Search Results - "Nacci, V" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Specific Targeting Highly Conserved Residues in the HIV-1 Reverse Transcriptase Primer Grip Region. Design, Synthesis, and Biological Evaluation of Novel, Potent, and Broad Spectrum NNRTIs with Antiviral Activity

Specific Targeting Highly Conserved Residues in the HIV-1 Reverse Transcriptase Primer Grip Region. Design, Synthesis, and Biological Evaluation of Novel, Potent, and Broad Spectrum NNRTIs with Antiviral Activity

by Fattorusso, Caterina, Gemma, Sandra, Butini, Stefania, Huleatt, Paul, Catalanotti, Bruno, Persico, Marco, De Angelis, Meri, Fiorini, Isabella, Nacci, Vito, Ramunno, Anna, Rodriquez, Manuela, Greco, Giovanni, Novellino, Ettore, Bergamini, Alberto, Marini, Stefano, Coletta, Massimo, Maga, Giovanni, Spadari, Silvio, Campiani, Giuseppe
Published in Journal of medicinal chemistry (17.11.2005)

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Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

by Campiani, Giuseppe, Aiello, Francesca, Fabbrini, Monica, Morelli, Elena, Ramunno, Anna, Armaroli, Silvia, Nacci, Vito, Garofalo, Antonio, Greco, Giovanni, Novellino, Ettore, Maga, Giovanni, Spadari, Silvio, Bergamini, Alberto, Ventura, Laura, Bongiovanni, Barbara, Capozzi, Marcella, Bolacchi, Francesca, Marini, Stefano, Coletta, Massimiliano, Guiso, Giovanna, Caccia, Silvio
Published in Journal of medicinal chemistry (01.02.2001)

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A Rational Approach to the Design of Selective Substrates and Potent Nontransportable Inhibitors of the Excitatory Amino Acid Transporter EAAC1 (EAAT3). New Glutamate and Aspartate Analogues as Potential Neuroprotective Agents

A Rational Approach to the Design of Selective Substrates and Potent Nontransportable Inhibitors of the Excitatory Amino Acid Transporter EAAC1 (EAAT3). New Glutamate and Aspartate Analogues as Potential Neuroprotective Agents

by Campiani, Giuseppe, De Angelis, Meri, Armaroli, Silvia, Fattorusso, Caterina, Catalanotti, Bruno, Ramunno, Anna, Nacci, Vito, Novellino, Ettore, Grewer, Christof, Ionescu, Diana, Rauen, Thomas, Griffiths, Roger, Sinclair, Colin, Fumagalli, Elena, Mennini, Tiziana
Published in Journal of medicinal chemistry (02.08.2001)

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Characterization of the 1H-Cyclopentapyrimidine-2,4(1H,3H)-dione Derivative (S)-CPW399 as a Novel, Potent, and Subtype-Selective AMPA Receptor Full Agonist with Partial Desensitization Properties

Characterization of the 1H-Cyclopentapyrimidine-2,4(1H,3H)-dione Derivative (S)-CPW399 as a Novel, Potent, and Subtype-Selective AMPA Receptor Full Agonist with Partial Desensitization Properties

by Campiani, Giuseppe, Morelli, Elena, Nacci, Vito, Fattorusso, Caterina, Ramunno, Anna, Novellino, Ettore, Greenwood, Jeremy, Liljefors, Tommy, Griffiths, Roger, Sinclair, Colin, Reavy, Helen, Kristensen, Anders S, Pickering, Darryl S, Schousboe, Arne, Cagnotto, Alfredo, Fumagalli, Elena, Mennini, Tiziana
Published in Journal of medicinal chemistry (20.12.2001)

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Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agents

Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agents

by Zisterer, D M, McGee, M M, Campiani, G, Ramunno, A, Fattorusso, C, Nacci, V, Lawler, M, Williams, D C
Published in Biochemical Society transactions (01.11.2001)

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New pyrrolobenzothiazepine derivatives as molecular probes of the ‘peripheral-type’ benzodiazepine receptor (PBR) binding site

New pyrrolobenzothiazepine derivatives as molecular probes of the ‘peripheral-type’ benzodiazepine receptor (PBR) binding site

by Campiani, G, Nacci, V, Fiorini, I, De Filippis, MP, Garofalo, A, Ciani, SM, Greco, G, Novellino, E, Manzoni, C, Mennini, T
Published in European journal of medicinal chemistry (1997)

