Cryptic glucocorticoid receptor-binding sites pervade genomic NF-κB response elements
Hudson, William H, Vera, Ian Mitchelle S de, Nwachukwu, Jerome C, Weikum, Emily R, Herbst, Austin G, Yang, Qin, Bain, David L, Nettles, Kendall W, Kojetin, Douglas J, Ortlund, Eric A
Published in Nature communications (06.04.2018)
Published in Nature communications (06.04.2018)
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Journal Article
Structural and Molecular Mechanisms of Cytokine-Mediated Endocrine Resistance in Human Breast Cancer Cells
Stender, Joshua D., Nwachukwu, Jerome C., Kastrati, Irida, Kim, Yohan, Strid, Tobias, Yakir, Maayan, Srinivasan, Sathish, Nowak, Jason, Izard, Tina, Rangarajan, Erumbi S., Carlson, Kathryn E., Katzenellenbogen, John A., Yao, Xin-Qiu, Grant, Barry J., Leong, Hon S., Lin, Chin-Yo, Frasor, Jonna, Nettles, Kendall W., Glass, Christopher K.
Published in Molecular cell (16.03.2017)
Published in Molecular cell (16.03.2017)
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Journal Article
Structural mechanism for signal transduction in RXR nuclear receptor heterodimers
Kojetin, Douglas J, Matta-Camacho, Edna, Hughes, Travis S, Srinivasan, Sathish, Nwachukwu, Jerome C, Cavett, Valerie, Nowak, Jason, Chalmers, Michael J, Marciano, David P, Kamenecka, Theodore M, Shulman, Andrew I, Rance, Mark, Griffin, Patrick R, Bruning, John B, Nettles, Kendall W
Published in Nature communications (20.08.2015)
Published in Nature communications (20.08.2015)
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Journal Article
Dual suppression of estrogenic and inflammatory activities for targeting of endometriosis
Zhao, Yuechao, Gong, Ping, Chen, Yiru, Nwachukwu, Jerome C, Srinivasan, Sathish, Ko, CheMyong, Bagchi, Milan K, Taylor, Robert N, Korach, Kenneth S, Nettles, Kendall W, Katzenellenbogen, John A, Katzenellenbogen, Benita S
Published in Science translational medicine (21.01.2015)
Published in Science translational medicine (21.01.2015)
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Journal Article
Full antagonism of the estrogen receptor without a prototypical ligand side chain
Srinivasan, Sathish, Nwachukwu, Jerome C, Bruno, Nelson E, Dharmarajan, Venkatasubramanian, Goswami, Devrishi, Kastrati, Irida, Novick, Scott, Nowak, Jason, Cavett, Valerie, Zhou, Hai-Bing, Boonmuen, Nittaya, Zhao, Yuechao, Min, Jian, Frasor, Jonna, Katzenellenbogen, Benita S, Griffin, Patrick R, Katzenellenbogen, John A, Nettles, Kendall W
Published in Nature chemical biology (01.01.2017)
Published in Nature chemical biology (01.01.2017)
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Journal Article
Resveratrol modulates the inflammatory response via an estrogen receptor-signal integration network
Nwachukwu, Jerome C, Srinivasan, Sathish, Bruno, Nelson E, Parent, Alexander A, Hughes, Travis S, Pollock, Julie A, Gjyshi, Olsi, Cavett, Valerie, Nowak, Jason, Garcia-Ordonez, Ruben D, Houtman, René, Griffin, Patrick R, Kojetin, Douglas J, Katzenellenbogen, John A, Conkright, Michael D, Nettles, Kendall W
Published in eLife (25.04.2014)
Published in eLife (25.04.2014)
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Journal Article
Predictive features of ligand‐specific signaling through the estrogen receptor
Nwachukwu, Jerome C, Srinivasan, Sathish, Zheng, Yangfan, Wang, Song, Min, Jian, Dong, Chune, Liao, Zongquan, Nowak, Jason, Wright, Nicholas J, Houtman, René, Carlson, Kathryn E, Josan, Jatinder S, Elemento, Olivier, Katzenellenbogen, John A, Zhou, Hai‐Bing, Nettles, Kendall W
Published in Molecular systems biology (01.04.2016)
Published in Molecular systems biology (01.04.2016)
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Journal Article
Thiophene-Core Estrogen Receptor Ligands Having Superagonist Activity
Min, Jian, Wang, Pengcheng, Srinivasan, Sathish, Nwachukwu, Jerome C, Guo, Pu, Huang, Minjian, Carlson, Kathryn E, Katzenellenbogen, John A, Nettles, Kendall W, Zhou, Hai-Bing
Published in Journal of medicinal chemistry (25.04.2013)
Published in Journal of medicinal chemistry (25.04.2013)
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Journal Article
Structural Mechanisms of Allostery and Autoinhibition in JNK Family Kinases
Laughlin, John D., Nwachukwu, Jerome C., Figuera-Losada, Mariana, Cherry, Lisa, Nettles, Kendall W., LoGrasso, Philip V.
