.2014)

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Journal Article

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

by Hua, Zihao, Huang, Xin, Bregman, Howard, Chakka, Nagasree, DiMauro, Erin F., Doherty, Elizabeth M., Goldstein, Jon, Gunaydin, Hakan, Huang, Hongbing, Mercede, Stephanie, Newcomb, John, Patel, Vinod F., Turci, Susan M., Yan, Jie, Wilson, Cindy, Martin, Matthew W.
Published in Bioorganic & medicinal chemistry letters (01.09.2012)

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Journal Article

Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

by Hua, Zihao, Bregman, Howard, Buchanan, John L, Chakka, Nagasree, Guzman-Perez, Angel, Gunaydin, Hakan, Huang, Xin, Gu, Yan, Berry, Virginia, Liu, Jingzhou, Teffera, Yohannes, Huang, Liyue, Egge, Bryan, Emkey, Renee, Mullady, Erin L, Schneider, Steve, Andrews, Paul S, Acquaviva, Lisa, Dovey, Jennifer, Mishra, Ankita, Newcomb, John, Saffran, Douglas, Serafino, Randy, Strathdee, Craig A, Turci, Susan M, Stanton, Mary, Wilson, Cindy, DiMauro, Erin F
Published in Journal of medicinal chemistry (27.12.2013)

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Journal Article

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

2-Phenylamino-6-cyano-1H-benzimidazole-based isoform selective casein kinase 1 gamma (CK1γ) inhibitors

by Hua, Zihao, Huang, Xin, Bregman, Howard, Chakka, Nagasree, DiMauro, Erin F., Doherty, Elizabeth M., Goldstein, Jon, Gunaydin, Hakan, Huang, Hongbing, Mercede, Stephanie, Newcomb, John, Patel, Vinod F., Turci, Susan M., Yan, Jie, Wilson, Cindy, Martin, Matthew W.
Published in Bioorganic & medicinal chemistry letters (01.09.2012)

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Journal Article

Structure-Based Design of Potent and Selective CK1γ Inhibitors

Structure-Based Design of Potent and Selective CK1γ Inhibitors

by Huang, Hongbing, Acquaviva, Lisa, Berry, Virginia, Bregman, Howard, Chakka, Nagasree, O’Connor, Anne, DiMauro, Erin F, Dovey, Jennifer, Epstein, Oleg, Grubinska, Barbara, Goldstein, Jon, Gunaydin, Hakan, Hua, Zihao, Huang, Xin, Huang, Liyue, Human, Jason, Long, Alex, Newcomb, John, Patel, Vinod F, Saffran, Doug, Serafino, Randy, Schneider, Steve, Strathdee, Craig, Tang, Jin, Turci, Susan, White, Ryan, Yu, Violeta, Zhao, Huilin, Wilson, Cindy, Martin, Matthew W
Published in ACS medicinal chemistry letters (13.12.2012)

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Journal Article

Discovery of a biarylamide series of potent, state-dependent Na V 1.7 inhibitors

Discovery of a biarylamide series of potent, state-dependent Na V 1.7 inhibitors

by Schenkel, Laurie B, DiMauro, Erin F, Nguyen, Hanh N, Chakka, Nagasree, Du, Bingfan, Foti, Robert S, Guzman-Perez, Angel, Jarosh, Michael, La, Daniel S, Ligutti, Joseph, Milgram, Benjamin C, Moyer, Bryan D, Peterson, Emily A, Roberts, John, Yu, Violeta L, Weiss, Matthew M
Published in Bioorganic & medicinal chemistry letters (15.08.2017)

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Journal Article

Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Nav1.7 antagonists

Discovery and hit-to-lead optimization of pyrrolopyrimidines as potent, state-dependent Nav1.7 antagonists

by Chakka, Nagasree, Bregman, Howie, Du, Bingfan, Nguyen, Hanh Nho, Buchanan, John L., Feric, Elma, Ligutti, Joseph, Liu, Dong, McDermott, Jeff S., Zou, Anruo, McDonough, Stefan I., DiMauro, Erin F.
Published in Bioorganic & medicinal chemistry letters (01.03.2012)

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Journal Article

Synthesis and conformational analysis of disaccharide analogues containing disulfide and selenosulfide functionalities in the interglycosidic linkages1

Synthesis and conformational analysis of disaccharide analogues containing disulfide and selenosulfide functionalities in the interglycosidic linkages1

by Chakka, Nagasree, Johnston, Blair D, Pinto, B Mario
Published in Canadian journal of chemistry (01.06.2005)

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Journal Article

Synthesis and conformational analysis of disaccharide analogues containing disulfide and selenosulfide functionalities in the interglycosidic linkages

Synthesis and conformational analysis of disaccharide analogues containing disulfide and selenosulfide functionalities in the interglycosidic linkages

by Chakka, Nagasree, Johnston, Blair D, Pinto, B Mario
Published in Canadian journal of chemistry (01.06.2005)

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Journal Article

BENZIMIDAZOLE DERIVATIVES AND THEIR USES

BENZIMIDAZOLE DERIVATIVES AND THEIR USES

by SCHENKEL, LAURIE, GAO, HUA, MALINOWSKI, JUSTIN, CHAKKA, NAGASREE, KIEFFER, MADELEINE, GUZMAN-PEREZ, ANGEL, JOHNSON, BRETT MICHAEL
Year of Publication 21.11.2023

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