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Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis and Biological Evaluation of Novel Quinoxalinylethylpyridylthioureas as Potent Antiviral Agents

Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis and Biological Evaluation of Novel Quinoxalinylethylpyridylthioureas as Potent Antiviral Agents

by Campiani, G, Fabbrini, M, Morelli, E, Nacci, V, Greco, G, Novellino, E, Maga, G, Spadari, S, Bergamini, A, Faggioli, E, Uccella, I, Bolacchi, F, Marini, S, Coletta, M, Fracasso, C, Caccia, S
Published in Antiviral chemistry & chemotherapy (01.03.2000)

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Thioanalogues of anti-tumor antibiotics. II. Synthesis and preliminary in vitro cytotoxicity evaluation of tricyclic [1,4]benzothiazepine derivatives

Thioanalogues of anti-tumor antibiotics. II. Synthesis and preliminary in vitro cytotoxicity evaluation of tricyclic [1,4]benzothiazepine derivatives

by Garofalo, A, Balconi, G, Botta, M, Corelli, F, D'Incalci, M, Fabrizi, G, Fiorini, I, Lamba, D, Nacci, V
Published in European journal of medicinal chemistry (1993)

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Synthesis and “in vitro” cardiovascular activity of 4-aryl-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,4]benzothiazin-1-ones and 7-acetoxy-6-phenyl-7a,8,9,10-tetrahydropyrrolo [2,1,-d][1,5]benzothiazepin-10-one

Synthesis and “in vitro” cardiovascular activity of 4-aryl-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,4]benzothiazin-1-ones and 7-acetoxy-6-phenyl-7a,8,9,10-tetrahydropyrrolo [2,1,-d][1,5]benzothiazepin-10-one

by Campiani, G., Garofalo, A., Fiorini, I., Nacci, V., Botta, M., Tafi, A., Chiarini, A., Budriesi, R., Bruni, G., Romeo, M.R.
Published in Bioorganic & medicinal chemistry letters (19.05.1994)

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Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors: Past, Present, and Future Perspectives

Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors: Past, Present, and Future Perspectives

by Campiani, Giuseppe, Ramunno, Anna, Maga, Giovanni, Nacci, Vito, Fattorusso, Caterina, Catalanotti, Bruno, Morelli, Elena, Novellino, Ettore
Published in Current pharmaceutical design (01.01.2002)

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Specific Targeting of Hepatitis C Virus NS3 RNA Helicase. Discovery of the Potent and Selective Competitive Nucleotide-Mimicking Inhibitor QU663

Specific Targeting of Hepatitis C Virus NS3 RNA Helicase. Discovery of the Potent and Selective Competitive Nucleotide-Mimicking Inhibitor QU663

by Maga, Giovanni, Gemma, Sandra, Fattorusso, Caterina, Locatelli, Giada A, Butini, Stefania, Persico, Marco, Kukreja, Gagan, Romano, Maria Pia, Chiasserini, Luisa, Savini, Luisa, Novellino, Ettore, Nacci, Vito, Spadari, Silvio, Campiani, Giuseppe
Published in Biochemistry (Easton) (19.07.2005)

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Development of Molecular Probes for the Identification of Extra Interaction Sites in the Mid-Gorge and Peripheral Sites of Butyrylcholinesterase (BuChE). Rational Design of Novel, Selective, and Highly Potent BuChE Inhibitors

Development of Molecular Probes for the Identification of Extra Interaction Sites in the Mid-Gorge and Peripheral Sites of Butyrylcholinesterase (BuChE). Rational Design of Novel, Selective, and Highly Potent BuChE Inhibitors

by Campiani, Giuseppe, Fattorusso, Caterina, Butini, Stefania, Gaeta, Alessandra, Agnusdei, Marianna, Gemma, Sandra, Persico, Marco, Catalanotti, Bruno, Savini, Luisa, Nacci, Vito, Novellino, Ettore, Holloway, Harold W, Greig, Nigel H, Belinskaya, Tatyana, Fedorko, James M, Saxena, Ashima
Published in Journal of medicinal chemistry (24.03.2005)

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Caspase-3 is not essential for DNA fragmentation in MCF-7 cells during apoptosis induced by the pyrrolo-1,5-benzoxazepine, PBOX-6

Caspase-3 is not essential for DNA fragmentation in MCF-7 cells during apoptosis induced by the pyrrolo-1,5-benzoxazepine, PBOX-6

by Mc Gee, Margaret M, Hyland, Edel, Campiani, Giuseppe, Ramunno, Anna, Nacci, Vito, Zisterer, Daniela M
Published in FEBS letters (27.03.2002)