Published in Structure (London) (05.12.2012)
Published in Structure (London) (05.12.2012)
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Journal Article
Triaryl-Substituted Schiff Bases Are High-Affinity Subtype-Selective Ligands for the Estrogen Receptor
Liao, Zong-Quan, Dong, Chune, Carlson, Kathryn E, Srinivasan, Sathish, Nwachukwu, Jerome C, Chesnut, Robert W, Sharma, Abhishek, Nettles, Kendall W, Katzenellenbogen, John A, Zhou, Hai-Bing
Published in Journal of medicinal chemistry (24.04.2014)
Published in Journal of medicinal chemistry (24.04.2014)
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Journal Article
Regulation of Androgen Receptor-Mediated Transcription by RPB5 Binding Protein URI/RMP
Mita, Paolo, Savas, Jeffrey N., Djouder, Nabil, Yates, John R., Ha, Susan, Ruoff, Rachel, Schafler, Eric D., Nwachukwu, Jerome C., Tanese, Naoko, Cowan, Nicholas J., Zavadil, Jiri, Garabedian, Michael J., Logan, Susan K.
Published in Molecular and Cellular Biology (01.09.2011)
Published in Molecular and Cellular Biology (01.09.2011)
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Journal Article
Asymmetric allostery in estrogen receptor-α homodimers drives responses to the ensemble of estrogens in the hormonal milieu
Min, Charles K, Nwachukwu, Jerome C, Hou, Yingwei, Russo, Robin J, Papa, Alexandra, Min, Jian, Peng, Rouming, Kim, Sung Hoon, Ziegler, Yvonne, Rangarajan, Erumbi S, Izard, Tina, Katzenellenbogen, Benita S, Katzenellenbogen, John A, Nettles, Kendall W
Published in Proceedings of the National Academy of Sciences - PNAS (11.06.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (11.06.2024)
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Journal Article
Tethering not required: the glucocorticoid receptor binds directly to activator protein-1 recognition motifs to repress inflammatory genes
Weikum, Emily R, de Vera, Ian Mitchelle S, Nwachukwu, Jerome C, Hudson, William H, Nettles, Kendall W, Kojetin, Douglas J, Ortlund, Eric A
Published in Nucleic acids research (21.08.2017)
Published in Nucleic acids research (21.08.2017)
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Journal Article
Activation of Crtc2/Creb1 in skeletal muscle enhances weight loss during intermittent fasting
Bruno, Nelson E., Nwachukwu, Jerome C., Hughes, David C., Srinivasan, Sathish, Hawkins, Richard, Sturgill, David, Hager, Gordon L., Hurst, Stephen, Sheu, Shey‐Shing, Bodine, Sue C., Conkright, Michael D., Nettles, Kendall W.
Published in The FASEB journal (01.12.2021)
Published in The FASEB journal (01.12.2021)
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Journal Article
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors
Tinivella, Annachiara, Nwachukwu, Jerome C., Angeli, Andrea, Foschi, Francesca, Benatti, Anna Laura, Pinzi, Luca, Izard, Tina, Ferraroni, Marta, Erumbi, Rangarajan, Christodoulou, Michael S., Passarella, Daniele, Supuran, Claudiu T., Nettles, Kendall W., Rastelli, Giulio
Published in European journal of medicinal chemistry (15.01.2023)
Published in European journal of medicinal chemistry (15.01.2023)
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Journal Article
Dual-mechanism estrogen receptor inhibitors
Min, Jian, Nwachukwu, Jerome C, Min, Charles K, Njeri, Jacqline W, Srinivasan, Sathish, Rangarajan, Erumbi S, Nettles, Charles C, Sanabria Guillen, Valeria, Ziegler, Yvonne, Yan, Shunchao, Carlson, Kathryn E, Hou, Yingwei, Kim, Sung Hoon, Novick, Scott, Pascal, Bruce D, Houtman, Rene, Griffin, Patrick R, Izard, Tina, Katzenellenbogen, Benita S, Katzenellenbogen, John A, Nettles, Kendall W
Published in Proceedings of the National Academy of Sciences - PNAS (31.08.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (31.08.2021)
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Journal Article
Systems Structural Biology Analysis of Ligand Effects on ERα Predicts Cellular Response to Environmental Estrogens and Anti-hormone Therapies
Nwachukwu, Jerome C., Srinivasan, Sathish, Bruno, Nelson E., Nowak, Jason, Wright, Nicholas J., Minutolo, Filippo, Rangarajan, Erumbi S., Izard, Tina, Yao, Xin-Qui, Grant, Barry J., Kojetin, Douglas J., Elemento, Olivier, Katzenellenbogen, John A., Nettles, Kendall W.
Published in Cell chemical biology (19.01.2017)
Published in Cell chemical biology (19.01.2017)
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Journal Article
Creb coactivators direct anabolic responses and enhance performance of skeletal muscle
Bruno, Nelson E, Kelly, Kimberly A, Hawkins, Richard, Bramah-Lawani, Mariam, Amelio, Antonio L, Nwachukwu, Jerome C, Nettles, Kendall W, Conkright, Michael D
Published in The EMBO journal (02.05.2014)
Published in The EMBO journal (02.05.2014)
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Journal Article
Chemical systems biology reveals mechanisms of glucocorticoid receptor signaling
Bruno, Nelson E, Nwachukwu, Jerome C, Srinivasan, Sathish, Nettles, Charles C, Izard, Tina, Jin, Zhuang, Nowak, Jason, Cameron, Michael D, Boregowda, Siddaraju V, Phinney, Donald G, Elemento, Olivier, Liu, Xu, Ortlund, Eric A, Houtman, René, Stavreva, Diana A, Hager, Gordon L, Kamenecka, Theodore M, Kojetin, Douglas J, Nettles, Kendall W
Published in Nature chemical biology (01.03.2021)
Published in Nature chemical biology (01.03.2021)
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