Synthesis and Biological Evaluation of Derivatives of Indoline as Highly Potent Antioxidant and Anti-inflammatory Agents
Zeeli, Shani, Weill, Tehilla, Finkin-Groner, Efrat, Bejar, Corina, Melamed, Michal, Furman, Svetlana, Zhenin, Michael, Nudelman, Abraham, Weinstock, Marta
Published in Journal of medicinal chemistry (10.05.2018)
Published in Journal of medicinal chemistry (10.05.2018)
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Journal Article
Cardioprotection by AN-7, a prodrug of the histone deacetylase inhibitor butyric acid: Selective activity in hypoxic cardiomyocytes and cardiofibroblasts
Nudelman, Vadim, Zahalka, Muayad A., Nudelman, Abraham, Rephaeli, Ada, Kessler-Icekson, Gania
Published in European journal of pharmacology (05.09.2020)
Published in European journal of pharmacology (05.09.2020)
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Journal Article
Doxorubicin-DNA adducts induce a non-topoisomerase II-mediated form of cell death
SWIFT, Lonnie P, REPHAELI, Ada, NUDELMAN, Abraham, PHILLIPS, Don R, CUTTS, Suzanne M
Published in Cancer research (Chicago, Ill.) (01.05.2006)
Published in Cancer research (Chicago, Ill.) (01.05.2006)
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Synthesis and preliminary biological evaluation of gabactyzine, a benactyzine-GABA mutual prodrug, as an organophosphate antidote
Weitman, Michal, Eisenkraft, Arik, TaShma, Zeev, Makarovsky, Igor, Last, David, Daniels, Dianne, Guez, David, Shneor, Ran, Mardor, Yael, Nudelman, Abraham, Krivoy, Amir
Published in Scientific reports (27.10.2022)
Published in Scientific reports (27.10.2022)
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Journal Article
Valproic Acid Prodrug Affects Selective Markers, Augments Doxorubicin Anticancer Activity and Attenuates Its Toxicity in a Murine Model of Aggressive Breast Cancer
Tarasenko, Nataly, Wilner, Harel Josef, Nudelman, Abraham, Kessler-Icekson, Gania, Rephaeli, Ada
Published in Pharmaceuticals (Basel, Switzerland) (30.11.2021)
Published in Pharmaceuticals (Basel, Switzerland) (30.11.2021)
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Journal Article
NMR Chemical Shifts of Common Laboratory Solvents as Trace Impurities
Gottlieb, Hugo E, Kotlyar, Vadim, Nudelman, Abraham
Published in Journal of organic chemistry (17.10.1997)
Published in Journal of organic chemistry (17.10.1997)
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Journal Article
Activation of DNA damage response pathways as a consequence of anthracycline-DNA adduct formation
Forrest, Robert A., Swift, Lonnie P., Rephaeli, Ada, Nudelman, Abraham, Kimura, Ken-Ichi, Phillips, Don R., Cutts, Suzanne M.
Published in Biochemical pharmacology (15.06.2012)
Published in Biochemical pharmacology (15.06.2012)
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Journal Article
The Therapeutic Potential of AN-7, a Novel Histone Deacetylase Inhibitor, for Treatment of Mycosis Fungoides/Sezary Syndrome Alone or with Doxorubicin
Moyal, Lilach, Feldbaum, Nataly, Goldfeiz, Neta, Rephaeli, Ada, Nudelman, Abraham, Weitman, Michal, Tarasenko, Nataly, Gorovitz, Batia, Maron, Leah, Yehezkel, Shiran, Amitay-Laish, Iris, Lubin, Ido, Hodak, Emmilia
Published in PloS one (2016)
Published in PloS one (2016)
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Potential Therapeutic Advantages of Doxorubicin when Activated by Formaldehyde to Function as a DNA Adduct-Forming Agent
Cutts, Suzanne M, Rephaeli, Ada, Nudelman, Abraham, Ugarenko, Michal, Phillips, Don R
Published in Current topics in medicinal chemistry (08.05.2015)
Published in Current topics in medicinal chemistry (08.05.2015)
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Journal Article
Development of GSK's NMR guides – a tool to encourage the use of more sustainable solvents
Gottlieb, Hugo E, Graczyk-Millbrandt, Grazyna, Inglis, Graham GA, Nudelman, Abraham, Perez, David, Qian, Yanqiu, Shuster, Leanna E, Sneddon, Helen F, Upton, Richard J
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2016)
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2016)
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Journal Article
Synthesis and in vitro evaluation of anti-inflammatory activity of ester and amine derivatives of indoline in RAW 264.7 and peritoneal macrophages
Furman, Svetlana, Nissim-Bardugo, Elinor, Zeeli, Shani, Weitman, Michal, Nudelman, Abraham, Finkin-Groner, Efrat, Moradov, Dorit, Shifrin, Helena, Schorer-Apelbaum, Donna, Weinstock, Marta
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
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Journal Article
The power and potential of doxorubicin-DNA adducts
Cutts, Suzanne M, Nudelman, Abraham, Rephaeli, Ada, Phillips, Don R
Published in IUBMB life (01.03.2005)
Published in IUBMB life (01.03.2005)
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Effect of Histone Deacetylase Inhibitor, Butyroyloxymethyl-Diethyl Phosphate (AN-7), on Corneal Neovascularization in a Mouse Model
Schaap-Fogler, Michal, Bahar, Irit, Rephaeli, Ada, Dahbash, Mor, Nudelman, Abraham, Livny, Eitan, Barliya, Tilda, Nisgav, Yael, Livnat, Tami
Published in Journal of ocular pharmacology and therapeutics (01.07.2017)
Published in Journal of ocular pharmacology and therapeutics (01.07.2017)
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Journal Article
Disparate impact of butyroyloxymethyl diethylphosphate (AN-7), a histone deacetylase inhibitor, and doxorubicin in mice bearing a mammary tumor
Tarasenko, Nataly, Cutts, Suzanne M, Phillips, Don R, Inbal, Aida, Nudelman, Abraham, Kessler-Icekson, Gania, Rephaeli, Ada
Published in PloS one (23.02.2012)
Published in PloS one (23.02.2012)
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Journal Article
Butyric acid prodrugs are histone deacetylase inhibitors that show antineoplastic activity and radiosensitizing capacity in the treatment of malignant gliomas
Entin-Meer, Michal, Rephaeli, Ada, Yang, Xiaodong, Nudelman, Abraham, VandenBerg, Scott R, Haas-Kogan, Daphne Adele
Published in Molecular cancer therapeutics (01.12.2005)
Published in Molecular cancer therapeutics (01.12.2005)
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Journal Article
De Novo Parallel Design, Synthesis and Evaluation of Inhibitors against the Reverse Transcriptase of Human Immunodeficiency Virus Type-1 and Drug-Resistant Variants
Herschhorn, Alon, Lerman, Lena, Weitman, Michal, Gleenberg, Iris Oz, Nudelman, Abraham, Hizi, Amnon
Published in Journal of medicinal chemistry (17.05.2007)
Published in Journal of medicinal chemistry (17.05.2007)
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