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Research on compounds with psychotropic activity. IX--Synthesis of 6-p-methoxyphenylpyrrolo[2,1-d][1,5]benzothiazepines and evaluation of their affinities for BDZ and GABA receptor subtypes

Research on compounds with psychotropic activity. IX--Synthesis of 6-p-methoxyphenylpyrrolo[2,1-d][1,5]benzothiazepines and evaluation of their affinities for BDZ and GABA receptor subtypes

by Nacci, V, Fiorini, I, Garofalo, A, Cagnotto, A
Published in Farmaco (Società chimica italiana : 1989) (01.05.1990)

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Novel Atypical Antipsychotic Agents: Rational Design, an Efficient Palladium-Catalyzed Route, and Pharmacological Studies

Novel Atypical Antipsychotic Agents: Rational Design, an Efficient Palladium-Catalyzed Route, and Pharmacological Studies

by Campiani, Giuseppe, Butini, Stefania, Fattorusso, Caterina, Trotta, Francesco, Gemma, Sandra, Catalanotti, Bruno, Nacci, Vito, Fiorini, Isabella, Cagnotto, Alfredo, Mereghetti, Ilario, Mennini, Tiziana, Minetti, Patrizia, Di Cesare, M. Assunta, Stasi, M. Antonietta, Di Serio, Stefano, Ghirardi, Orlando, Tinti, Ornella, Carminati, Paolo
Published in Journal of medicinal chemistry (24.03.2005)

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Pyrroloquinoxaline Derivatives as High-Affinity and Selective 5-HT3 Receptor Agonists: Synthesis, Further Structure−Activity Relationships, and Biological Studies

Pyrroloquinoxaline Derivatives as High-Affinity and Selective 5-HT3 Receptor Agonists: Synthesis, Further Structure−Activity Relationships, and Biological Studies

by Campiani, Giuseppe, Morelli, Elena, Gemma, Sandra, Nacci, Vito, Butini, Stefania, Hamon, Michel, Novellino, Ettore, Greco, Giovanni, Cagnotto, Alfredo, Goegan, Mara, Cervo, Luigi, Dalla Valle, Fabio, Fracasso, Claudia, Caccia, Silvio, Mennini, Tiziana
Published in Journal of medicinal chemistry (21.10.1999)

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Neuronal High-Affinity Sodium-Dependent Glutamate Transporters (EAATs): Targets for the Development of Novel Therapeutics Against Neurodegenerative Diseases

Neuronal High-Affinity Sodium-Dependent Glutamate Transporters (EAATs): Targets for the Development of Novel Therapeutics Against Neurodegenerative Diseases

by Campiani, Giuseppe, Fattorusso, Caterina, De Angelis, Meri, Catalanotti, Bruno, Butini, Stefania, Fattorusso, Roberto, Fiorini, Isabella, Nacci, Vito, Novellino, Ettore
Published in Current pharmaceutical design (01.01.2003)

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Erosion of cohesive sediments as a rate process

Erosion of cohesive sediments as a rate process

by Gularte, R.C., Kelly, W.E., Nacci, V.A.
Published in Ocean engineering (1980)

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Thiazolothiazepine Inhibitors of HIV-1 Integrase

Thiazolothiazepine Inhibitors of HIV-1 Integrase

by Neamati, Nouri, Turpin, Jim A, Winslow, Heather E, Christensen, John L, Williamson, Karen, Orr, Ann, Rice, William G, Pommier, Yves, Garofalo, Antonio, Brizzi, Antonella, Campiani, Giuseppe, Fiorini, Isabella, Nacci, Vito
Published in Journal of medicinal chemistry (26.08.1999)

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Activation of the c-Jun N-terminal Kinase (JNK) Signaling Pathway Is Essential during PBOX-6-induced Apoptosis in Chronic Myelogenous Leukemia (CML) Cells

Activation of the c-Jun N-terminal Kinase (JNK) Signaling Pathway Is Essential during PBOX-6-induced Apoptosis in Chronic Myelogenous Leukemia (CML) Cells

by Mc Gee, Margaret M., Campiani, Giuseppe, Ramunno, Anna, Nacci, Vito, Lawler, Mark, Williams, D. Clive, Zisterer, Daniela M.
Published in The Journal of biological chemistry (24.05.2002)

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